| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Cytochrome P450 2E1 | Homo sapiens | P05181 | | 76100 nM|99600 nM|= 76100.0 nM|= 99600.0 nM | | | BindingDB, NPASS |
| Vanilloid receptor | Homo sapiens | Q8NER1 | = 320.0 nM | = 290.0 nM | | | NPASS |
| Transient receptor potential cation channel subfamily A member 1 | Rattus norvegicus | Q6RI86 | = 16000.0 nM | = 16700.0 nM | | | NPASS |
| Serotonin 1a (5-HT1a) receptor | Homo sapiens | P08908 | | | | = 18020.0 nM | NPASS |
| NON-PROTEIN TARGET | | | | = 15600.0 nM|= 18700.0 nM|= 8000.0 nM|= 12870.0 nM|> 100000.0 nM | | | NPASS |
| Leukotriene A4 hydrolase | Homo sapiens | P09960 | | = 12540.0 nM|= 24610.0 nM | | | NPASS |
| HepG2 | Homo sapiens | | | = 88000.0 nM | | | NPASS |
| Cytochrome P450 2D6 | Homo sapiens | P10635 | | 87000 nM|> 100000.0 nM|= 87000.0 nM | | | BindingDB, NPASS |
| Cytochrome P450 3A4 | Homo sapiens | P08684 | | 8300 nM|65200 nM|4000 nM|= 77700.0 nM|= 8300.0 nM|= 65200.0 nM|= 4000.0 nM | | | BindingDB, NPASS |
| Cytochrome P450 2C8 | Homo sapiens | P10632 | | 2900 nM|= 2900.0 nM | | | BindingDB, NPASS |
| Cytochrome P450 2C9 | Homo sapiens | P11712 | | 3300 nM|29200 nM|= 3300.0 nM|= 29200.0 nM | | | BindingDB, NPASS |
| Cytochrome P450 2C19 | Homo sapiens | P33261 | | 18800 nM|= 18800.0 nM | | | BindingDB, NPASS |
| Cytochrome P450 2B6 | Homo sapiens | P20813 | | 5800 nM|= 5800.0 nM | | | BindingDB, NPASS |
| Cytochrome P450 2A6 | Homo sapiens | P11509 | | 83300 nM|= 83300.0 nM | | | BindingDB, NPASS |
| Cytochrome P450 1A2 | Homo sapiens | P05177 | | 20700 nM|2500 nM|= 2500.0 nM|= 20700.0 nM | | | BindingDB, NPASS |
| BV-2 | Mus musculus | | | = 5590.0 nM | | | NPASS |
| Arachidonate 5-lipoxygenase | Homo sapiens | P09917 | | = 7400.0 nM | | | NPASS |