| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Tyrosyl-DNA phosphodiesterase 1 | Homo sapiens | Q9NUW8 | | >100000 nM|> 100000.0 nM | | | BindingDB, NPASS |
| Tyrosine-protein phosphatase non-receptor type 1 [1-405] | Homo sapiens | P18031 | | | | 1000 nM | BindingDB |
| Tyrosine-protein phosphatase non-receptor type 1 [1-321] | Homo sapiens | P18031 | | | | 2500 nM | BindingDB |
| Tyrosine-protein phosphatase non-receptor type 1 | Homo sapiens | P18031 | | 15600 nM | | | BindingDB |
| Trypanosoma cruzi | Trypanosoma cruzi | | | > 32000.0 nM | | | NPASS |
| Trypanosoma brucei brucei | Trypanosoma brucei brucei | | | = 27800.0 nM | | | NPASS |
| Trypanosoma brucei | Trypanosoma brucei | | | > 32000.0 nM | | | NPASS |
| Transcription factor p65 | Homo sapiens | Q04206 | | >10000 nM | | | BindingDB |
| RAW264.7 | Mus musculus | | | > 100000.0 nM | | | NPASS |
| Protein-tyrosine phosphatase 1B | Homo sapiens | P18031 | | = 15600.0 nM | | | NPASS |
| WI-38 VA13 | Homo sapiens | | | = 58300.0 nM | | | NPASS |
| Polyunsaturated fatty acid lipoxygenase ALOX15B | Homo sapiens | O15296 | | >40000 nM | | | BindingDB |
| Polyunsaturated fatty acid 5-lipoxygenase | Homo sapiens | P09917 | | 42000 nM | | | BindingDB |
| OVCAR-3 | Homo sapiens | | | > 10000.0 nM | | | NPASS |
| Nuclear factor NF-kappa-B p65 subunit | Homo sapiens | Q04206 | | > 10000.0 nM | | | NPASS |
| Lu1 | Homo sapiens | | | = 53300.0 nM | | | NPASS |
| MDA-MB-435 | Homo sapiens | | | > 10000.0 nM | | | NPASS |
| NON-PROTEIN TARGET | | | | = 214000.0 nM | | | NPASS |
| Arachidonate 15-lipoxygenase, type II | Homo sapiens | O15296 | | > 40000.0 nM | | | NPASS |
| Arachidonate 5-lipoxygenase | Homo sapiens | P09917 | | = 42000.0 nM | | | NPASS |
| B16 | Mus musculus | | | = 46800.0 nM | | | NPASS |
| Bile acid receptor FXR | Homo sapiens | Q96RI1 | = 0.0 nM | | | | NPASS |
| G-protein coupled bile acid receptor 1 | Homo sapiens | Q8TDU6 | >10000 nM|> 10000.0 nM | | | | BindingDB, NPASS |
| A549 | Homo sapiens | | | > 316000.0 nM | | | NPASS |
| HepG2 | Homo sapiens | | | = 53700.0 nM | | | NPASS |
| J774 | Mus musculus | | | = 155800.0 nM | | | NPASS |
| KB | Homo sapiens | | | = 37700.0 nM | | | NPASS |
| MCF7 | Homo sapiens | | | = 58200.0 nM | | | NPASS |
| MDA-MB-231 | Homo sapiens | | | > 10000.0 nM | | | NPASS |
| HT-29 | Homo sapiens | | | > 10000.0 nM | | | NPASS |