| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| LNCaP C4-2 | Homo sapiens | | | = 30300.0 nM | | | NPASS |
| Xanthine dehydrogenase/oxidase | Homo sapiens | P47989 | | >100000 nM | | | BindingDB |
| Xanthine dehydrogenase | Homo sapiens | P47989 | | > 100000.0 nM | | | NPASS |
| Phytophthora citrophthora | Phytophthora citrophthora | | | = 590000.0 nM | | | NPASS |
| PC-3 | Homo sapiens | | | = 122600.0 nM | | | NPASS |
| P-glycoprotein 1 | Homo sapiens | P08183 | | = 11500.0 nM | | | NPASS |
| NON-PROTEIN TARGET | | | | > 100000.0 nM | | | NPASS |
| HL-60 | Homo sapiens | | | = 41500.0 nM|= 0.01 ug.mL-1 | | | NPASS |
| HT-29 | Homo sapiens | | | = 24000.0 nM | | | NPASS |
| CWR22R | Homo sapiens | | | = 36530.0 nM | | | NPASS |
| Broad substrate specificity ATP-binding cassette transporter ABCG2 | Homo sapiens | Q9UNQ0 | | 4400 nM|4900 nM | | | BindingDB |
| ATP-dependent translocase ABCB1 | Homo sapiens | P08183 | | 11500 nM | | | BindingDB |
| ATP-binding cassette sub-family G member 2 | Homo sapiens | Q9UNQ0 | | = 4900.0 nM|= 4400.0 nM | | | NPASS |
| A549/TR | Homo sapiens | | | = 9000.0 nM | | | NPASS |
| A2780/Taxol | Homo sapiens | | | = 9000.0 nM | | | NPASS |
| 3T3-L1 | Mus musculus | | | = 50000.0 nM | | | NPASS |
| DU-145 | Homo sapiens | | | = 144500.0 nM | | | NPASS |