| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| NON-PROTEIN TARGET | | | = 84480.0 nM | = 1840.0 nM | | | NPASS |
| Oryctolagus cuniculus | Oryctolagus cuniculus | | = 2000.0 nM | | | | NPASS |
| Mitogen-activated protein kinase 14 | Homo sapiens | Q16539 | | 2.70e+3 nM | | | BindingDB |
| L6 | Rattus norvegicus | | | = 38.5 ug.mL-1 | | | NPASS |
| Mitogen-activated protein kinase 10 | Homo sapiens | P53779 | | 2.6e+3 nM | | | BindingDB |
| MCF-10A | Homo sapiens | | | = 2440.0 nM | | | NPASS |
| Leishmania donovani | Leishmadonovani | | | = 0.6 ug.mL-1 | | | NPASS |
| Lactoylglutathione lyase | Homo sapiens | Q04760 | | | | 13200 nM | BindingDB |
| LNCaP | Homo sapiens | | | = 34100.0 nM | | | NPASS |
| HepG2 | Homo sapiens | | | > 400000.0 nM | | | NPASS |
| Human immunodeficiency virus type 1 integrase | Human immunodeficiency virus 1 | Q7ZJM1 | | = 28400.0 nM|= 8500.0 nM | | | NPASS |
| Human immunodeficiency virus 1 | Human immunodeficiency virus 1 | | < 100000.0 nM|= 122000.0 nM | | | | NPASS |
| Histone deacetylase 6 | Homo sapiens | Q9UBN7 | | = 2308.0 nM | | | NPASS |
| HT-22 | Mus musculus | | = 2800.0 nM|= 3000.0 nM | | | | NPASS |
| H9 | Homo sapiens | | | = 157000.0 nM | | | NPASS |
| Glyoxalase I | Homo sapiens | Q04760 | | | | = 13182.57 nM | NPASS |
| PC-3 | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| Glycogen synthase kinase-3 beta | Rattus norvegicus | P18266 | | 420 nM | | | BindingDB |
| Glycogen synthase kinase-3 | Homo sapiens | P49841 | | = 420.0 nM | | | NPASS |
| Integrase | Human immunodeficiency virus 1 | | | 8500 nM|28400 nM | | | BindingDB |
| PWR-1E | Homo sapiens | | | = 5390.0 nM | | | NPASS |
| Serine/threonine-protein kinase pim-1 | Homo sapiens | P11309 | | 850 nM|851 nM | | | BindingDB |
| Polyunsaturated fatty acid lipoxygenase ALOX12 | Homo sapiens | P18054 | | 950 nM | | | BindingDB |
| Xanthine dehydrogenase/oxidase | Homo sapiens | P47989 | | 4330 nM | | | BindingDB |
| Filobasidiella neoformans | Cryptococcus neoformans | | | > 50.0 ug.mL-1 | | | NPASS |
| Xanthine dehydrogenase | Homo sapiens | P47989 | | = 4330.0 nM | | | NPASS |
| Tyrosine-protein kinase SYK | Homo sapiens | P43405 | 19000 nM|= 19000.0 nM | 15000 nM|= 15000.0 nM | | | BindingDB, NPASS |
| Tyrosine-protein kinase Lck | Homo sapiens | P06239 | | 13900 nM | | | BindingDB |
| Tyrosine-protein kinase LCK | Homo sapiens | P06239 | | = 4.0 ug.mL-1 | | | NPASS |
| Trypanosoma cruzi | Trypanosoma cruzi | | | > 30.0 ug.mL-1 | | | NPASS |
| Trypanosoma brucei rhodesiense | Trypanosoma brucei rhodesiense | | | = 3.3 ug.mL-1 | | | NPASS |
| THP-1 | Homo sapiens | | | = 30000.0 nM | | | NPASS |
| Plasmodium falciparum | Plasmodium falciparum | | | = 8200.0 nM|= 6500.0 nM | | | NPASS |
| Solute carrier organic anion transporter family member 2B1 | Homo sapiens | O94956 | | = 6700.0 nM|= 6760.83 nM | | | NPASS |
| Ribosomal protein S6 kinase alpha 3 | Homo sapiens | P51812 | | = 2780.0 nM | | | NPASS |
| Ribosomal protein S6 kinase alpha 2 | Homo sapiens | Q15349 | | = 891.0 nM | | | NPASS |
| Ribosomal protein S6 kinase alpha 1 | Homo sapiens | Q15418 | | = 3790.0 nM | | | NPASS |
| Rattus norvegicus | Rattus norvegicus | | | = 200.0 nM | | | NPASS |
| Radical scavenging activity | | | | = 9.26 ug.mL-1 | | | NPASS |
| Pyruvate kinase isozymes M1/M2 | Homo sapiens | P14618 | | = 900.0 nM | | | NPASS |
| Pyruvate kinase PKM | Homo sapiens | P14618 | | 900 nM | | | BindingDB |
| Polyunsaturated fatty acid lipoxygenase ALOX15B | Homo sapiens | O15296 | | >100000 nM | | | BindingDB |
| Polyunsaturated fatty acid lipoxygenase ALOX15 | Homo sapiens | P16050 | | 1400 nM | | | BindingDB |
| Salivary alpha-amylase | Homo sapiens | P04745 | | = 19600.0 nM | | | NPASS |
| Fatty acid synthase | Plasmodium falciparum | Q965D7 | | = 2000.0 nM | | | NPASS |
| Cruzipain | Trypanosoma cruzi | P25779 | | 30000 nM|>60000 nM|= 30000.0 nM|> 60000.0 nM | | | BindingDB, NPASS |
