| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| HT-22 | Mus musculus | | > 100000.0 nM | | | | NPASS |
| HL-60 | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| HEK293 | Homo sapiens | | | > 15000000.0 nM | | | NPASS |
| Dihydroorotate dehydrogenase (fumarate) | Leishmamajor | Q4QEW7 | | = 922000.0 nM|= 1000000.0 nM | | | NPASS |
| Carbonic anhydrase XIV | Homo sapiens | Q9ULX7 | | | | = 690.0 nM | NPASS |
| Cyclooxygenase-2 | Homo sapiens | P35354 | | = 25400.0 nM | | | NPASS |
| Cathepsin L | Homo sapiens | P07711 | | > 59642.0 nM | | | NPASS |
| M18 aspartyl aminopeptidase | Plasmodium falciparum (isolate 3D7) | | | 479.4 nM | | | BindingDB |
| Dihydroorotate dehydrogenase (fumarate) | Leishmamajor | | | 922000 nM|1000000 nM | | | BindingDB |
| M18 aspartyl aminopeptidase | Plasmodium falciparum 3D7 | Q8I2J3 | | = 479.4 nM | | | NPASS |
| Tyrosinase | Agaricus bisporus | O42713 | | > 100000.0 nM | | | NPASS |
| NON-PROTEIN TARGET | | | = 2560.0 nM|= 4.0 ug.mL-1 | = 15700.0 nM|= 3310.0 nM|= 13.0 ug.mL-1|= 2.47 ug.mL-1 | | | NPASS |
| Plasmodium falciparum | Plasmodium falciparum | | | > 5.0 ug.mL-1 | | | NPASS |
| Polyphenol oxidase 2 | Agaricus bisporus | O42713 | | >100000 nM | | | BindingDB |
| Procathepsin L | Homo sapiens | P07711 | | >59642 nM | | | BindingDB |
| Prolyl 4-hydroxylase subunit alpha-1 | Gallus gallus | P16924 | | | | 5000 nM | BindingDB |
| Radical scavenging activity | | | = 2.1 ug.mL-1|= 8830.0 nM | = 77.63 ug.mL-1|= 6.9 ug.mL-1 | | | NPASS |
| SMMC-7721 | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| SW480 | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| Trypanosoma brucei rhodesiense | Trypanosoma brucei rhodesiense | | | = 111600.0 nM | | | NPASS |
| Carbonic anhydrase XII | Homo sapiens | O43570 | | | | = 4090.0 nM | NPASS |
| Xanthine dehydrogenase/oxidase | Bos taurus | P80457 | | 5.8e+3 nM | | | BindingDB |
| Meloidogyne incognita | Meloidogyne incognita | | > 1000.0 ug.mL-1 | | | | NPASS |
| Carbonic anhydrase VII | Homo sapiens | P43166 | | | | = 7870.0 nM | NPASS |
| Carbonic anhydrase I | Homo sapiens | P00915 | | | | = 1080.0 nM | NPASS |
| Carbonic anhydrase IX | Homo sapiens | Q16790 | | | | = 4450.0 nM | NPASS |
| 3-dehydroquinate synthase | Escherichia coli (strain K12) | P07639 | | | | 65000 nM|44000 nM | BindingDB |
| 3-dehydroquinate synthase | Escherichia coli K-12 | P07639 | | | | = 44000.0 nM|= 65000.0 nM | NPASS |
| A549 | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| Carbonic anhydrase VI | Homo sapiens | P23280 | | | | = 4720.0 nM | NPASS |
| Alpha-(1,3)-fucosyltransferase 7 | Homo sapiens | Q11130 | | 137000 nM | | | BindingDB |
| Alpha-glucosidase MAL12 | Saccharomyces cerevisiae | P53341 | | >3.00e+5 nM | | | BindingDB |
| Alpha-glucosidase MAL12 | Saccharomyces cerevisiae (strain ATCC 204508 / S288c) | P53341 | | 8.51e+4 nM | | | BindingDB |
| Anthrax toxin receptor 2 | Homo sapiens | P58335 | | >300000 nM|> 300000.0 nM | | | BindingDB, NPASS |
| BV-2 | Mus musculus | | | > 100000.0 nM | | | NPASS |
| Carbonic anhydrase | Dicentrarchus labrax | | | | | 3210 nM | BindingDB |
| Aldose reductase | Homo sapiens | P15121 | | = 42.7 ug.mL-1 | | | NPASS |
| Carbonic anhydrase 1 | Homo sapiens | P00915 | | | | 1080 nM | BindingDB |
| Carbonic anhydrase | Dicentrarchus labrax | Q2PCB5 | | | | = 3210.0 nM | NPASS |
| Carbonic anhydrase IV | Homo sapiens | P22748 | | | | = 2450.0 nM | NPASS |
| Carbonic anhydrase 9 | Homo sapiens | Q16790 | | | | 4450 nM | BindingDB |
| Carbonic anhydrase 7 | Homo sapiens | P43166 | | | | 7870 nM | BindingDB |
| Carbonic anhydrase II | Homo sapiens | P00918 | | | | = 470.0 nM | NPASS |
| Carbonic anhydrase 4 | Homo sapiens | P22748 | | | | 2450 nM | BindingDB |
| Carbonic anhydrase 2 | Homo sapiens | P00918 | | | | 470 nM | BindingDB |
| Carbonic anhydrase 14 | Homo sapiens | Q9ULX7 | | | | 690 nM | BindingDB |
| Carbonic anhydrase 12 | Homo sapiens | O43570 | | | | 4090 nM | BindingDB |
| Carbonic anhydrase 6 | Homo sapiens | P23280 | | | | 4720 nM | BindingDB |