For more information regarding the endpoints, refer to the 'ToxCast Endpoints' file on the
DOWNLOAD page.
ToxCast Endpoints for intended target type: RNA
Assay Name | Tissue | Target Gene ID | Target HGNC Symbol | Target UniProt ID | Response | AC50 value |
---|
CLD_CYP1A2_24hr | Liver | 1544 | CYP1A2 | P05177 | Gain | 20.00 μM |
CLD_CYP2B6_24hr | Liver | 1555 | CYP2B6 | P20813 | Gain | 6.24 μM |
CLD_CYP1A1_48hr | Liver | 1543 | CYP1A1 | P04798 | Gain | 20.00 μM |
CLD_CYP1A2_48hr | Liver | 1544 | CYP1A2 | P05177 | Gain | 9.96 μM |
CLD_CYP2B6_48hr | Liver | 1555 | CYP2B6 | P20813 | Gain | 8.64 μM |
ToxCast Endpoints for intended target type: Protein
Assay Name | Tissue | Target Gene ID | Target HGNC Symbol | Target UniProt ID | Response | AC50 value |
---|
CCTE_GLTED_hTTR_0.125uM | | 7276 | TTR | | Loss | 14.18 μM |
NVS_ADME_hCYP19A1 | | 1588 | CYP19A1 | P11511 | Loss | 4.05 μM |
NVS_TR_hNET | | 6530 | SLC6A2 | P23975 | Loss | 15.03 μM |
ATG_ERE_CIS | Liver | 2099 | ESR1 | P03372 | Activatory | 13.14 μM |
ATG_PXRE_CIS | Liver | 8856 | NR1I2 | O75469 | Activatory | 13.48 μM |
BSK_LPS_PGE2 | Vascular | 5732 | PTGER2 | P43116 | Inhibitory | 4.65 μM |
BSK_LPS_TNFa | Vascular | 7124 | TNF | P01375 | Activatory | 14.77 μM |
TOX21_p450_CYP1A2_Antagonist | | 1544 | CYP1A2 | P05177 | Loss | 15.95 μM |
TOX21_p450_CYP1A2_Antagonist | | 1544 | CYP1A2 | P05177 | Loss | 17.74 μM |
No ToxCast endpoints for intended target type: Molecular Messengers
No ToxCast endpoints for intended target type: Pathway
ToxCast Endpoints for intended target type: Cellular
Assay Name | Tissue | Response | AC50 value |
---|
TOX21_MMP_rhodamine | Liver | Loss | 13.73 μM |
TOX21_MMP_ratio | Liver | Inhibitory | 11.80 μM |
No ToxCast endpoints for intended target type: Extracellular