| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| NON-PROTEIN TARGET | | | = 12000000.0 nM|= 105300.0 nM|= 31.01 ug.mL-1|= 134.1 ug.mL-1|= 122.0 ug.mL-1|= 149.7 ug.mL-1|= 44.18 ug.mL-1 | = 1130.0 nM|= 8660.0 nM|= 3750.0 nM|= 8.03 ug.mL-1|= 2.56 ug.mL-1|> 50.0 ug.mL-1|> 100000.0 nM | | | NPASS |
| NADPH oxidase 4 | Homo sapiens | Q9NPH5 | | 850 nM|= 850.0 nM | | | BindingDB, NPASS |
| NAD-dependent protein deacylase sirtuin-6 | Homo sapiens | Q8N6T7 | 270000 nM | 1900 nM | | | BindingDB |
| NAD-dependent protein deacetylase sirtuin-6 | Homo sapiens | Q8N6T7 | = 270000.0 nM | = 1900.0 nM | | | NPASS |
| Monoamine oxidase B | Homo sapiens | P27338 | | = 59700.0 nM | | | NPASS |
| Matrix metalloproteinase-9 | Homo sapiens | P14780 | | 5620 nM | | | BindingDB |
| Poly [ADP-ribose] polymerase 1 | Homo sapiens | P09874 | | 4200 nM | | | BindingDB |
| Mitogen-activated protein kinase 14 | Homo sapiens | Q16539 | | 1.80e+4 nM | | | BindingDB |
| Mitogen-activated protein kinase 10 | Homo sapiens | P53779 | | 2.3e+3 nM | | | BindingDB |
| Nakaseomyces glabratus | Nakaseomyces glabratus | | | = 15.0 ug.mL-1 | | | NPASS |
| Monoamine oxidase A | Homo sapiens | P21397 | | = 4900.0 nM | | | NPASS |
| Neuraminidase | InflueA virus | B4URF0 | | = 33700.0 nM|= 32600.0 nM|= 53300.0 nM|= 11000.0 nM | | = 19600.0 nM | NPASS |
| Nonstructural protein 3 | Zika virus | | | 53000 nM | | | BindingDB |
| Neuraminidase | InflueA virus (A/WSN/1933(H1N1)) | P03470 | | 32600 nM|53300 nM|33700 nM | | | BindingDB |
| Neuraminidase | InflueA virus (strain A/Puerto Rico/8/1934 H1N1) | P03468 | | 33800 nM|33700 nM | | | BindingDB |
| Neutrophil elastase | Homo sapiens | P08246 | | 12700 nM | | 10100 nM | BindingDB |
| Matrix metalloproteinase-2 | Homo sapiens | P08253 | | = 3610.0 nM|= 40900.0 nM | | | NPASS |
| Zinc finger protein mex-5 | Caenorhabditis elegans | Q9XUB2 | 31000 nM|= 31000.0 nM | | | | BindingDB, NPASS |
| P-glycoprotein 1 | Homo sapiens | P08183 | | = 19600.0 nM | | | NPASS |
| PC4 and SFRS1-interacting protein | Homo sapiens | O75475 | | 14730 nM|1059 nM | | | BindingDB |
| POsterior Segregation | Caenorhabditis elegans | | 60374 nM | | | | BindingDB |
| Peroxisome proliferator-activated receptor gamma | Mus musculus | P37238 | 2300 nM|= 2300.0 nM | | | | BindingDB, NPASS |
| Phenol oxidase | Plutella xylostella | B5U2Z5 | | = 470000.0 nM | | = 13110000.0 nM | NPASS |
| Plasmodium falciparum | Plasmodium falciparum | | | = 10700.0 nM|= 9600.0 nM | | | NPASS |
| Platelet | | | | = 43500.0 nM | | | NPASS |
| Neuraminidase | InflueA virus (A/Puerto Rico/8/1934(H1N1)) | P03468 | | = 9.65 ug.mL-1 | | | NPASS |
| Matrix metalloproteinase 9 | Homo sapiens | P14780 | | = 5620.0 nM | | | NPASS |
| LNCaP | Homo sapiens | | | = 5000.0 nM | | | NPASS |
