
| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|---|---|---|---|---|---|---|
| SK-BR-3 | Homo sapiens | = 780.0 nM | NPASS | ||||
| Vero | Chlorocebus aethiops | = 700.0 nM | NPASS | ||||
| Pyruvate kinase isozymes M1/M2 | Homo sapiens | P14618 | = 900.0 nM | NPASS | |||
| PC-3 | Homo sapiens | = 3250.0 nM | NPASS | ||||
| NON-PROTEIN TARGET | = 3840.0 nM | NPASS | |||||
| NIH3T3 | Mus musculus | = 5210.0 nM | NPASS | ||||
| MDA-MB-231 | Homo sapiens | = 4270.0 nM | NPASS | ||||
| MCF7 | Homo sapiens | = 3060.0 nM|= 2400.0 nM|= 2620.0 nM | NPASS | ||||
| SAOS-2 | Homo sapiens | = 2310.0 nM | NPASS | ||||
| K562 | Homo sapiens | = 1300.0 nM|= 1500.0 nM | NPASS | ||||
| HepG2 | Homo sapiens | = 3800.0 nM | NPASS | ||||
| HeLa | Homo sapiens | = 910.0 nM | NPASS | ||||
| HT-29 | Homo sapiens | = 4030.0 nM | NPASS | ||||
| HCT-15 | Homo sapiens | = 1110.0 nM | NPASS | ||||
| Fibroblast | Homo sapiens | = 1500.0 nM|= 1800.0 nM | NPASS | ||||
| DU-145 | Homo sapiens | = 5020.0 nM|= 19900.0 nM | NPASS | ||||
| AU565 | Homo sapiens | = 900.0 nM | NPASS | ||||
| LNCaP | Homo sapiens | = 10740.0 nM | NPASS |