IMPPAT Phytochemical information: 
Sinensetin

Sinensetin
Bioactivity information
Target nameTarget organismUniProt identifierEC50IC50KdKiSource
Human immunodeficiency virus 1Human immunodeficiency virus 1>= 100000.0 nMNPASS
Phytophthora citrophthoraPhytophthora citrophthora= 910000.0 nMNPASS
P-glycoprotein 1Homo sapiensP08183= 29000.0 nM|= 3200.0 nMNPASS
MDA-MB-468Homo sapiens= 200.0 nMNPASS
MDA-MB-231Homo sapiens= 268700.0 nMNPASS
MCF-10AHomo sapiens= 65000.0 nMNPASS
HT-29Homo sapiens= 67000.0 nMNPASS
Broad substrate specificity ATP-binding cassette transporter ABCG2Homo sapiensQ9UNQ08300 nM|9000 nMBindingDB
DNA polymerase etaHomo sapiensQ9Y253> 100000.0 nMNPASS
Aurora kinase BHomo sapiensQ96GD45.31e+3 nMBindingDB
ATP-dependent translocase ABCB1Homo sapiensP0818329000 nM|3200 nMBindingDB
ATP-binding cassette sub-family G member 2Homo sapiensQ9UNQ0= 9000.0 nM|= 8300.0 nMNPASS
3T3-L1Mus musculus= 59000.0 nMNPASS
HL-60Homo sapiens> 100000.0 nMNPASS