| Matrix metalloproteinase 3 | Homo sapiens | P08254 | | = 16200.0 nM | | | NPASS |
| K562 | Homo sapiens | | | = 14650.0 nM | | | NPASS |
| KB | Homo sapiens | | | = 45300.0 nM | | | NPASS |
| L6 | Rattus norvegicus | | | = 9.4 ug.mL-1 | | | NPASS |
| L929 | Mus musculus | | > 250000.0 nM | | | | NPASS |
| Poly [ADP-ribose] polymerase tankyrase-1 | Homo sapiens | O95271 | | 2400 nM | | | BindingDB |
| Lactoylglutathione lyase | Homo sapiens | Q04760 | | 7700 nM | | | BindingDB |
| Large T antigen | Simian virus 40 | P03070 | 47930 nM | | | | BindingDB |
| Leishmania donovani | Leishmadonovani | | = 2800.0 nM | = 114300.0 nM|= 90900.0 nM|= 89000.0 nM|= 7700.0 nM|= 0.8 ug.mL-1 | | | NPASS |
| Leukocyte elastase | Homo sapiens | P08246 | | = 12700.0 nM | | = 10100.0 nM | NPASS |
| Liver | Rattus norvegicus | | | = 24660.0 nM | | | NPASS |
| Lu1 | Homo sapiens | | | = 40800.0 nM | | | NPASS |
| Lymphocyte differentiation antigen CD38 | Homo sapiens | P28907 | | = 8200.0 nM | | | NPASS |
| Lysosomal alpha-glucosidase | Homo sapiens | P10253 | | 20800 nM|= 5.96 ug.mL-1 | | | BindingDB, NPASS |
| M1 family aminopeptidase | Plasmodium falciparum (isolate FcB1 / Columbia) | O96935 | | 22860 nM | | | BindingDB |
| M1-family aminopeptidase | Plasmodium falciparum 3D7 | Q8IEK1 | | = 22860.0 nM | | | NPASS |
| MAP kinase signal-integrating kinase 2 | Homo sapiens | Q9HBH9 | | = 579.0 nM | | | NPASS |
| MAP kinase-interacting serine/threonine-protein kinase 1 | Homo sapiens | Q9BUB5 | | 179 nM | | | BindingDB |
| MAP kinase-interacting serine/threonine-protein kinase 2 | Homo sapiens | Q9HBH9 | | 579 nM | | | BindingDB |
| MAP kinase-interacting serine/threonine-protein kinase MNK1 | Homo sapiens | Q9BUB5 | | = 179.0 nM | | | NPASS |
| MCF7 | Homo sapiens | | | = 14300.0 ug.mL-1|= 9.5 ug.mL-1|= 44400.0 nM|= 5000.0 nM | | | NPASS |
| MDA-MB-231 | Homo sapiens | | | = 9.65 ug.mL-1|= 7290.0 nM | | | NPASS |
| METTL3/METTL14 | Homo sapiens | Q86U44|Q9HCE5 | | = 6230.0 nM | | | NPASS |
| MOLM-13 | Homo sapiens | | | = 4500.0 nM | | | NPASS |
| MV4-11 | Homo sapiens | | | = 3100.0 nM | | | NPASS |
| Macrophage metalloelastase | Homo sapiens | P39900 | | 980 nM | | | BindingDB |
| Matrix metalloproteinase 12 | Homo sapiens | P39900 | | = 980.0 nM | | | NPASS |
| Matrix metalloproteinase 13 | Homo sapiens | P45452 | | = 10050.0 nM|= 18300.0 nM | | | NPASS |
| Matrix metalloproteinase 7 | Homo sapiens | P09237 | | = 68200.0 nM | | | NPASS |
| Poly [ADP-ribose] polymerase tankyrase-2 | Homo sapiens | Q9H2K2 | | 1100 nM | | | BindingDB |
| Short transient receptor potential channel 5 | Homo sapiens | Q9UL62 | | >10000 nM|> 10000.0 nM | | | BindingDB, NPASS |
| Polyunsaturated fatty acid 5-lipoxygenase | Homo sapiens | P09917 | | 1600 nM | | | BindingDB |
