| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Pancreatic alpha-amylase | Sus scrofa | P00690 | | >200000 nM|> 200000.0 nM | | | BindingDB, NPASS |
| PC-3 | Homo sapiens | | | > 250000.0 nM|= 17900.0 nM|= 22400.0 nM | | | NPASS |
| OVCAR-3 | Homo sapiens | | | > 10000.0 nM | | | NPASS |
| Nuclear factor NF-kappa-B p65 subunit | Homo sapiens | Q04206 | | = 8800.0 nM | | | NPASS |
| NON-PROTEIN TARGET | | | = 28800.0 nM|> 30000.0 nM | > 20000.0 nM|= 17000.0 nM|> 50000.0 nM|= 46000.0 nM|= 26000.0 nM|> 10000.0 nM | | | NPASS |
| NIH3T3 | Mus musculus | | > 30000.0 nM | | | | NPASS |
| NCI-H460 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| MDCK | Canis lupus familiaris | | | > 20000.0 nM | | | NPASS |
| MGC-803 | Homo sapiens | | | = 30200.0 nM | | | NPASS |
| MDA-MB-435 | Homo sapiens | | | > 10000.0 nM | | | NPASS |
| MDA-MB-231 | Homo sapiens | | | > 500000.0 nM|> 10000.0 nM|= 96190.0 nM|= 24570.0 nM | | | NPASS |
| MCF7 | Homo sapiens | | = 24400.0 nM|> 30000.0 nM | = 23300.0 nM|= 19300.0 nM|> 500000.0 nM|= 43880.0 nM | | | NPASS |
| LN-229 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| L02 | Homo sapiens | | | = 26820.0 nM | | | NPASS |
| MIA PaCa-2 | Homo sapiens | | | = 95000.0 nM | | | NPASS |
| Plasmodium falciparum | Plasmodium falciparum | | = 3938.0 nM | | | | NPASS |
| Protein kinase C epsilon | Homo sapiens | Q02156 | | > 150000.0 nM | | | NPASS |
| Protein kinase C beta type | Homo sapiens | P05771 | | >150000 nM | | | BindingDB |
| K562 | Homo sapiens | | | > 250000.0 nM|= 12890.0 nM|> 100000.0 nM | | | NPASS |
| Z-138 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| WI-38 VA13 | Homo sapiens | | | = 20300.0 nM | | | NPASS |
| Vero | Chlorocebus aethiops | | | > 10.0 ug.mL-1|> 500000.0 nM | | | NPASS |
| Tyrosine-protein phosphatase non-receptor type 1 [1-405] | Homo sapiens | P18031 | | | | 2000 nM | BindingDB |
| Tyrosine-protein phosphatase non-receptor type 1 [1-321] | Homo sapiens | P18031 | | | | 3000 nM | BindingDB |
| Trypanosoma brucei brucei | Trypanosoma brucei brucei | | | = 8900.0 nM | | | NPASS |
| Transcription factor p65 | Homo sapiens | Q04206 | | 8800 nM | | | BindingDB |
| T47D | Homo sapiens | | | = 20720.0 nM | | | NPASS |
| SiHa | Homo sapiens | | | > 500000.0 nM | | | NPASS |
| Semliki forest virus | Semliki forest virus | | | = 45500.0 nM|= 45708.82 nM | | | NPASS |
| SK-MEL-2 | Homo sapiens | | | > 250000.0 nM | | | NPASS |
| SARS-CoV-2 | Severe acute respiratory syndrome coronavirus 2 | | | > 20000.0 nM|> 19952.62 nM | | | NPASS |
| Reverse transcriptase | Human immunodeficiency virus 1 | | | >451000 nM | | | BindingDB |
| Protein kinase C epsilon type | Homo sapiens | Q02156 | | >150000 nM | | | BindingDB |
| Protein kinase C beta | Homo sapiens | P05771 | | > 150000.0 nM | | | NPASS |
| J774 | Mus musculus | | | = 67100.0 nM | | | NPASS |
| KB | Homo sapiens | | | > 10.0 ug.mL-1|> 500000.0 nM | | | NPASS |
| Human immunodeficiency virus 1 | Human immunodeficiency virus 1 | | = 23000.0 nM|= 23014.42 nM | = 13800.0 nM | | | NPASS |
