| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| NON-PROTEIN TARGET | | | | = 43100.0 nM|= 23900.0 nM|= 55400.0 nM | | | NPASS |
| Pancreatic alpha-amylase | Sus scrofa | P00690 | | | | 48000 nM|= 48000.0 nM | BindingDB, NPASS |
| PBMC | Homo sapiens | | | = 27000.0 nM | | | NPASS |
| PANC-1 | Homo sapiens | | | = 26000.0 nM | | | NPASS |
| P388 | Mus musculus | | | = 9630.0 nM | | | NPASS |
| Pancreatic triacylglycerol lipase | Sus scrofa | P00591 | | 84410 nM|= 84410.0 nM | | | BindingDB, NPASS |
| Monoamine oxidase B | Homo sapiens | P27338 | | = 1410.0 nM|= 1412537.54 nM | | = 56.0 nM | NPASS |
| Leishmania braziliensis | Leishmabraziliensis | | | = 13700.0 nM | | | NPASS |
| MDA-MB-231 | Homo sapiens | | | = 6700.0 nM|= 42800.0 nM|> 10000.0 nM | | | NPASS |
| MCF7 | Homo sapiens | | | = 63000.0 nM|= 12600.0 nM|> 10000.0 nM | | | NPASS |
| Leishmania infantum | Leishmaitum | | = 1.3 ug.mL-1|= 1.5 ug.mL-1|= 5.1 ug.mL-1|= 5.7 ug.mL-1|= 8890.0 nM | | | | NPASS |
| ZR-75-1 | Homo sapiens | | | = 13700.0 nM | | | NPASS |
| Leishmania donovani | Leishmadonovani | | | = 20000.0 nM | | | NPASS |
| Perilipin-1 | Homo sapiens | O60240 | | 4194 nM | | | BindingDB |
| Monoamine oxidase A | Homo sapiens | P21397 | | | | = 14.6 10^3nM | NPASS |
| Perilipin-5 | Homo sapiens | Q00G26 | | 4245 nM | | | BindingDB |
| Tumor necrosis factor receptor superfamily member 1A | Homo sapiens | P19438 | | 23000 nM | | | BindingDB |
| Polyunsaturated fatty acid 5-lipoxygenase | Mus musculus | P48999 | | 12200 nM | | | BindingDB |
| Leishmania amazonensis | Leishmaamazonensis | | = 13200.0 nM | | | | NPASS |
| Tumor necrosis factor receptor R1 | Homo sapiens | P19438 | | = 23000.0 nM | | | NPASS |
| Tubulin | Homo sapiens | Q9BUF5 | | = 620000.0 nM | | | NPASS |
| Trypanosoma cruzi | Trypanosoma cruzi | | = 102640.0 nM|= 26900.0 nM | | | | NPASS |
| Trypanosoma brucei | Trypanosoma brucei | | | = 0.473 ug.mL-1 | | | NPASS |
| Thioredoxin reductase 1, cytoplasmic | Rattus norvegicus | O89049 | | 46400 nM|26700 nM|= 26700.0 nM|= 46400.0 nM | | | BindingDB, NPASS |
| Plasmodium falciparum | Plasmodium falciparum | | | = 6.7 ug.mL-1 | | | NPASS |
| TK-10 | Homo sapiens | | | = 42000.0 nM | | | NPASS |
| Sortase family protein | Staphylococcus aureus | | | 53150 nM | | | BindingDB |
| Sortase A | Streptococcus mutans | Q8CM62 | | = 5000.0 nM | | | NPASS |
| Sortase A | Staphylococcus aureus | Q9S446 | | = 53150.0 nM | | | NPASS |
| Prostaglandin G/H synthase 2 | Mus musculus | Q05769 | | 11200 nM | | | BindingDB |
| Prostaglandin G/H synthase 1 | Mus musculus | P22437 | | 22100 nM | | | BindingDB |
| Polyunsaturated fatty acid 5-lipoxygenase | Rattus norvegicus | P12527 | | 43000 nM | | | BindingDB |
