For more information regarding the endpoints, refer to the 'ToxCast Endpoints' file on the
DOWNLOAD page.
No ToxCast endpoints for intended target type: RNA
ToxCast Endpoints for intended target type: Protein
Assay Name | Tissue | Target Gene ID | Target HGNC Symbol | Target UniProt ID | Response | AC50 value |
---|
ATG_Ahr_CIS | Liver | 196 | AHR | P35869 | Activatory | 32.98 μM |
ATG_ERE_CIS | Liver | 2099 | ESR1 | P03372 | Activatory | 66.84 μM |
ATG_NRF2_ARE_CIS | Liver | 4780 | NFE2L2 | Q16236 | Activatory | 36.63 μM |
BSK_BE3C_PAI1 | Lung | 5054 | SERPINE1 | P05121 | Inhibitory | 3.97 μM |
TOX21_AhR_LUC_Agonist | Liver | 196 | AHR | P35869 | Gain | 34.80 μM |
TOX21_p450_CYP3A4_Antagonist | | 1576 | CYP3A4 | P08684 | Loss | 62.34 μM |
TOX21_p450_CYP2C19_Antagonist | | 1557 | CYP2C19 | P33261 | Loss | 44.58 μM |
TOX21_p450_CYP2C9_Antagonist | | 1559 | CYP2C9 | P11712 | Loss | 24.19 μM |
TOX21_p450_CYP1A2_Antagonist | | 1544 | CYP1A2 | P05177 | Loss | 11.36 μM |
No ToxCast endpoints for intended target type: Molecular Messengers
No ToxCast endpoints for intended target type: Pathway
ToxCast Endpoints for intended target type: Cellular
Assay Name | Tissue | Response | AC50 value |
---|
BSK_3C_Proliferation | Vascular | Inhibitory | 5.46 μM |
BSK_hDFCGF_Proliferation | Skin | Inhibitory | 5.13 μM |
ACEA_ER_AUC_viability | Breast | Loss | 14.26 μM |
No ToxCast endpoints for intended target type: Extracellular