| Spike glycoprotein [668-1255] | SARS-CoV | P59594 | 10600 nM | | | | BindingDB |
| Stromelysin-1 | Homo sapiens | P08254 | | 16200 nM | | | BindingDB |
| THP-1 | Homo sapiens | | | = 70000.0 nM | | | NPASS |
| Tankyrase-1 | Homo sapiens | O95271 | | = 2398.83 nM|= 2400.0 nM | | | NPASS |
| Tankyrase-2 | Homo sapiens | Q9H2K2 | | = 1071.52 nM|= 1100.0 nM | | | NPASS |
| Transthyretin | Homo sapiens | P02766 | | 7000 nM|= 6400.0 nM|= 7000.0 nM | 70 nM|= 70.0 nM | | BindingDB, NPASS |
| Trypanosoma brucei brucei | Trypanosoma brucei brucei | | | < 30000.0 nM | | | NPASS |
| Trypanosoma brucei rhodesiense | Trypanosoma brucei rhodesiense | | = 14100.0 nM | = 3.7 ug.mL-1 | | | NPASS |
| Trypanosoma cruzi | Trypanosoma cruzi | | | = 21.4 ug.mL-1 | | | NPASS |
| Trypsin I | Bos taurus | P00760 | | = 35300.0 nM | | | NPASS |
| Tyrosinase | Homo sapiens | P14679 | | 60000 nM|= 60000.0 nM|= 0.613 ug.mL-1 | | | BindingDB, NPASS |
| Tyrosine-protein kinase LCK | Homo sapiens | P06239 | | = 10.0 ug.mL-1 | | | NPASS |
| Spike glycoprotein | Severe acute respiratory syndrome coronavirus 2 | P0DTC2 | | = 10600.0 nM | | | NPASS |
| Tyrosine-protein kinase Lck | Homo sapiens | P06239 | | 34900 nM | | | BindingDB |
| Tyrosine-protein kinase YES | Homo sapiens | P07947 | | | | = 2380.0 nM | NPASS |
| Tyrosine-protein kinase Yes | Homo sapiens | P07947 | | | | 2380 nM | BindingDB |
| Tyrosine-protein kinase receptor FLT3 | Homo sapiens | P36888 | | = 830.0 nM | | | NPASS |
| U-937 | Homo sapiens | | | = 36000.0 nM|= 28000.0 nM|= 20000.0 nM | | | NPASS |
| Urease subunit alpha/Urease subunit beta | Helicobacter pylori (strain ATCC 700392 / 26695) (Campylobacterpylori) | | | = 35400.0 nM | | | NPASS |
| Urease subunit beta | Helicobacter pylori (strain ATCC 700392 / 26695) | P69996 | | 35400 nM | | | BindingDB |
| Verticillium dahliae | Verticillium dahliae | | | = 7.0 ug.mL-1 | | | NPASS |
| Xanthine dehydrogenase | Bos taurus | P80457 | | = 10200.0 nM | | = 1900.0 nM | NPASS |
| Xanthine dehydrogenase | Homo sapiens | P47989 | | = 550.0 nM|= 11540.0 nM|= 7800.0 nM | | = 2900.0 nM | NPASS |
| Xanthine dehydrogenase/oxidase | Bos taurus | P80457 | | 10200 nM | | 1900 nM | BindingDB |
| Xanthine dehydrogenase/oxidase | Homo sapiens | P47989 | | 7800 nM|11540 nM|550 nM | | 2900 nM | BindingDB |
| Interstitial collagenase [100-268] | Human | P03956 | | 3.03e+3 nM | | | BindingDB |
| Tyrosine-protein kinase SYK | Homo sapiens | P43405 | 4500 nM|= 4500.0 nM | 12000 nM|= 12000.0 nM | | | BindingDB, NPASS |
| Poly [ADP-ribose] polymerase-1 | Homo sapiens | P09874 | | = 4265.8 nM|= 4200.0 nM | | | NPASS |
| Solute carrier organic anion transporter family member 2B1 | Homo sapiens | O94956 | | = 3900.0 nM|= 3890.45 nM | | | NPASS |
