| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Transient receptor potential cation channel subfamily M member 8 | Rattus norvegicus | Q8R455 | 75000 nM | | | | BindingDB |
| Voltage-gated L-type calcium channel alpha-1C subunit | Oryctolagus cuniculus | P15381 | | = 74600.0 nM | | | NPASS |
| Transient receptor potential cation channel subfamily M member 8 | Human | Q7Z2W7 | 3800 nM | | | | BindingDB |
| Transient receptor potential cation channel subfamily M member 8 | Homo sapiens | Q7Z2W7 | 10100 nM|29000 nM|3000 nM|= 10100.0 nM|= 60000.0 nM | 92000 nM | 14400 nM | | BindingDB, NPASS |
| Transient receptor potential cation channel subfamily A member 1 | Mus musculus | Q8BLA8 | 56000 nM | | | | BindingDB |
| Transient receptor potential cation channel subfamily A member 1 | Homo sapiens | O75762 | 96000 nM|28400 nM|= 96000.0 nM | | | | BindingDB, NPASS |