| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Dual-specificity tyrosine-phosphorylation regulated kinase 2 | Homo sapiens | Q92630 | | > 10000.0 nM | | | NPASS |
| SMMC-7721 | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| NON-PROTEIN TARGET | | | = 6650.0 nM | = 5030.0 nM|> 30000.0 nM | | | NPASS |
| NCI-H460 | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| MDA-MB-231 | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| MCF7 | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| HeLa | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| HT-22 | Mus musculus | | | > 100000.0 nM | | | NPASS |
| Glycogen synthase kinase-3 beta | Homo sapiens | P49841 | | > 10000.0 nM | | | NPASS |
| Dual-specificity tyrosine-phosphorylation regulated kinase 3 | Homo sapiens | O43781 | | > 10000.0 nM | | | NPASS |
| SW1990 | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| Dual-specificity tyrosine-phosphorylation regulated kinase 1A | Homo sapiens | Q13627 | | > 10000.0 nM | | | NPASS |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1B | Homo sapiens | Q9Y463 | | > 10000.0 nM | | | NPASS |
| Dual specificity tyrosine-phosphorylation-regulated kinase 4 | Homo sapiens | Q9NR20 | | > 10000.0 nM | | | NPASS |
| Casein kinase I epsilon | Homo sapiens | P49674 | | > 10000.0 nM | | | NPASS |
| Cyclin-dependent kinase 5/CDK5 activator 1 | Homo sapiens | Q00535|Q15078 | | > 10000.0 nM | | | NPASS |
| DU-145 | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| A549 | Homo sapiens | | | > 50000.0 nM | | | NPASS |
| Dual specificity protein kinase CLK2 | Homo sapiens | P49760 | | > 10000.0 nM | | | NPASS |
| Dual specificity protein kinase CLK3 | Homo sapiens | P49761 | | > 10000.0 nM | | | NPASS |
| Dual specificity protein kinase CLK4 | Homo sapiens | Q9HAZ1 | | > 10000.0 nM | | | NPASS |
| Dual specificity protein kinase CLK1 | Homo sapiens | P49759 | | > 10000.0 nM | | | NPASS |