| Solute carrier family 22 member 1 | Homo sapiens | O15245 | | = 46080.0 nM | | | NPASS |
| Polyunsaturated fatty acid lipoxygenase ALOX15 | Homo sapiens | P16050 | | 5000 nM | | | BindingDB |
| Prostaglandin G/H synthase 2 | Homo sapiens | P35354 | | 8730 nM|<349000 nM | | | BindingDB |
| Proteasome Macropain subunit MB1 | Homo sapiens | P28074 | | = 1300.0 nM|= 1500.0 nM | | | NPASS |
| Proteasome subunit beta type-5 | Homo sapiens | P28074 | | 1500 nM|1300 nM | | | BindingDB |
| Protein polybromo-1 | Homo sapiens | Q86U86 | | | 12900 nM|= 12900.0 nM | | BindingDB, NPASS |
| RAW264.7 | Mus musculus | | | = 7390.0 nM|= 7500.0 nM|= 10400.0 nM|= 43200.0 nM|= 210.0 nM|= 7200.0 nM|= 18950.0 nM|= 5060.0 nM|= 2870.0 nM|= 5600.0 nM|= 14400.0 nM|> 50000.0 nM|= 5800.0 nM|= 8100.0 nM|= 9200.0 nM|> 40000.0 nM | | | NPASS |
| RBL-2H3 | Rattus norvegicus | | | = 5800.0 nM|= 3700.0 nM|= 82000.0 nM|= 58200.0 nM | | | NPASS |
| Radical scavenging activity | | | = 6120.0 nM|= 44.18 ug.mL-1 | = 7.2 ug.mL-1|= 16180.0 nM|= 0.99 ug.mL-1 | | | NPASS |
| Receptor-type tyrosine-protein kinase FLT3 | Homo sapiens | P36888 | | 830 nM | | | BindingDB |
| Replicase polyprotein 1ab | Human SARS coronavirus | P0C6X7 | 10600 nM | 20000 nM | | | BindingDB |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome coronavirus | P0C6X7 | | 20000 nM | | | BindingDB |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome coronavirus 2 | P0DTD1 | = 10600.0 nM | 4600 nM|= 4600.0 nM | | | BindingDB, NPASS |
| Solute carrier family 22 member 2 | Homo sapiens | O15244 | | = 41030.0 nM | | | NPASS |
| Ribosomal protein S6 kinase alpha 3 | Homo sapiens | P51812 | | = 4420.0 nM | | | NPASS |
| SARS-CoV-2 | Severe acute respiratory syndrome coronavirus 2 | | | > 20000.0 nM|> 19952.62 nM | | | NPASS |
| SW1573 | Homo sapiens | | | > 10.0 ug.mL-1 | | | NPASS |
| Salivary alpha-amylase | Homo sapiens | P04745 | | = 18400.0 nM | | | NPASS |
| Seed linoleate 13S-lipoxygenase-1 | Glycine max | P08170 | | 3200 nM | | 121700 nM | BindingDB |
| Seed lipoxygenase-1 | Glycine max | P08170 | | = 3200.0 nM | | = 121700.0 nM | NPASS |
| Sensor protein kinase WalK family protein | Streptococcus pneumo PCS8203 | M5KM83 | | = 216000.0 nM | | | NPASS |
| Serine protease 1 | Bos taurus | P00760 | | 35300 nM | | | BindingDB |
| Serine/threonine-protein kinase pim-1 | Homo sapiens | P11309 | | 1600 nM|1585 nM | | | BindingDB |
| Sialidase | Clostridium perfringens | P10481 | | 4300 nM|= 4300.0 nM | | | BindingDB, NPASS |
| Sialidase 2 | Homo sapiens | Q9Y3R4 | | = 130000.0 nM | | | NPASS |
| Sialidase-2 | Homo sapiens | Q9Y3R4 | | 130000 nM | | | BindingDB |
| Sodium-dependent dopamine transporter | Rattus norvegicus | P23977 | 1450 nM | | | | BindingDB |