| Stromal cell-derived factor 1 | Homo sapiens | P48061 | | >5.00e+5 nM | | | BindingDB |
| L929 | Mus musculus | | | = 6.92 ug.mL-1 | | | NPASS |
| Homo sapiens | Homo sapiens | | | = 6280.0 nM|= 12700.0 nM|= 12500.0 nM | | | NPASS |
| KB | Homo sapiens | | | > 10000.0 nM | | | NPASS |
| Carboxylic ester hydrolase | Equus caballus | | | 1.090e+5 nM | | | BindingDB |
| CHO | Cricetulus griseus | | | = 23000.0 nM | | | NPASS |
| Butyrylcholinesterase | Homo sapiens | P06276 | | = 87000.0 nM | | | NPASS |
| Blood | Homo sapiens | | | = 162560.0 nM | | | NPASS |
| BT-20 | Homo sapiens | | | = 21100.0 nM | | | NPASS |
| Arachidonate 5-lipoxygenase | Rattus norvegicus | P12527 | | = 43000.0 nM | | | NPASS |
| Cholinesterase | Homo sapiens | P06276 | | 87000 nM | | | BindingDB |
| Arachidonate 5-lipoxygenase | Mus musculus | P48999 | | = 12200.0 nM | | | NPASS |
| Androgen Receptor | Rattus norvegicus | P15207 | | = 64565.42 nM | | | NPASS |
| Amine oxidase [flavin-containing] B | Homo sapiens | P27338 | | 1410 nM|1412538 nM | | 56 nM | BindingDB |
| Amine oxidase [flavin-containing] A | Homo sapiens | P21397 | | | | 14600 nM | BindingDB |
| A549 | Homo sapiens | | | > 10000.0 nM|= 69190.0 nM|= 12200.0 nM | | | NPASS |
| A2780 | Homo sapiens | | | = 67500.0 nM | | | NPASS |
| 2008 | Homo sapiens | | | = 33400.0 nM | | | NPASS |
| Androgen receptor | Rattus norvegicus | P15207 | | 64565.42 nM | | | BindingDB |
| Cyclooxygenase | Rattus norvegicus | Q63921 | | = 43000.0 nM | | | NPASS |
| L1210 | Mus musculus | | | = 41400.0 nM|> 100000.0 nM | | | NPASS |
| Cyclooxygenase-2 | Mus musculus | Q05769 | | = 11200.0 nM | | | NPASS |
| Cyclooxygenase-1 | Mus musculus | P22437 | | = 22100.0 nM | | | NPASS |
| K562 | Homo sapiens | | | = 3800.0 nM|= 4300000.0 nM | | | NPASS |
| Jurkat | Homo sapiens | | | = 17100.0 nM | | | NPASS |
| Human Tumor Cell lines | | | | = 8320.0 nM | | | NPASS |
| HeLa | Homo sapiens | | > 50000.0 nM | | | | NPASS |
| HT-29 | Homo sapiens | | = 14000.0 nM | = 70000.0 nM|= 45900.0 nM | | | NPASS |
| HEK293 | Homo sapiens | | | = 10700.0 nM | | | NPASS |
| HepG2 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| Entamoeba histolytica HM-1:IMSS | Eoeba histolytica HM-1:IMSS | | | = 12860.0 nM | | | NPASS |
| Entamoeba histolytica | Eoeba histolytica | | | = 1700.0 nM | | | NPASS |
| Dihydrofolate reductase | Homo sapiens | P00374 | | >100000 nM|> 100000.0 nM | | | BindingDB, NPASS |
| DU-145 | Homo sapiens | | | = 50100.0 nM | | | NPASS |
| DLD-1 | Homo sapiens | | = 25000.0 nM | | | | NPASS |
| Cytochrome P450 3A4 | Homo sapiens | P08684 | | > 10000.0 nM | | | NPASS |
| HCT-116 | Homo sapiens | | = 9500.0 nM|= 11000.0 nM | | | | NPASS |