For more information regarding the endpoints, refer to the 'ToxCast Endpoints' file on the
DOWNLOAD page.
ToxCast Endpoints for intended target type: RNA
Assay Name | Tissue | Target Gene ID | Target HGNC Symbol | Target UniProt ID | Response | AC50 value |
---|
LTEA_HepaRG_CYP2B6 | Liver | 1555 | CYP2B6 | P20813 | Activatory | 5.03 μM |
LTEA_HepaRG_CYP2C19 | Liver | 1557 | CYP2C19 | P33261 | Activatory | 9.15 μM |
LTEA_HepaRG_CYP3A7 | Liver | 1551 | CYP3A7 | P24462 | Activatory | 9.36 μM |
ToxCast Endpoints for intended target type: Protein
Assay Name | Tissue | Target Gene ID | Target HGNC Symbol | Target UniProt ID | Response | AC50 value |
---|
NVS_ADME_hCYP1A2 | | 1544 | CYP1A2 | P05177 | Loss | 7.21 μM |
NVS_ENZ_hBACE | | 23621 | BACE1 | P56817 | Loss | 1.18 μM |
NVS_ENZ_hMMP3 | | 4314 | MMP3 | P08254 | Loss | 5.24 μM |
ATG_M_19_CIS | Liver | | | | Inhibitory | 0.01 μM |
ATG_M_32_CIS | Liver | | | | Inhibitory | 0.01 μM |
ATG_NURR1_TRANS | Liver | 4929 | NR4A2 | P43354 | Gain | 159.91 μM |
BSK_3C_TissueFactor | Vascular | 2152 | F3 | P13726 | Inhibitory | 0.67 μM |
BSK_LPS_TNFa | Vascular | 7124 | TNF | P01375 | Activatory | 4.36 μM |
ATG_mPXR_XSP2 | Liver | 8856 | NR1I2 | O75469 | Gain | 7.91 μM |
TOX21_AR_LUC_MDAKB2_Antagonist_0.5nM_R1881 | Breast | 367 | AR | P10275 | Loss | 5.26 μM |
TOX21_p450_CYP2D6_Antagonist | | 1565 | CYP2D6 | P10635 | Loss | 0.00 μM |
TOX21_p450_CYP1A2_Antagonist | | 1544 | CYP1A2 | P05177 | Loss | 0.72 μM |
TOX21_AR_LUC_MDAKB2_Antagonist_0.5nM_R1881 | Breast | 367 | AR | P10275 | Loss | 5.59 μM |
TOX21_p450_CYP1A2_Antagonist | | 1544 | CYP1A2 | P05177 | Loss | 0.87 μM |
No ToxCast endpoints for intended target type: Molecular Messengers
ToxCast Endpoints for intended target type: Pathway
Assay Name | Tissue | Target Gene ID | Target HGNC Symbol | Target UniProt ID | Response | AC50 value |
---|
APR_HepG2_CellCycleArrest_72hr | Liver | | | | Inhibitory | 110.93 μM |
ToxCast Endpoints for intended target type: Cellular
Assay Name | Tissue | Response | AC50 value |
---|
ACEA_AR_antagonist_AUC_viability | Prostate | Loss | 8.92 μM |
No ToxCast endpoints for intended target type: Extracellular