| SARS-CoV | Severe acute respiratory syndrome-related coronavirus | | = 10600.0 nM | | | | NPASS |
| Integrase | Human immunodeficiency virus 1 | | | 32900 nM|450 nM|>20000 nM|8900 nM|25000 nM | | | BindingDB |
| Cyclin-dependent kinase 5/CDK5 activator 1 | Homo sapiens | Q15078 | | = 3800.0 nM | | | NPASS |
| Inositol hexakisphosphate kinase 2 | Homo sapiens | Q9UHH9 | | 1300 nM|= 1300.0 nM | | | BindingDB, NPASS |
| Arachidonate 5-lipoxygenase | Homo sapiens | P09917 | | = 1600.0 nM | | | NPASS |
| Arginase-1 | Rattus norvegicus | P07824 | | = 9000.0 nM | | | NPASS |
| Aurora kinase B | Homo sapiens | Q96GD4 | | 3.88e+3 nM | | | BindingDB |
| Beta amyloid A4 protein | Homo sapiens | P05067 | | = 6400.0 nM | | | NPASS |
| Beta-secretase 1 | Homo sapiens | P56817 | | = 520.0 nM | | | NPASS |
| Brain | Rattus norvegicus | | = 79000.0 nM | | | | NPASS |
| Broad substrate specificity ATP-binding cassette transporter ABCG2 | Homo sapiens | Q9UNQ0 | | 8900 nM | | | BindingDB |
| Butyrylcholinesterase | Homo sapiens | P06276 | | | | = 166100.0 nM | NPASS |
| CCRF-CEM | Homo sapiens | | | > 10.0 ug.mL-1 | | | NPASS |
| Ca9-22 | Homo sapiens | | | = 8.55 ug.mL-1 | | | NPASS |
| Candida albicans | Candida albicans | | | > 50.0 ug.mL-1 | | | NPASS |
| Carbonic anhydrase 1 | Homo sapiens | P00915 | | | | 2200 nM|>10000 nM | BindingDB |
| Carbonic anhydrase 12 | Homo sapiens | O43570 | | | | 60 nM | BindingDB |
| Carbonic anhydrase 2 | Homo sapiens | P00918 | | | | 740 nM|3692 nM | BindingDB |
| Carbonic anhydrase 3 | Bovine | Q3SZX4 | | | | 5400 nM | BindingDB |
| Carbonic anhydrase 4 | Homo sapiens | P22748 | | | | 4400 nM|293 nM | BindingDB |
| Carbonic anhydrase 7 | Homo sapiens | P43166 | | | | 4.7 nM | BindingDB |
| Carbonic anhydrase I | Homo sapiens | P00915 | | | | > 10000.0 nM | NPASS |
| Carbonic anhydrase II | Homo sapiens | P00918 | | | | = 3691.6 nM | NPASS |
| Carbonic anhydrase IV | Homo sapiens | P22748 | | | | = 293.0 nM | NPASS |
| Carbonic anhydrase VII | Homo sapiens | P43166 | | | | = 4.7 nM | NPASS |
| Carbonic anhydrase XII | Homo sapiens | O43570 | | | | = 60.3 nM | NPASS |
| Casein kinase 2 | Homo sapiens | | | = 500.0 nM | | = 240.0 nM | NPASS |
| Casein kinase 2 | Rattus norvegicus | | | = 500.0 nM | | | NPASS |
| Casein kinase II | Homo sapiens | P19784 | | < 1000.0 nM | | | NPASS |
| Arachidonate 15-lipoxygenase | Homo sapiens | P16050 | | = 5000.0 nM | | | NPASS |
| Aorta | Rattus norvegicus | | | = 156000.0 nM|= 72000.0 nM|= 68000.0 nM | | | NPASS |
| Angiotensin-converting enzyme | Oryctolagus cuniculus | P12822 | | 290000 nM|= 290000.0 nM | | | BindingDB, NPASS |
| Amyloid-beta precursor protein | Homo sapiens | P05067 | | 6400 nM | | | BindingDB |
