| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| PC-3 | Homo sapiens | | | = 88700.0 nM | | | NPASS |
| NON-PROTEIN TARGET | | | | = 65400.0 nM|= 7000.0 nM|= 6000.0 nM|= 17000.0 nM | | | NPASS |
| Mycobacterium tuberculosis H37Rv | Mycobacterium tuberculosis H37Rv | | | = 1.2 nM | | | NPASS |
| ME-180 | Homo sapiens | | | = 65400.0 nM | | | NPASS |
| M-phase inducer phosphatase 2 | Homo sapiens | P30305 | | 1980 nM | | | BindingDB |
| MDA-MB-231 | Homo sapiens | | | = 7150.0 nM|= 75760.0 nM|= 6150.0 nM|= 75700.0 nM | | | NPASS |
| MCF7 | Homo sapiens | | | = 16500.0 nM|= 13000.0 nM | | | NPASS |
| Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 | Homo sapiens | Q13526 | | 10120 nM|10810 nM|5900 nM|10030 nM|= 10120.0 nM|= 10810.0 nM|= 5900.0 nM|= 10030.0 nM|= 5000.0 nM | | | BindingDB, NPASS |
| LNCaP | Homo sapiens | | | = 13800.0 nM | | | NPASS |
| MDA-MB-453 | Homo sapiens | | | = 27520.0 nM|= 27500.0 nM | | | NPASS |
| Platelet | | | | = 4450.0 nM|= 1180.0 nM | | | NPASS |
| RPMI-8226 | Homo sapiens | | | = 3950.0 nM | | | NPASS |
| Protein disulfide-isomerase A3 | Homo sapiens | P30101 | | = 2400.0 nM | | | NPASS |
| Protein disulfide-isomerase A4 | Homo sapiens | P13667 | | = 3160.0 nM | | | NPASS |
| SARS-CoV-2 | Severe acute respiratory syndrome coronavirus 2 | | | > 20000.0 nM|> 19952.62 nM | | | NPASS |
| SK-MEL-28 | Homo sapiens | | | = 7000.0 nM | | | NPASS |
| Serine/threonine-protein kinase Aurora-A | Homo sapiens | O14965 | | = 50.0 nM | | | NPASS |
| Serine/threonine-protein kinase Aurora-B | Homo sapiens | Q96GD4 | | = 620.0 nM | | | NPASS |
| Transient receptor potential cation channel subfamily A member 1 | Homo sapiens | O75762 | 1700 nM|= 1700.0 nM | | | | BindingDB, NPASS |
| Trypanosoma cruzi | Trypanosoma cruzi | | | = 6510.0 nM | | | NPASS |
| U-87 MG | Homo sapiens | | | = 7450.0 nM | | | NPASS |
| KB 3-1 | Homo sapiens | | | = 26400.0 nM | | | NPASS |
| Protein disulfide-isomerase | Homo sapiens | P07237 | | = 1100.0 nM|= 630.0 nM | | | NPASS |
| KB | Homo sapiens | | | = 6550.0 nM | | | NPASS |
| 5-lipoxygenase | Bos taurus | | | 17000 nM | | | BindingDB |
| Indoleamine 2,3-dioxygenase 1 | Homo sapiens | P14902 | | 1000 nM | | | BindingDB |
| J774.2 | Mus musculus | | | = 13360.0 nM | | | NPASS |
| 3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ | Francisella tularensis | | | 5.4e+3 nM | | | BindingDB |
| A2780 | Homo sapiens | | | = 1400.0 nM | | | NPASS |
| A549 | Homo sapiens | | | = 7000.0 nM|= 11870.0 nM | | | NPASS |
| Amine oxidase | Homo sapiens | | | 4.36e+3 nM | | | BindingDB |
| Amine oxidase [flavin-containing] A | Homo sapiens | P21397 | | 1.71e+3 nM | | | BindingDB |
| Arachidonate 5-lipoxygenase | Bos taurus | Q9BEG3 | | = 17000.0 nM | | | NPASS |
| Aurora kinase A | Homo sapiens | O14965 | | 50 nM | | | BindingDB |
| Aurora kinase B | Homo sapiens | Q96GD4 | | 620 nM | | | BindingDB |
| DNA topoisomerase 1 | Homo sapiens | P11387 | | 8260 nM | | | BindingDB |
| 3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ [1-175] | Yersipestis | B1JQH1 | | 5.3e+3 nM | | | BindingDB |
| DU-145 | Homo sapiens | | | = 11670.0 nM | | | NPASS |
| Dual specificity phosphatase Cdc25B | Homo sapiens | P30305 | | = 1980.0 nM | | | NPASS |
| Dual specificity protein phosphatase 1 | Mus musculus | P28563 | | 13000 nM|= 13000.0 nM | | | BindingDB, NPASS |
| Dual specificity protein phosphatase 6 | Rattus norvegicus | Q64346 | | 12400 nM|= 12400.0 nM | | | BindingDB, NPASS |
| EA.hy 926 | Homo sapiens | | | = 5570.0 nM | | | NPASS |
| HCT-116 | Homo sapiens | | | = 31600.0 nM | | | NPASS |
| HT-29 | Homo sapiens | | | = 7710.0 nM|> 100000.0 nM | | | NPASS |
| HaCaT | Homo sapiens | | | = 800.0 nM | | | NPASS |
| Indoleamine 2,3-dioxygenase | Homo sapiens | P14902 | | = 1000.0 nM | | | NPASS |
| HeLa | Homo sapiens | | | = 68460.0 nM|= 65460.0 nM|= 93700.0 nM|= 15730.0 nM | | | NPASS |
| DNA topoisomerase I | Homo sapiens | P11387 | | = 8260.0 nM | | | NPASS |