| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| V79 | Cricetulus griseus | | | > 100000.0 nM | | | NPASS |
| Carbonic anhydrase IV | Homo sapiens | P22748 | | | | = 8300.0 nM | NPASS |
| Carbonic anhydrase IX | Homo sapiens | Q16790 | | | | = 9800.0 nM | NPASS |
| Carbonic anhydrase VA | Homo sapiens | P35218 | | | | = 5100.0 nM | NPASS |
| Carbonic anhydrase VB | Homo sapiens | Q9Y2D0 | | | | > 500000.0 nM | NPASS |
| Carbonic anhydrase VI | Homo sapiens | P23280 | | | | = 5500.0 nM | NPASS |
| Carbonic anhydrase VII | Homo sapiens | P43166 | | | | = 2400.0 nM | NPASS |
| Carbonic anhydrase XII | Homo sapiens | O43570 | | | | = 9700.0 nM | NPASS |
| Carbonic anhydrase III | Homo sapiens | P07451 | | | | = 96000.0 nM | NPASS |
| Carbonic anhydrase XIV | Homo sapiens | Q9ULX7 | | | | = 9000.0 nM | NPASS |
| Cytochrome P450 19A1 | Homo sapiens | P11511 | | > 10000.0 nM | | | NPASS |
| Entamoeba histolytica | Eoeba histolytica | | | = 8920000.0 nM | | | NPASS |
| Exportin-1 | Homo sapiens | O14980 | | >25000 nM|> 25000.0 nM | | | BindingDB, NPASS |
| NON-PROTEIN TARGET | | | = 244000.0 nM | = 84000.0 nM | | | NPASS |
| RAW264.7 | Mus musculus | | | = 12400.0 nM | | | NPASS |
| Sorbitol dehydrogenase | Homo sapiens | Q00796 | | 124000 nM|= 124000.0 nM | | | BindingDB, NPASS |
| Carbonic anhydrase XIII | Mus musculus | Q9D6N1 | | | | = 8900.0 nM | NPASS |
| Carbonic anhydrase II | Homo sapiens | P00918 | | | | > 500000.0 nM | NPASS |
| Carbonic anhydrase 7 | Homo sapiens | P43166 | | | | 2400 nM | BindingDB |
| Carbonic anhydrase 9 | Homo sapiens | Q16790 | | | | 9800 nM | BindingDB |
| Aldo-keto reductase family 1 member B1 | Homo sapiens | P15121 | | 67500 nM|131000 nM | | | BindingDB |
| Aldose reductase | Homo sapiens | P15121 | | = 67500.0 nM|= 131000.0 nM | | | NPASS |
| Aromatase | Homo sapiens | P11511 | | >10000 nM | | | BindingDB |
| Beta-secretase 1 | Homo sapiens | P56817 | | >500000 nM|> 500000.0 nM | | | BindingDB, NPASS |
| Carbonic anhydrase 1 | Homo sapiens | P00915 | | | | 5900 nM | BindingDB |
| Carbonic anhydrase 12 | Homo sapiens | O43570 | | | | 9700 nM | BindingDB |
| Carbonic anhydrase 13 | Mus musculus | Q9D6N1 | | | | 8900 nM | BindingDB |
| Carbonic anhydrase 14 | Homo sapiens | Q9ULX7 | | | | 9000 nM | BindingDB |
| Carbonic anhydrase 15 | Mus musculus | Q99N23 | | | | 8400 nM|= 8400.0 nM | BindingDB, NPASS |
| Carbonic anhydrase 2 | Homo sapiens | P00918 | | | | >500000 nM | BindingDB |
| Carbonic anhydrase 3 | Homo sapiens | P07451 | | | | 96000 nM | BindingDB |
| Carbonic anhydrase 4 | Homo sapiens | P22748 | | | | 8300 nM | BindingDB |
| Carbonic anhydrase 5A, mitochondrial | Homo sapiens | P35218 | | | | 5100 nM | BindingDB |
| Carbonic anhydrase 5B, mitochondrial | Homo sapiens | Q9Y2D0 | | | | >500000 nM | BindingDB |
| Carbonic anhydrase 6 | Homo sapiens | P23280 | | | | 5500 nM | BindingDB |
| Carbonic anhydrase I | Homo sapiens | P00915 | | | | = 5900.0 nM | NPASS |