| 1-deoxy-D-xylulose 5-phosphate reductoisomerase | Escherichia coli (strain K12) | P45568 | | 3.4e+3 nM | | | BindingDB |
| 3-hydroxyacyl-[acyl-carrier-protein] dehydratase | Plasmodium falciparum | | | 5000 nM | | 11500 nM | BindingDB |
| 3-oxoacyl-acyl-carrier protein reductase | Plasmodium falciparum | | | 4000 nM | | 1800 nM|800 nM | BindingDB |
| 3-oxoacyl-acyl-carrier protein reductase | Plasmodium falciparum | Q965D6 | | = 4000.0 nM | | = 1800.0 nM|= 800.0 nM | NPASS |
| Inositol polyphosphate multikinase | Homo sapiens | Q8NFU5 | | 5500 nM|= 5500.0 nM | | | BindingDB, NPASS |
| A549 | Homo sapiens | | | = 12900.0 ug.mL-1|= 10.23 ug.mL-1 | | | NPASS |
| ADAMTS4 | Homo sapiens | O75173 | | = 9800.0 nM | | | NPASS |
| ADAMTS5 | Homo sapiens | Q9UNA0 | | = 12200.0 nM | | | NPASS |
| ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1 | Homo sapiens | P28907 | | 8200 nM | | | BindingDB |
| ATP-binding cassette sub-family G member 2 | Homo sapiens | Q9UNQ0 | | = 8900.0 nM | | | NPASS |
| ATP-dependent translocase ABCB1 | Homo sapiens | P08183 | | 19600 nM | | | BindingDB |
| Acetylcholinesterase | Homo sapiens | P22303 | | | | 65800 nM|= 65800.0 nM | BindingDB, NPASS |
| Casein kinase II subunit alpha 3 | Homo sapiens | Q8NEV1 | | 500 nM | | | BindingDB |
| Adenosine A1 receptor | Rattus norvegicus | P25099 | | | | = 1660.0 nM|= 1550.0 nM | NPASS |
| Aldo-keto reductase family 1 member B1 | Homo sapiens | P15121 | | 600 nM|3200 nM | | | BindingDB |
| Aldo-keto reductase family 1 member B1 | Rattus norvegicus | P07943 | | 1540 nM | | | BindingDB |
| Aldo-keto reductase family 1 member B1 [K65Q] | Bos taurus | P16116 | | 9570 nM|754 nM | | | BindingDB |
| Aldo-keto reductase family 1 member B10 | Homo sapiens | O60218 | | 107800 nM|9200 nM|= 107800.0 nM|= 9200.0 nM | | | BindingDB, NPASS |
| Aldose reductase | Bos taurus | P16116 | | = 9570.0 nM|= 754.0 nM | | | NPASS |
| Aldose reductase | Homo sapiens | P15121 | | = 600.0 nM|= 3200.0 nM | | | NPASS |
| Aldose reductase | Rattus norvegicus | P07943 | | = 1540.0 nM | | | NPASS |
| Alpha-amylase 1A | Homo sapiens | P0DUB6 | | 18400 nM | | | BindingDB |
| Alpha-glucosidase MAL62 | Saccharomyces cerevisiae | P07265 | | 20989 nM | | | BindingDB |
| Alpha-synuclein | Homo sapiens | P37840 | | 28000 nM|= 28000.0 nM | | | BindingDB, NPASS |
| Amine oxidase [flavin-containing] A | Homo sapiens | P21397 | | 4900 nM | | | BindingDB |
| Amine oxidase [flavin-containing] B | Homo sapiens | P27338 | | 59700 nM | | | BindingDB |
| Adenosine receptor A1 | Rattus norvegicus | P25099 | | | | 1660 nM|1550 nM | BindingDB |
| Cell division protein kinase 5 | Rattus norvegicus | Q03114 | > 250000.0 nM | | | | NPASS |
| 72 kDa type IV collagenase | Homo sapiens | P08253 | | 3610 nM | | | BindingDB |
