| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Vitamin D3 receptor | Bos taurus | Q28037 | 0.05 nM|0.0710 nM | 0.048000 nM | | | BindingDB |
| Vitamin D3 receptor | Sus scrofa | A3RGC1 | | | 0.070 nM | | BindingDB |
| Vitamin D3 receptor | Rattus norvegicus | P13053 | 0.2 nM|0.3 nM|0.05 nM|0.1 nM | | | 0.100 nM|0.040000 nM|0.05 nM|0.1 nM|0.2 nM | BindingDB |
| Vitamin D3 receptor A | Danio rerio | Q9PTN2 | 5.5 nM | | 1200 nM | | BindingDB |
| Vitamin D3 receptor | Homo sapiens | P11473 | 1 nM|7.7 nM|322 nM|515 nM|0.120000 nM|0.600000 nM|3.9 nM|223 nM|250 nM|10 nM|0.300000 nM|0.01 nM|9.0 nM|0.5 nM|0.555 nM|0.0106 nM|3.52 nM|2.5 nM|3.28 nM|>0.900000 nM|0.070000 nM|3.0 nM|0.026000 nM|15 nM|1.6 nM|0.011000 nM|0.100000 nM|7.0 nM|4.9 nM | 0.080000 nM|0.70 nM|0.8 nM|0.060000 nM|0.350000 nM|0.100000 nM|0.160000 nM|1.1 nM|13 nM|1.24 nM|0.040000 nM|0.050000 nM|9.3 nM|1.3 nM|0.095300 nM|1.4 nM|6430 nM|1.2 nM | 0.065 nM | | BindingDB |
| Vitamin D3 receptor | Gallus gallus | O42392 | | | | 0.025000 nM | BindingDB |
| Vitamin D-binding protein | Homo sapiens | | | | 24 nM | | BindingDB |
| Vitamin D3 receptor | Mus musculus | P48281 | 100 nM | | | | BindingDB |
| Bile salt export pump | Homo sapiens | O95342 | | 39700 nM | | | BindingDB |
| Androgen receptor | Homo sapiens | P10275 | | >10000 nM | | | BindingDB |
| ATP-binding cassette sub-family C member 4 | Homo sapiens | O15439 | | >133000 nM | | | BindingDB |
| ATP-binding cassette sub-family C member 3 | Homo sapiens | O15438 | | >133000 nM | | | BindingDB |
| ATP-binding cassette sub-family C member 2 | Homo sapiens | Q92887 | | >133000 nM | | | BindingDB |
| 1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial | Homo sapiens | Q07973 | 3.0 nM | | | | BindingDB |
| Retinoic acid receptor RXR-alpha/Vitamin D3 receptor | Homo sapiens | P11473|P19793 | 1.6 nM | | | | BindingDB |