| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Proteasome Macropain subunit MB1 | Homo sapiens | P28074 | | > 100000.0 nM | | | NPASS |
| N9 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| NON-PROTEIN TARGET | | | | = 83600.0 nM|> 100000.0 nM|= 56100.0 nM | | | NPASS |
| Neuraminidase | InflueA virus | B4URF0 | | > 100000.0 nM|= 5040.0 nM|= 3040.0 nM|= 1370.0 nM | | | NPASS |
| Neuraminidase | InflueA virus (A/WSN/1933(H1N1)) | P03470 | | >100000 nM|5040 nM|3040 nM|1370 nM | | | BindingDB |
| Monoamine oxidase B | Mus musculus | Q8BW75 | | = 11000.0 nM | | | NPASS |
| PC-3 | Homo sapiens | | | = 57010.0 nM | | | NPASS |
| Proteasome subunit beta type-5 | Homo sapiens | P28074 | | >100000 nM | | | BindingDB |
| Sortase family protein | Staphylococcus aureus | | | 74900 nM | | | BindingDB |
| SGC-7901 | Homo sapiens | | | = 2170.0 nM | | | NPASS |
| SH-SY5Y | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| Sortase A | Staphylococcus aureus | Q9S446 | | = 74900.0 nM | | | NPASS |
| Trypanosoma brucei brucei | Trypanosoma brucei brucei | | | = 90200.0 nM | | | NPASS |
| U-937 | Homo sapiens | | | = 50000.0 nM|= 44000.0 nM|= 45000.0 nM | | | NPASS |
| Urease subunit alpha/Urease subunit beta | Helicobacter pylori (strain ATCC 700392 / 26695) (Campylobacterpylori) | | | = 2003000.0 nM | | | NPASS |
| Urease subunit beta | Helicobacter pylori (strain ATCC 700392 / 26695) | P69996 | | 2003000 nM | | | BindingDB |
| Monoamine oxidase B | Homo sapiens | P27338 | | = 25800.0 nM | | | NPASS |
| SARS-CoV-2 | Severe acute respiratory syndrome coronavirus 2 | | | > 20000.0 nM|> 19952.62 nM | | | NPASS |
| Monoamine oxidase A | Mus musculus | Q64133 | | = 21200.0 nM | | | NPASS |
| Influenza A virus | InflueA virus | | | = 42600.0 nM|= 38200.0 nM | | | NPASS |
| MGC-803 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| Monoamine oxidase A | Homo sapiens | P21397 | | = 31200.0 nM | | | NPASS |
| A549 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| Amine oxidase [flavin-containing] A | Homo sapiens | P21397 | | 31200 nM | | | BindingDB |
| Amine oxidase [flavin-containing] A | Mus musculus | O75477 Q64133 | | 21200 nM | | | BindingDB |
| Amine oxidase [flavin-containing] B | Mus musculus | Q8BW75 | | 11000 nM | | | BindingDB |
| BV-2 | Mus musculus | | | > 100000.0 nM|= 13190.0 nM|> 50000.0 nM | | | NPASS |
| Cytochrome P450 1A1 | Homo sapiens | P04798 | | <100000 nM|< 100000.0 nM | | | BindingDB, NPASS |
| Cytochrome P450 1B1 | Homo sapiens | Q16678 | | | | 3700 nM|= 3700.0 nM | BindingDB, NPASS |
| DU-145 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| Amine oxidase [flavin-containing] B | Homo sapiens | P27338 | | 25800 nM | | | BindingDB |
| Giardia intestinalis | Giardia intestinalis | | | < 1.0 ug.mL-1|= 0.03 ug.mL-1 | | | NPASS |
| HCT-116 | Homo sapiens | | | = 60970.0 nM | | | NPASS |
| HT-1080 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| HeLa | Homo sapiens | | | > 100000.0 nM|= 8510.0 nM | | | NPASS |
| Interleukin-2 | Homo sapiens | P60568 | | | 5470 nM|= 5470.0 nM | | BindingDB, NPASS |
| HepG2 | Homo sapiens | | | = 60500.0 nM | | | NPASS |
| Histone deacetylase 6 | Homo sapiens | Q9UBN7 | | = 287.9 nM|= 590.7 nM | | | NPASS |
| ECa-109 cell line | | | | > 100000.0 nM | | | NPASS |