| Chikungunya virus | Chikunguvirus | | | = 22500.0 nM | | | NPASS |
| Fatty acid synthase | Chicken | P12276 | | 6.25e+4 nM | | | BindingDB |
| Fatty acid synthase | Homo sapiens | P49327 | | 62500 nM|= 62500.0 nM | | | BindingDB, NPASS |
| Fatty acid synthase | Plasmodium falciparum | Q965D7 | | = 5000.0 nM | | = 11500.0 nM | NPASS |
| Filobasidiella neoformans | Cryptococcus neoformans | | | > 50.0 ug.mL-1 | | | NPASS |
| G-protein coupled receptor 35 | Homo sapiens | Q9HC97 | 7240 nM|3200 nM|= 7240.0 nM|= 3200.0 nM | 18600 nM|= 18600.0 nM | | | BindingDB, NPASS |
| GATA4/NKX2-5 | Mus musculus | | | = 22000.0 nM | | | NPASS |
| Genome polyprotein | Zika virus | A0A024AXB9 | | = 53000.0 nM | | | NPASS |
| Glycogen synthase kinase-3 | Homo sapiens | P49841 | | = 800.0 nM | | | NPASS |
| Glycogen synthase kinase-3 beta | Homo sapiens | P49841 | 3812 nM | 1500 nM|= 1500.0 nM | | | BindingDB, NPASS |
| Glycogen synthase kinase-3 beta | Rattus norvegicus | P18266 | | 800 nM | | | BindingDB |
| Glyoxalase I | Homo sapiens | Q04760 | | = 7700.0 nM | | | NPASS |
| H9 | Homo sapiens | | | = 16000.0 nM | | | NPASS |
| Entamoeba histolytica | Eoeba histolytica | | | = 17.8 ug.mL-1 | | | NPASS |
| H9c2 | Rattus norvegicus | | = 5530.0 nM | | | | NPASS |
| HeLa | Homo sapiens | | | = 16254.0 nM | | | NPASS |
| HepG2 | Homo sapiens | | | = 7.36 ug.mL-1|= 71200.0 nM|= 80800.0 nM|= 34700.0 nM|= 47300.0 nM | | | NPASS |
| Hepatitis C virus | Hepatitis C virus | | = 4700.0 nM|= 6600.0 nM | = 1120.0 nM | | | NPASS |
| Histidine kinase | Streptococcus pneumo PCS8203 | | | 216000 nM | | | BindingDB |
| Histone deacetylase 6 | Homo sapiens | Q9UBN7 | | = 1438.0 nM | | | NPASS |
| Histone-lysine N-methyltransferase SETD7 | Homo sapiens | Q8WTS6 | | 6080 nM|= 6080.0 nM | | | BindingDB, NPASS |
| Homeobox protein Nkx-2.5/Transcription factor GATA-4 | Mus musculus | P42582|Q08369 | | 22000 nM | | | BindingDB |
| Human immunodeficiency virus 1 | Human immunodeficiency virus 1 | | = 10000.0 nM|= 2.48 ug.mL-1 | | | | NPASS |
| Human immunodeficiency virus type 1 integrase | Human immunodeficiency virus 1 | Q7ZJM1 | | = 32900.0 nM|= 25000.0 nM|> 20000.0 nM|= 8900.0 nM|= 450.0 nM | | | NPASS |
| Influenza A virus | InflueA virus | | = 103100.0 nM | = 6820.0 nM | | | NPASS |
| Influenza A virus (A/PR/8/34(H1N1)) | InflueA virus (A/Puerto Rico/8/1934(H1N1)) | | = 84000.0 nM | | | | NPASS |
| Chemotaxis protein CheA | Escherichia coli (strain K12) | P07363 | | 111000 nM|= 111000.0 nM | | | BindingDB, NPASS |
| HL-60 | Homo sapiens | | | = 12.1 ug.mL-1|> 10.0 ug.mL-1 | | | NPASS |
| Enoyl-acyl-carrier protein reductase | Plasmodium falciparum | Q965D5 | | = 2000.0 nM | | = 2100.0 nM | NPASS |
| HT-29 | Homo sapiens | | | = 45000.0 nM | | | NPASS |