| DNA topoisomerase 2-alpha | Homo sapiens | P11388 | | 38600 nM | | | BindingDB |
| DLD-1 | Homo sapiens | | | = 6600.0 nM|> 200000.0 nM | | | NPASS |
| CCRF-CEM | Homo sapiens | | | > 250000.0 nM|= 250000.0 nM|= 50800.0 nM | | | NPASS |
| CAPAN-1 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| Bile acid transporter | Homo sapiens | Q14973 | | = 109000.0 nM | | | NPASS |
| Bile acid receptor FXR | Homo sapiens | Q96RI1 | = 0.0 nM | | | | NPASS |
| BGC-823 | Homo sapiens | | | > 20000.0 nM | | | NPASS |
| B16 | Mus musculus | | | = 27400.0 nM | | | NPASS |
| ADR5000 cell line | | | | = 56500.0 nM | | | NPASS |
| A549 | Homo sapiens | | = 20600.0 nM|> 30000.0 nM | = 3800.0 nM|> 316000.0 nM|> 200000.0 nM|> 10000.0 nM|= 18150.0 nM|= 59730.0 nM | | | NPASS |
| A2780 | Homo sapiens | | = 29300.0 nM|> 30000.0 nM | = 6100.0 nM|> 10000.0 nM | | | NPASS |
| A-375 | Homo sapiens | | > 30000.0 nM | = 28000.0 nM | | | NPASS |
| 8505C | Homo sapiens | | > 30000.0 nM | | | | NPASS |
| 5'-nucleotidase | Mus musculus | Q61503 | | 50320 nM|= 50320.0 nM | | | BindingDB, NPASS |
| 5'-nucleotidase | Homo sapiens | P21589 | | 22660 nM|= 22660.0 nM | | | BindingDB, NPASS |
| DNA topoisomerase II alpha | Homo sapiens | P11388 | | = 38600.0 nM | | | NPASS |
| DU-145 | Homo sapiens | | | = 136700.0 nM | | | NPASS |
| Bcap37 | Homo sapiens | | | = 25500.0 nM | | | NPASS |
| Ectonucleoside triphosphate diphosphohydrolase 1 | Mus musculus | P55772 | | 49760 nM|= 49760.0 nM | | | BindingDB, NPASS |
| ECa-109 cell line | | | | = 26640.0 nM | | | NPASS |
| Human immunodeficiency virus type 1 reverse transcriptase | Human immunodeficiency virus 1 | Q72547 | | > 200.0 ug.mL-1 | | | NPASS |
| Human herpesvirus 1 strain KOS | Human herpesvirus 1 strain KOS | | | = 700.0 nM | | | NPASS |
| Herpes simplex virus (type 1 / strain F) | Herpes simplex virus (type 1 / strain F) | | | = 900.0 nM | | | NPASS |
| HepG2 | Homo sapiens | | | = 10700.0 nM|> 20000.0 nM | | | NPASS |
| HeLa | Homo sapiens | | > 30000.0 nM | > 10.0 ug.mL-1|> 500000.0 nM|= 12200.0 nM | | | NPASS |
| HT-29 | Homo sapiens | | > 30000.0 nM | > 250000.0 nM|> 10000.0 nM|> 20000.0 nM | | | NPASS |
| HL-60 | Homo sapiens | | | = 30940.0 nM|> 100000.0 nM | | | NPASS |
| Human herpesvirus 2 strain G | Human herpesvirus 2 strain G | | | = 9400.0 nM | | | NPASS |
| HEK293 | Homo sapiens | | | > 500000.0 nM | | | NPASS |
| HCT-116 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| H9 | Homo sapiens | | = 23000.0 nM | = 43700.0 nM|= 45000.0 nM | | | NPASS |
| Glycogen phosphorylase, muscle form | Oryctolagus cuniculus | P00489 | | 17000 nM|41500 nM|= 17000.0 nM|= 41500.0 nM|= 16982.44 nM | | | BindingDB, NPASS |
| G-protein coupled bile acid receptor 1 | Homo sapiens | Q8TDU6 | >10000 nM|> 10000.0 nM | | | | BindingDB, NPASS |
| FaDu | Homo sapiens | | > 30000.0 nM | | | | NPASS |
| HEp-2 | Homo sapiens | | | > 10.0 ug.mL-1|> 500000.0 nM | | | NPASS |
