
| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|---|---|---|---|---|---|---|
| Leishmania infantum | Leishmaitum | > 50000.0 nM | NPASS | ||||
| U-937 | Homo sapiens | = 589900.0 nM | NPASS | ||||
| Neutrophils | > 100000.0 nM | NPASS | |||||
| NON-PROTEIN TARGET | = 80000.0 nM | > 50000.0 nM|= 42860.0 nM|= 41400.0 nM|> 30000.0 nM|= 8.25 ug.mL-1|> 100000.0 nM|= 54400.0 nM | NPASS | ||||
| Leishmania mexicana | Leishmamexicana | = 9.11 ug.mL-1 | NPASS | ||||
| Leishmania major | Leishmamajor | = 14.37 ug.mL-1 | NPASS | ||||
| Leishmania chagasi | Leishmachagasi | = 21.4 ug.mL-1 | NPASS | ||||
| Leishmania donovani | Leishmadonovani | = 27.51 ug.mL-1 | NPASS | ||||
| Leishmania amazonensis | Leishmaamazonensis | > 50000.0 nM | NPASS | ||||
| A549 | Homo sapiens | > 100000.0 nM | NPASS | ||||
| Beta-secretase 1 | Homo sapiens | P56817 | >500000 nM|> 500000.0 nM | BindingDB, NPASS | |||
| Collagenase ColH | Hathewaya histolytica | Q46085 | 24 nM|= 24.0 nM | BindingDB, NPASS | |||
| Leishmania braziliensis | Leishmabraziliensis | > 50000.0 nM | NPASS | ||||
| HL-60 | Homo sapiens | = 1.1 ug.mL-1 | NPASS | ||||
| Induced myeloid leukemia cell differentiation protein Mcl-1 | Homo sapiens | Q07820 | 25140 nM|= 25140.0 nM | 9540 nM|= 9540.0 nM | BindingDB, NPASS | ||
| DLD-1 | Homo sapiens | > 100000.0 nM | NPASS |