| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Cytochrome P450 3A4 | Homo sapiens | P08684 | | >30000 nM|30000 nM|> 30000.0 nM|= 30000.0 nM | | | BindingDB, NPASS |
| Cytochrome P450 2C8 | Homo sapiens | P10632 | | 5100 nM|3800 nM|8300 nM|= 5100.0 nM|= 8300.0 nM|= 3800.0 nM | | | BindingDB, NPASS |
| Cytochrome P450 2D6 | Homo sapiens | P10635 | | >30000 nM|> 30000.0 nM | | | BindingDB, NPASS |
| NON-PROTEIN TARGET | | | | = 84000.0 nM|= 66500.0 nM | | | NPASS |
| Cytochrome P450 2C9 | Homo sapiens | P11712 | | 13600 nM|9900 nM|10500 nM|= 13600.0 nM|= 9900.0 nM|= 10500.0 nM | | | BindingDB, NPASS |
| Cytochrome P450 1A2 | Homo sapiens | P05177 | | 21400 nM|7100 nM|19600 nM|= 7100.0 nM|= 19600.0 nM|= 21400.0 nM | | | BindingDB, NPASS |
| Cytochrome P450 2C19 | Homo sapiens | P33261 | | 17600 nM|5800 nM|3600 nM|= 17600.0 nM|= 3600.0 nM|= 5800.0 nM | | | BindingDB, NPASS |
| Cytochrome P450 2B6 | Homo sapiens | P20813 | | 6300 nM|15400 nM|6200 nM|= 15400.0 nM|= 6300.0 nM|= 6200.0 nM | | | BindingDB, NPASS |
| Cytochrome P450 2A6 | Homo sapiens | P11509 | | >30000 nM|> 30000.0 nM | | | BindingDB, NPASS |