| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| MCF7 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| NON-PROTEIN TARGET | | | > 50000.0 nM|= 13300.0 nM | = 220000.0 nM | | | NPASS |
| Polyunsaturated fatty acid 5-lipoxygenase | Homo sapiens | P09917 | | >40000 nM | | | BindingDB |
| Protein-tyrosine phosphatase 1B | Homo sapiens | P18031 | | = 19260.0 nM | | | NPASS |
| Lu1 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| Tyrosine-protein phosphatase non-receptor type 1 | Homo sapiens | P18031 | | 19260 nM | | | BindingDB |
| Tyrosine-protein phosphatase non-receptor type 1 [1-321] | Homo sapiens | P18031 | | | | 6000 nM | BindingDB |
| Tyrosine-protein phosphatase non-receptor type 1 [1-405] | Homo sapiens | P18031 | | | | 4000 nM | BindingDB |
| WI-38 VA13 | Homo sapiens | | | > 235000.0 nM | | | NPASS |
| Trypanosoma brucei brucei | Trypanosoma brucei brucei | | | = 114500.0 nM | | | NPASS |
| KB | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| DNA topoisomerase I | Homo sapiens | P11387 | | > 250000.0 nM | | | NPASS |
| HepG2 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| G-protein coupled bile acid receptor 1 | Homo sapiens | Q8TDU6 | >10000 nM|> 10000.0 nM | | | | BindingDB, NPASS |
| DNA topoisomerase II alpha | Homo sapiens | P11388 | | > 250000.0 nM | | | NPASS |
| DNA topoisomerase 2-alpha | Homo sapiens | P11388 | | >250000 nM | | | BindingDB |
| DNA topoisomerase 1 | Homo sapiens | P11387 | | >250000 nM | | | BindingDB |
| Bile acid receptor FXR | Homo sapiens | Q96RI1 | = 0.0 nM | | | | NPASS |
| B16 | Mus musculus | | | = 50000.0 nM | | | NPASS |
| Arachidonate 5-lipoxygenase | Homo sapiens | P09917 | | > 40000.0 nM | | | NPASS |
| A2780 | Homo sapiens | | | = 20.6 ug.mL-1 | | | NPASS |
| J774 | Mus musculus | | | = 128500.0 nM | | | NPASS |