For more information regarding the endpoints, refer to the 'ToxCast Endpoints' file on the
DOWNLOAD page.
No ToxCast endpoints for intended target type: RNA
ToxCast Endpoints for intended target type: Protein
Assay Name | Tissue | Target Gene ID | Target HGNC Symbol | Target UniProt ID | Response | AC50 value |
---|
ATG_Ahr_CIS | Liver | 196 | AHR | P35869 | Activatory | 56.56 μM |
ATG_PXR_TRANS | Liver | 8856 | NR1I2 | O75469 | Gain | 57.04 μM |
TOX21_TRHR_HEK293_Agonist | Kidney | 7201 | TRHR | | Gain | 0.26 μM |
TOX21_TRHR_HEK293_Antagonist | Kidney | 7201 | TRHR | | Loss | 1.26 μM |
TOX21_p450_CYP2C9_Antagonist | | 1559 | CYP2C9 | P11712 | Loss | 41.70 μM |
No ToxCast endpoints for intended target type: Molecular Messengers
ToxCast Endpoints for intended target type: Pathway
Assay Name | Tissue | Target Gene ID | Target HGNC Symbol | Target UniProt ID | Response | AC50 value |
---|
TOX21_ERb_BLA_Antagonist_ch1 | Kidney | | | | Gain | 55.61 μM |
TOX21_PR_BLA_Antagonist_ch1 | Kidney | | | | Gain | 53.28 μM |
ToxCast Endpoints for intended target type: Cellular
Assay Name | Tissue | Response | AC50 value |
---|
TOX21_AR_LUC_MDAKB2_Antagonist_0.5nM_R1881_viability | Breast | Loss | 45.24 μM |
TOX21_AR_LUC_MDAKB2_Agonist_3uM_Nilutamide_viability | Breast | Loss | 44.97 μM |
TOX21_RT_HEK293_FLO_00hr_viability | Kidney | Gain | 2.45 μM |
TOX21_RT_HEK293_FLO_24hr_viability | Kidney | Gain | 3.27 μM |
TOX21_RT_HEK293_FLO_32hr_viability | Kidney | Gain | 2.93 μM |
TOX21_RT_HEPG2_GLO_00hr_viability | Liver | Loss | 51.78 μM |
TOX21_CASP3_HEPG2_viability | Liver | Loss | 42.46 μM |
No ToxCast endpoints for intended target type: Extracellular