| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| LNCaP C4-2B | Homo sapiens | | | = 240000.0 ug.mL-1 | | | NPASS |
| NON-PROTEIN TARGET | | | | = 74200.0 nM|= 150000.0 nM | | | NPASS |
| PC-3 | Homo sapiens | | | = 250000.0 ug.mL-1 | | | NPASS |
| Prostaglandin G/H synthase 1 | Homo sapiens | P23219 | | 129000 nM | | | BindingDB |
| Prostaglandin G/H synthase 2 | Homo sapiens | P35354 | | 125000 nM | | | BindingDB |
| Transient receptor potential cation channel subfamily A member 1 | Rattus norvegicus | Q6RI86 | 10400 nM | >100000 nM | | | BindingDB |
| SCC-4 | Homo sapiens | | | = 500000000.0 nM | | | NPASS |
| Serotonin 1a (5-HT1a) receptor | Homo sapiens | P08908 | | | | > 100000.0 nM | NPASS |
| Transient receptor potential cation channel subfamily V member 1 | Homo sapiens | Q8NER1 | 3300 nM | 5000 nM | | | BindingDB |
| LNCaP C4-2 | Homo sapiens | | | = 512000.0 ug.mL-1 | | | NPASS |
| Regulatory protein RhlR | Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) | P54292 | | = 945000.0 nM | | | NPASS |
| LNCaP | Homo sapiens | | | = 75000.0 ug.mL-1 | | | NPASS |
| HeLa | Homo sapiens | | | = 636000000.0 nM | | | NPASS |
| Cytochrome P450 1A2 | Homo sapiens | P05177 | | 19000 nM|= 19000.0 nM | | | BindingDB, NPASS |
| HTH-type quorum-sensing regulator RhlR | Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22644 / CIP 104116 / JCM 14847 / LMG 12228 / 1C / PRS 101 / PAO1) | P54292 | | 945000 nM | | | BindingDB |
| DU-145 | Homo sapiens | | | = 95000.0 ug.mL-1 | | | NPASS |
| Cytochrome P450 3A4 | Homo sapiens | P08684 | | 42900 nM|37400 nM|21800 nM|32000 nM|73400 nM|= 73400.0 nM|= 37400.0 nM|= 32000.0 nM|= 42900.0 nM|= 21800.0 nM | | | BindingDB, NPASS |
| Cytochrome P450 2C9 | Homo sapiens | P11712 | | 12100 nM|27900 nM|= 27900.0 nM|= 12100.0 nM | | | BindingDB, NPASS |
| Cytochrome P450 2C8 | Homo sapiens | P10632 | | 22100 nM|= 22100.0 nM | | | BindingDB, NPASS |
| Cytochrome P450 2C19 | Homo sapiens | P33261 | | 30700 nM|10900 nM|= 10900.0 nM|= 30700.0 nM | | | BindingDB, NPASS |
| Cytochrome P450 2B6 | Homo sapiens | P20813 | | 40800 nM|= 40800.0 nM | | | BindingDB, NPASS |
| Cyclooxygenase-2 | Homo sapiens | P35354 | | = 125000.0 nM | | | NPASS |
| Cyclooxygenase-1 | Homo sapiens | P23219 | | = 129000.0 nM | | | NPASS |
| 5-hydroxytryptamine receptor 1A | Homo sapiens | P08908 | | | | >100000 nM | BindingDB |
| KB | Homo sapiens | | | = 480000000.0 nM | | | NPASS |