| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Polyunsaturated fatty acid 5-lipoxygenase | Homo sapiens | P09917 | | >40000 nM | | | BindingDB |
| Plasmodium falciparum | Plasmodium falciparum | | | = 21100.0 nM|= 8600.0 nM | | | NPASS |
| NON-PROTEIN TARGET | | | | = 13700.0 nM|= 36200.0 nM | | | NPASS |
| NIH3T3 | Mus musculus | | = 21100.0 nM|= 16600.0 nM | = 16600.0 nM|= 21400.0 nM|= 21100.0 nM | | | NPASS |
| Muscle glycogen phosphorylase | Homo sapiens | P11217 | | = 28000.0 nM | | | NPASS |
| MCF7 | Homo sapiens | | > 30000.0 nM|= 37200.0 nM|= 24400.0 nM | = 24400.0 nM|= 16600.0 nM|> 10000.0 nM|> 100000.0 nM | | | NPASS |
| Lu1 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| Prostaglandin G/H synthase 1 | Ovis aries | P05979 | | 42000 nM | | | BindingDB |
| NCI-N87 | Homo sapiens | | | > 10000.0 nM | | | NPASS |
| Prostaglandin G/H synthase 2 | Homo sapiens | P35354 | | >40000 nM | | | BindingDB |
| T-cell protein-tyrosine phosphatase | Homo sapiens | P17706 | | = 19470.0 nM | | | NPASS |
| Protease | Human immunodeficiency virus 1 | Q9YQ12 | | = 62700.0 nM | | | NPASS |
| Protein-tyrosine phosphatase 1B | Homo sapiens | P18031 | | = 5930.0 nM | | | NPASS |
| Protein-tyrosine phosphatase 1C | Homo sapiens | P29350 | | > 40000.0 nM | | | NPASS |
| Protein-tyrosine phosphatase 2C | Homo sapiens | Q06124 | | > 40000.0 nM | | | NPASS |
| Receptor-type tyrosine-protein phosphatase F | Homo sapiens | P10586 | | >4E4 nM | | | BindingDB |
| Receptor-type tyrosine-protein phosphatase F (LAR) | Homo sapiens | P10586 | | > 40000.0 nM | | | NPASS |
| Tyrosine-protein phosphatase non-receptor type 1 | Homo sapiens | P18031 | | 5.93E3 nM | | | BindingDB |
| Tyrosine-protein phosphatase non-receptor type 11 | Homo sapiens | Q06124 | | >4E4 nM | | | BindingDB |
| Tyrosine-protein phosphatase non-receptor type 2 | Homo sapiens | P17706 | | 1.947E4 nM | | | BindingDB |
| Tyrosine-protein phosphatase non-receptor type 6 | Homo sapiens | P29350 | | >4E4 nM | | | BindingDB |
| Protease | Human immunodeficiency virus 1 | | | 62700 nM | | | BindingDB |
| Liver glycogen phosphorylase | Rattus norvegicus | P09811 | | = 99000.0 nM | | | NPASS |
| Hypoxia-inducible factor prolyl hydroxylase | Homo sapiens | | > 50000.0 nM | | | | NPASS |
| HepG2 | Homo sapiens | | | = 99200.0 nM|> 10000.0 nM|> 100000.0 nM | | | NPASS |
| KB | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| 518A2 | Homo sapiens | | = 13700.0 nM | | | | NPASS |
| 8505C | Homo sapiens | | = 17000.0 nM | = 17000.0 nM | | | NPASS |
| A2780 | Homo sapiens | | = 19500.0 nM | = 19500.0 nM | | | NPASS |
| A549 | Homo sapiens | | = 23400.0 nM | = 23400.0 nM | | | NPASS |
| Acetylcholinesterase | Electrophorus electricus | O42275 | | | | >100000 nM|> 100000.0 nM | BindingDB, NPASS |
| Aldo-keto reductase family 1 member B10 | Homo sapiens | O60218 | | 630 nM|= 630.0 nM | | | BindingDB, NPASS |
| Aldose reductase | Homo sapiens | P15121 | | = 72000.0 nM | | | NPASS |
| Arachidonate 5-lipoxygenase | Homo sapiens | P09917 | | > 40000.0 nM | | | NPASS |
| B16-F10 | Mus musculus | | | = 36200.0 nM|> 10000.0 nM | | | NPASS |
| Aldo-keto reductase family 1 member B1 | Homo sapiens | P15121 | | 72000 nM | | | BindingDB |
| Cholinesterase | Equus caballus | P81908 | | | | >100000 nM|> 100000.0 nM | BindingDB, NPASS |
| Cyclooxygenase-1 | Ovis aries | P05979 | | = 42000.0 nM | | | NPASS |
| Cyclooxygenase-2 | Homo sapiens | P35354 | | > 40000.0 nM | | | NPASS |
| Egl nine homolog 1/Prolyl hydroxylase EGLN2/Prolyl hydroxylase EGLN3/Transmembrane prolyl 4-hydroxylase | Homo sapiens | Q96KS0|Q9GZT9|Q9H6Z9|Q9NXG6 | >50000 nM | | | | BindingDB |
| FaDu | Homo sapiens | | = 17000.0 nM | | | | NPASS |
| Glycogen phosphorylase, liver form | Rattus norvegicus | P09811 | | 99000 nM | | | BindingDB |
| Glycogen phosphorylase, muscle form | Homo sapiens | P11217 | | 28000 nM | | | BindingDB |
| Glycogen phosphorylase, muscle form | Oryctolagus cuniculus | P00489 | | 28000 nM|= 28000.0 nM|= 28183.83 nM | | | BindingDB, NPASS |
| BV-2 | Mus musculus | | | = 17800.0 nM | | | NPASS |
| HT-29 | Homo sapiens | | = 28800.0 nM | = 28800.0 nM|= 32200.0 nM|> 10000.0 nM | | | NPASS |