IMPPAT Phytochemical information: 
Shikonin

Shikonin
Bioactivity information
Target nameTarget organismUniProt identifierEC50IC50KdKiSource
NCI-H2342Homo sapiens= 134.45 nMNPASS
NCI-H23Homo sapiens= 34982.99 nMNPASS
NCI-H226Homo sapiens= 645.17 nMNPASS
NCI-H2171Homo sapiens= 908.96 nMNPASS
NCI-H2227Homo sapiens= 4886.99 nMNPASS
NCI-H2196Homo sapiens= 654.27 nMNPASS
NCI-H2170Homo sapiens= 1717.23 nMNPASS
NCI-H2228Homo sapiens= 900.95 nMNPASS
NCI-H2347Homo sapiens= 967.81 nMNPASS
NCI-H292= 853.29 nMNPASS
NCI-H2452Homo sapiens= 225928.37 nMNPASS
NCI-H28Homo sapiens= 1008.35 nMNPASS
NCI-H322MHomo sapiens= 32481.64 nMNPASS
NCI-H345Homo sapiens= 989.57 nMNPASS
NCI-H358Homo sapiens= 657.76 nMNPASS
NCI-H441Homo sapiens= 15808.87 nMNPASS
NCI-H2141Homo sapiens= 1711.56 nMNPASS
NCI-H446Homo sapiens= 39554.32 nMNPASS
NCI-H2405Homo sapiens= 674.53 nMNPASS
NCI-H2126Homo sapiens= 15645.4 nMNPASS
NCI-H1882Homo sapiens= 576.09 nMNPASS
NCI-H209Homo sapiens= 12309.4 nMNPASS
NCI-H1694Homo sapiens= 840.09 nMNPASS
NCI-H1703Homo sapiens= 2297.23 nMNPASS
NCI-H1734Homo sapiens= 6895.11 nMNPASS
NCI-H1755Homo sapiens= 30252.11 nMNPASS
NCI-H1770Homo sapiens= 243.14 nMNPASS
NCI-H1792Homo sapiens= 104969.83 nMNPASS
NCI-H1793Homo sapiens= 916685.09 nMNPASS
NCI-H1838Homo sapiens= 22434.84 nMNPASS
NCI-H2122Homo sapiens= 27553.9 nMNPASS
NCI-H187Homo sapiens= 2359.32 nMNPASS
NCI-H1963Homo sapiens= 100.11 nMNPASS
NCI-H1975Homo sapiens= 4280.0 nM|= 4560.0 nMNPASS
NCI-H1993Homo sapiens= 2940.26 nMNPASS
NCI-H2009Homo sapiens= 20.54 nMNPASS
NCI-H2030Homo sapiens= 562.65 nMNPASS
NCI-H2052Homo sapiens= 61.13 nMNPASS
NCI-H2081Homo sapiens= 1524.77 nMNPASS
NCI-H2087Homo sapiens= 440.72 nMNPASS
NCI-H460Homo sapiens= 1277.69 nM|= 5040.0 nM|= 7570.0 nMNPASS
NCI-H510AHomo sapiens= 165511.55 nMNPASS
NCI-H716Homo sapiens= 1136510.63 nMNPASS
NCI-H522Homo sapiens= 559.79 nMNPASS
NOMO-1Homo sapiens= 1155.91 nMNPASS
NON-PROTEIN TARGET= 18100.0 nM|= 670.0 nM|= 1410.0 nM|= 40.0 nMNPASS
NOS-1Homo sapiens= 282233.85 nMNPASS
NTERA-2-cl-D1Homo sapiens= 143.57 nMNPASS
NUGC-3Homo sapiens= 765.43 nMNPASS
NYHomo sapiens= 1045.57 nMNPASS
NeuraminidaseInflueA virus (strain A/Brevig Mission/1/1918 H1N1) (InflueAvirus (strain A/South Carolina/1/1918 H1N1))Q9IGQ6= 34100.0 nMNPASS
OAW-28Homo sapiens= 1198.21 nMNPASS
NMC-G1Homo sapiens= 1297.14 nMNPASS
OAW-42Homo sapiens= 577.68 nMNPASS
OCUB-MHomo sapiens= 865.23 nMNPASS
OE19Homo sapiens= 807.34 nMNPASS
OE33Homo sapiens= 1813.21 nMNPASS
OMC-1Homo sapiens= 1748.88 nMNPASS
ONS-76Homo sapiens= 358.07 nMNPASS
OPM-2Homo sapiens= 343.26 nMNPASS
OS-RC-2Homo sapiens= 313.89 nMNPASS
OVCAR-3Homo sapiens= 382.81 nMNPASS
