IMPPAT Phytochemical information: 
Ouabain

Ouabain
Bioactivity information
Target nameTarget organismUniProt identifierEC50IC50KdKiSource
SARS-CoV-2Severe acute respiratory syndrome coronavirus 2> 20000.0 nM|> 19952.62 nMNPASS
SK-BR-3Homo sapiens= 403.0 nMNPASS
SK-MEL-28Homo sapiens= 211.0 nMNPASS
Signal transducer and activator of transcription 1-alpha/betaHomo sapiensP42224>55700 nM|> 55700.0 nMBindingDB, NPASS
Signal transducer and activator of transcription 3Homo sapiensP40763= 1154.0 nMNPASS
Signal transducer and activator of transcription 3 [702-738,740-752]Homo sapiensP407631154 nMBindingDB
Sodium/potassium-transporting ATPaseHomo sapiensP54710= 6000.0 nM|= 3.4 ug.mL-1|= 6600.0 nMNPASS
Sodium/potassium-transporting ATPase subunit alpha-1/beta-1HumanP05023|P0502697 nMBindingDB
Sodium/potassium-transporting ATPase subunit alpha-1/beta-1Rattus norvegicusP06685|P073404300 nMBindingDB
Sodium/potassium-transporting ATPase subunit alpha-2/beta-1HumanP05026|P5099390 nMBindingDB
Sodium/potassium-transporting ATPase subunit alpha-2/beta-1Rattus norvegicusP06686|P07340170 nMBindingDB
Sodium/potassium-transporting ATPase subunit alpha-3/beta-1Rattus norvegicusP06687|P0734031.0 nMBindingDB
Sodium/potassium-transporting ATPase subunit alpha-4/beta-1Rattus norvegicusP07340|Q645414.3 nMBindingDB
Sodium/potassium-transporting ATPase subunit alpha-4/beta-3Rattus norvegicusQ63377|Q645411.8 nMBindingDB
T47DHomo sapiens= 385.0 nMNPASS
Trypanosoma brucei rhodesienseTrypanosoma brucei rhodesiense> 450000.0 nMNPASS
Trypanosoma cruziTrypanosoma cruzi> 450000.0 nMNPASS
Vaccinia virusVaccivirus= 250.0 nMNPASS
Reverse transcriptaseHuman immunodeficiency virus 1>342000 nMBindingDB
Replicase polyprotein 1ab2019-nCoVP0DTD1<97 nMBindingDB
VeroChlorocebus aethiops< 50.0 nMNPASS
Potassium voltage-gated channel subfamily H member 2Homo sapiensQ128095800 nMBindingDB
A549Homo sapiens= 27.0 nMNPASS
B16-F10Mus musculus> 10000.0 nMNPASS
Bile salt export pumpHomo sapiensO95342>1000000 nM|> 1000000.0 nMBindingDB, NPASS
HERGHomo sapiensQ12809= 5800.0 nMNPASS
Hs-578THomo sapiens= 110.0 nM|= 93000.0 nMNPASS
Human immunodeficiency virus type 1 reverse transcriptaseHuman immunodeficiency virus 1Q72547> 200.0 ug.mL-1NPASS
Krueppel-like factor 5Homo sapiensQ1388729.73 nMBindingDB
Kruppel-like factor 5Homo sapiensQ13887= 164.55 nMNPASS
Leishmania donovaniLeishmadonovani> 450000.0 nMNPASS
Potassium-transporting ATPase alpha chain 2Homo sapiensP54707200000 nM|= 200000.0 nMBindingDB, NPASS
Meloidogyne incognitaMeloidogyne incognita> 1000.0 ug.mL-1NPASS
N+/K+ ATPase alpha-4/beta-1Rattus norvegicus= 4.3 nMNPASS
N+/K+ ATPase alpha-4/beta-3Rattus norvegicus= 1.8 nMNPASS
NON-PROTEIN TARGET> 10000.0 nM|= 77.0 nM|= 28.0 nMNPASS
Na+/K+ ATPase alpha-1/beta-1Rattus norvegicus= 4300.0 nMNPASS
Na+/K+ ATPase alpha-2/beta-1Rattus norvegicus= 170.0 nMNPASS
Na+/K+ ATPase alpha-3/beta-1Rattus norvegicus= 31.0 nMNPASS
PC-3Homo sapiens= 43.0 nMNPASS
Plasmodium falciparumPlasmodium falciparum= 12589.25 nMNPASS
MCF7Homo sapiens= 10600.0 nM|= 133.0 nMNPASS