| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Cytochrome P450 2A6 | Homo sapiens | P11509 | | 25000 nM|25003 nM|= 25000.0 nM|= 25003.45 nM | | | BindingDB, NPASS |
| Cytochrome P450 1A2 | Homo sapiens | P05177 | | 700000 nM|= 700000.0 nM | | | BindingDB, NPASS |
| Alpha-2C adrenergic receptor | Homo sapiens | P18825 | | | | 3.31 nM | BindingDB |
| Cytochrome P450 2A5 | Mus musculus | P20852 | | 74000 nM|73961 nM|= 74000.0 nM|= 73960.53 nM | | | BindingDB, NPASS |
| Alpha-2A adrenergic receptor | Mus musculus | | | | | 7.76 nM|9.33 nM | BindingDB |
| Alpha-2A adrenergic receptor | Homo sapiens | P08913 | | | | 4.57 nM | BindingDB |
| Alpha-2B adrenergic receptor | Homo sapiens | P18089 | | | | 16.98 nM | BindingDB |