| Enoyl-[acyl-carrier-protein] reductase [NADH] FabI | Escherichia coli (strain K12) | P0AEK4 | | | | 7050 nM | BindingDB |
| Cholinesterase | Homo sapiens | P06276 | | | | 166100 nM | BindingDB |
| Enoyl-acyl-carrier protein reductase | Plasmodium falciparum | | | 2000 nM | | 2100 nM | BindingDB |
| Collagenase 3 | Homo sapiens | P45452 | | 10050 nM | | | BindingDB |
| Cruzipain | Trypanosoma cruzi | P25779 | | 155700 nM|27300 nM|= 155700.0 nM|= 27300.0 nM | | | BindingDB, NPASS |
| Cyclin homolog/dependent kinase 6 | Saimiriine herpesvirus 2 (strain 11) | Q00534|Q01043 | | >300000 nM | | | BindingDB |
| Cyclin-dependent kinase 1/G2/mitotic-specific cyclin-B | Marthasterias glacialis | P15206|Q9DGD3 | | 6200 nM | | | BindingDB |
| Cyclin-dependent kinase 1/cyclin B | Homo sapiens | O95067 | | = 6200.0 nM | | | NPASS |
| Cyclin-dependent kinase 5 | Rattus norvegicus | Q03114 | >250000 nM | | | | BindingDB |
| Cyclin-dependent kinase 5 activator 1 [99-307] | Homo sapiens | Q00535|Q15078 | | 3800 nM | | | BindingDB |
| Cyclin-dependent kinase 6 | Homo sapiens | Q00534 | | >300000 nM|> 300000.0 nM | | | BindingDB, NPASS |
| Cyclooxygenase-2 | Homo sapiens | P35354 | | < 100.0 ug.mL-1|= 2.5 ug.mL-1 | | | NPASS |
| Cytochrome P450 19A1 | Homo sapiens | P11511 | | = 1199.5 nM | | | NPASS |
| Cytochrome P450 1A1 | Homo sapiens | P04798 | | 1249 nM|= 1249.0 nM | | 890 nM|2400 nM|= 890.0 nM|= 2400.0 nM | BindingDB, NPASS |
| Cyclin-dependent kinase 2 | Homo sapiens | P24941 | | 20000 nM|= 20000.0 nM | | | BindingDB, NPASS |
| Dipeptidyl peptidase 3 | Homo sapiens | Q9NY33 | | 2.20e+4 nM | | | BindingDB |
| Dopamine transporter | Rattus norvegicus | P23977 | = 1450.0 nM | | | | NPASS |
| Cytochrome P450 1A2 | Homo sapiens | P05177 | | 3370 nM|= 3370.0 nM | | | BindingDB, NPASS |
| Dipeptidyl peptidase IV | Homo sapiens | P27487 | | = 120.0 nM | | | NPASS |
| Dipeptidyl peptidase 4 | Homo sapiens | P27487 | | 120 nM | | | BindingDB |
| Death-associated protein kinase 1 | Homo sapiens | P53355 | | 21000 nM|= 21000.0 nM | | | BindingDB, NPASS |
| DNA topoisomerase 1 | Rattus norvegicus | Q9WUL0 | | 660 nM|5000 nM|= 660.0 nM|= 5000.0 nM | | | BindingDB, NPASS |
| Enoyl-[acyl-carrier-protein] reductase | Escherichia coli K-12 | P0AEK4 | | | | = 7050.0 nM | NPASS |
| DNA polymerase eta | Homo sapiens | Q9Y253 | | = 12700.0 nM | | | NPASS |
| Cytosol aminopeptidase [33-68,L62W] | Sus scrofa | P28839 | | 49600 nM | | | BindingDB |
| Cytosol aminopeptidase | Sus scrofa | P28839 | | = 49600.0 nM | | | NPASS |
| Cytoplasmic zinc-finger protein | Caenorhabditis elegans | G5EF15 | = 60374.0 nM | | | | NPASS |
| Cytochrome P450 1B1 | Homo sapiens | Q16678 | | 79 nM|360 nM|= 79.0 nM|= 360.0 nM | | 56 nM|= 56.0 nM | BindingDB, NPASS |