| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Hydroxycarboxylic acid receptor 2 | Homo sapiens | Q8TDS4 | | | | 4900 nM|= 4900.0 nM | BindingDB, NPASS |
| Leishmania amazonensis | Leishmaamazonensis | | | = 15500.0 nM | | | NPASS |
| Leishmania donovani | Leishmadonovani | | | = 37820.0 nM | | | NPASS |
| MCF7 | Homo sapiens | | | = 108000.0 nM | | | NPASS |
| MIA PaCa-2 | Homo sapiens | | | = 1330000.0 nM | | | NPASS |
| Meloidogyne incognita | Meloidogyne incognita | | > 250.0 ug.mL-1 | | | | NPASS |
| Mus musculus | Mus musculus | | | > 100000.0 nM|= 180.0 nM | | | NPASS |
| NCI-H460 | Homo sapiens | | | = 2100000.0 nM | | | NPASS |
| Xanthine dehydrogenase/oxidase | Homo sapiens | P47989 | | 175000 nM | | | BindingDB |
| Polyphenol oxidase 2 | Agaricus bisporus | O42713 | | 410000 nM|>350000 nM | | | BindingDB |
| Poly [ADP-ribose] polymerase tankyrase-1/tankyrase-2 | Homo sapiens | O95271|Q9H2K2 | | 685 nM | | | BindingDB |
| Radical scavenging activity | | | > 250000.0 nM | = 96.7 ug.mL-1 | | | NPASS |
| Tankyrase 1/2 | Homo sapiens | O95271 | | = 685.0 nM | | | NPASS |
| Trypanosoma brucei rhodesiense | Trypanosoma brucei rhodesiense | | | = 222900.0 nM | | | NPASS |
| Trypanosoma cruzi | Trypanosoma cruzi | | | = 202630.0 nM | | | NPASS |
| Tyrosinase | Agaricus bisporus | O42713 | | = 410000.0 nM|> 350000.0 nM|= 209500.0 nM | | | NPASS |
| Xanthine dehydrogenase | Homo sapiens | P47989 | | = 26.4 ug.mL-1 | | | NPASS |
| Histone deacetylase | Homo sapiens | Q969S8 | | | | = 8.21 nM | NPASS |
| NON-PROTEIN TARGET | | | | = 671400.0 nM|= 50180.0 nM|= 24810.0 nM | | | NPASS |
| Histone deacetylase | Homo sapiens | O15379|P56524|Q13547|Q8WUI4|Q92769|Q969S8|Q96DB2|Q9BY41|Q9UBN7|Q9UKV0|Q9UQL6 | | | | 8.2 nM | BindingDB |
| Aldose reductase | Homo sapiens | P15121 | | = 68.1 ug.mL-1 | | | NPASS |
| HT-22 | Mus musculus | | > 10000.0 nM | | | | NPASS |
| 3-oxoacyl-[acyl-carrier-protein] synthase 3 | Escherichia coli | | | 43400 nM | | | BindingDB |
| 3-oxoacyl-[acyl-carrier-protein] synthase 3 | Escherichia coli | C3TDZ2 | | = 43400.0 nM | | | NPASS |
| A-375 | Homo sapiens | | | = 64000.0 nM | | | NPASS |
| A549 | Homo sapiens | | | = 87000.0 nM|= 3540000.0 nM | | | NPASS |
| HT-29 | Homo sapiens | | | = 114000.0 nM | | | NPASS |
| Acetylcholinesterase | Electrophorus electricus | O42275 | | = 9900000.0 nM | | | NPASS |
| Acetylcholinesterase | Homo sapiens | P22303 | | 9.900e+6 nM | | | BindingDB |
| Aldo-keto reductase family 1 member B1 | Homo sapiens | P15121 | | | | 280000 nM | BindingDB |
| ACHN | Homo sapiens | | | = 91000.0 nM | | | NPASS |
| Alpha-glucosidase MAL62 | Saccharomyces cerevisiae | P07265 | | >300000 nM|> 300000.0 nM | | | BindingDB, NPASS |
| Amyloid-beta precursor protein | Homo sapiens | P05067 | | >100000 nM | | | BindingDB |
| BV-2 | Mus musculus | | > 10000.0 nM | > 100000.0 nM | | | NPASS |
| Beta amyloid A4 protein | Homo sapiens | P05067 | | > 100000.0 nM | | | NPASS |
| CaM kinase II alpha | Homo sapiens | Q9UQM7 | | | | > 100000.0 nM | NPASS |
| Dihydroorotate dehydrogenase (fumarate) | Leishmamajor | | | 398107 nM|391600 nM | | | BindingDB |
| Dihydroorotate dehydrogenase (fumarate) | Leishmamajor | Q4QEW7 | | = 391600.0 nM|= 398107.17 nM | | | NPASS |
| HT-144 | Homo sapiens | | | = 2400000.0 nM|= 1070000.0 nM | | | NPASS |
| Aldo-keto reductase family 1 member B1 [W220Y,C299A] | Homo sapiens | P15121 | | | | 1390000 nM | BindingDB |