IMPPAT Phytochemical information: 
Alkannin

Alkannin
Bioactivity information
Target nameTarget organismUniProt identifierEC50IC50KdKiSource
SK-BR-3Homo sapiens= 780.0 nMNPASS
VeroChlorocebus aethiops= 700.0 nMNPASS
Pyruvate kinase isozymes M1/M2Homo sapiensP14618= 900.0 nMNPASS
PC-3Homo sapiens= 3250.0 nMNPASS
NON-PROTEIN TARGET= 3840.0 nMNPASS
NIH3T3Mus musculus= 5210.0 nMNPASS
MDA-MB-231Homo sapiens= 4270.0 nMNPASS
MCF7Homo sapiens= 3060.0 nM|= 2400.0 nM|= 2620.0 nMNPASS
SAOS-2Homo sapiens= 2310.0 nMNPASS
K562Homo sapiens= 1300.0 nM|= 1500.0 nMNPASS
HepG2Homo sapiens= 3800.0 nMNPASS
HeLaHomo sapiens= 910.0 nMNPASS
HT-29Homo sapiens= 4030.0 nMNPASS
HCT-15Homo sapiens= 1110.0 nMNPASS
FibroblastHomo sapiens= 1500.0 nM|= 1800.0 nMNPASS
DU-145Homo sapiens= 5020.0 nM|= 19900.0 nMNPASS
AU565Homo sapiens= 900.0 nMNPASS
LNCaPHomo sapiens= 10740.0 nMNPASS