| Enoyl-acyl-carrier protein reductase | Plasmodium falciparum | Q965D5 | | = 1000.0 nM | | | NPASS |
| Casein kinase 2 | Homo sapiens | | | = 350.0 nM | | | NPASS |
| Candida albicans | Candida albicans | | | > 50.0 ug.mL-1 | | | NPASS |
| CWR22R | Homo sapiens | | | = 25900.0 nM | | | NPASS |
| Butyrylcholinesterase | Homo sapiens | P06276 | | | | = 90000.0 nM | NPASS |
| BV-2 | Mus musculus | | | = 73020.0 nM|= 13500.0 nM | | | NPASS |
| Aurora kinase B | Homo sapiens | Q96GD4 | | 2.63e+3 nM | | | BindingDB |
| Entamoeba histolytica | Eoeba histolytica | | | = 189.01 ug.mL-1 | | | NPASS |
| Arachidonate 15-lipoxygenase, type II | Homo sapiens | O15296 | | > 100000.0 nM | | | NPASS |
| Arachidonate 15-lipoxygenase | Homo sapiens | P16050 | | = 1400.0 nM | | | NPASS |
| Arachidonate 12-lipoxygenase | Homo sapiens | P18054 | | = 950.0 nM | | | NPASS |
| Amyloid-beta A4 protein | Homo sapiens | P05067 | | = 12500.0 nM | | | NPASS |
| Alpha-glucosidase MAL62 | Saccharomyces cerevisiae | P07265 | | 13002 nM | | | BindingDB |
| Alpha-amylase 1A | Homo sapiens | P0DUB6 | | 19600 nM | | | BindingDB |
| Acetylcholinesterase | Homo sapiens | P22303 | | 12 nM|= 12.0 nM | | 100200 nM|= 100200.0 nM | BindingDB, NPASS |
| 3-oxoacyl-acyl-carrier protein reductase | Plasmodium falciparum | Q965D6 | | = 4100.0 nM | | | NPASS |
| 3-oxoacyl-acyl-carrier protein reductase | Plasmodium falciparum | | | 4100 nM | | | BindingDB |
| 3-hydroxyacyl-[acyl-carrier-protein] dehydratase | Plasmodium falciparum | | | 2000 nM | | | BindingDB |
| 17-beta-hydroxysteroid dehydrogenase type 3 | Homo sapiens | P37058 | | 3.24e+4 nM | | | BindingDB |
| 1-deoxy-D-xylulose 5-phosphate reductoisomerase | Escherichia coli (strain K12) | P45568 | | 3.5e+3 nM | | | BindingDB |
| Casein kinase 2 | Rattus norvegicus | | | = 350.0 nM | | | NPASS |
| Casein kinase II | Homo sapiens | P19784 | | = 350.0 nM|< 1000.0 nM | | = 170.0 nM | NPASS |
| Arginase-1 | Rattus norvegicus | P07824 | | = 1400.0 nM | | | NPASS |
| Casein kinase II subunit alpha | Homo sapiens | P68400 | | | | 350 nM | BindingDB |
| Casein kinase II alpha | Homo sapiens | P68400 | | | | = 350.0 nM | NPASS |
| Endoribonuclease toxin MazF | Escherichia coli (strain K12) | P0AE70 | >99000 nM | | | | BindingDB |
| Dipeptidyl peptidase 3 | Homo sapiens | Q9NY33 | | 2.49e+4 nM | | | BindingDB |
| Dengue virus 2 | Dengue virus 2 | | | = 55.0 ug.mL-1 | | | NPASS |
| DU-145 | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| DNA topoisomerase II alpha | Homo sapiens | P11388 | | = 8.2 ug.mL-1 | | | NPASS |
| DNA topoisomerase 2-alpha | Homo sapiens | P11388 | | 28600 nM | | | BindingDB |
| DNA gyrase A/A/B/B tetramer | Escherichia coli (strain K12) | P0AES4|P0AES6 | | 289000 nM | | | BindingDB |
| DNA gyrase | Escherichia coli K-12 | P0AES4 | | = 83.3 ug.mL-1 | | | NPASS |
| Enoyl-acyl-carrier protein reductase | Plasmodium falciparum | | | 1000 nM | | | BindingDB |
| Cyclin-dependent kinase 5/CDK5 activator 1 | Homo sapiens | Q15078 | | = 570.0 nM | | | NPASS |
| Cyclin-dependent kinase 6 | Homo sapiens | Q00534 | | 850 nM|= 850.0 nM | | | BindingDB, NPASS |
| Chikungunya virus | Chikunguvirus | | | = 29500.0 nM | | | NPASS |
| Cholinesterase | Homo sapiens | P06276 | | | | 90000 nM | BindingDB |
| Cyclin homolog/dependent kinase 6 | Saimiriine herpesvirus 2 (strain 11) | Q00534|Q01043 | | 850 nM | | | BindingDB |
| Casein kinase II subunit alpha 3 | Homo sapiens | Q8NEV1 | | 350 nM | | | BindingDB |
| Cyclin-dependent kinase 1/cyclin B | Homo sapiens | O95067 | | = 790.0 nM | | | NPASS |
| Cyclin-dependent kinase 2 | Homo sapiens | P24941 | | 5000 nM|= 5000.0 nM | | | BindingDB, NPASS |
| Cyclin-dependent kinase 5 activator 1 [99-307] | Homo sapiens | Q00535|Q15078 | | 570 nM | | | BindingDB |
| Cyclin-dependent kinase 1/G2/mitotic-specific cyclin-B | Marthasterias glacialis | P15206|Q9DGD3 | | 790 nM | | | BindingDB |