OCI-AML2Homo sapiens= 298.37 nMNPASS
NKM-1Homo sapiens= 101.2 nMNPASS
NH-12Homo sapiens= 850.19 nMNPASS
NEC8Homo sapiens= 839.9 nMNPASS
NCI-H524Homo sapiens= 998680.59 nMNPASS
NCI-H526Homo sapiens= 2636.52 nMNPASS
NCI-H596= 817.86 nMNPASS
NCI-H630Homo sapiens= 1303.9 nMNPASS
NCI-H64Homo sapiens= 547.1 nMNPASS
NCI-H650Homo sapiens= 665.19 nMNPASS
NCI-H661Homo sapiens= 5428.73 nMNPASS
NCI-H69Homo sapiens= 6713.8 nMNPASS
NCI-H1693Homo sapiens= 66678.0 nMNPASS
NCI-H719Homo sapiens= 2611.26 nMNPASS
NCI-H720Homo sapiens= 1136712.95 nMNPASS
NCI-H727Homo sapiens= 638.3 nMNPASS
NCI-H747Homo sapiens= 441.39 nMNPASS
NCI-H748Homo sapiens= 1782.46 nMNPASS
NCI-H810Homo sapiens= 502.62 nMNPASS
NCI-H82Homo sapiens= 407349.28 nMNPASS
NCI-H838Homo sapiens= 136106.82 nMNPASS
NCI-H889Homo sapiens= 1636835.36 nMNPASS
NCI-N87Homo sapiens= 2942.3 nMNPASS
NCI-H520= 1354.54 nMNPASS
NCI-H1651Homo sapiens= 22750.27 nMNPASS
NCI-H1355Homo sapiens= 2822.51 nMNPASS
NCI-H1648Homo sapiens= 11147.41 nMNPASS
MDA-MB-436Homo sapiens= 3610.0 nMNPASS
MDA-MB-453Homo sapiens= 2518.94 nMNPASS
MDA-MB-468Homo sapiens= 966.84 nM|= 3280.0 nMNPASS
ME-180Homo sapiens= 278.91 nMNPASS
MEG-01Homo sapiens= 451.25 nMNPASS
MEL-HOHomo sapiens= 148.82 nMNPASS
MEL-JUSOHomo sapiens= 540.14 nMNPASS
MES-SAHomo sapiens= 41.32 nMNPASS
MDA-MB-415Homo sapiens= 2276.74 nMNPASS
MFE-280Homo sapiens= 4946.54 nMNPASS
MFH-inoHomo sapiens= 863.85 nMNPASS
MFM-223Homo sapiens= 898.77 nMNPASS
MG-63Homo sapiens= 256.77 nM|= 7360.0 nM|= 5670.0 nMNPASS
MGC-803Homo sapiens= 1510.0 nM|= 1280.0 nMNPASS
MHH-CALL-2Homo sapiens= 715.04 nMNPASS
MHH-ES-1Homo sapiens= 688.56 nMNPASS
MHH-NB-11Homo sapiens= 485.95 nMNPASS
MHH-PREB-1Homo sapiens= 251.57 nMNPASS
MFE-296Homo sapiens= 662.44 nMNPASS
MDA-MB-361Homo sapiens= 1732.36 nMNPASS
MDA-MB-231Homo sapiens= 6600.0 nM|= 1015.44 nM|= 3940.0 nM|= 8750.0 nM|= 6500.0 nM|= 2770.0 nM|= 1580.0 nM|= 108000.0 nM|= 7620.0 nM|= 8980.0 nM|= 2880.0 nMNPASS
MDA-MB-175-VIIHomo sapiens= 2053.07 nMNPASS
OVCAR-4Homo sapiens= 669.55 nMNPASS
LS174THomo sapiens= 8900.0 nMNPASS
LU-134-AHomo sapiens= 809.71 nMNPASS
LU-139Homo sapiens= 6264.09 nMNPASS
LU-165Homo sapiens= 634.05 nMNPASS
LU-99AHomo sapiens= 1295.65 nMNPASS
LXF-289 cell line= 3271.56 nMNPASS
LoVoHomo sapiens= 1335.09 nMNPASS
Lu-65Homo sapiens= 221073.67 nMNPASS
M059JHomo sapiens= 134.19 nMNPASS
M14Homo sapiens= 1492.69 nMNPASS
MC-CARHomo sapiens= 813.62 nMNPASS
MC-IXCHomo sapiens= 387.38 nMNPASS
MC116Homo sapiens= 1786.36 nMNPASS
MCF-10AHomo sapiens= 93400.0 nM|= 23500.0 nM|= 20940.0 nMNPASS
MCF10Homo sapiens= 4560.0 nMNPASS
MCF7Homo sapiens= 1450.0 nM|= 1900.0 nM|= 434.85 nM|= 1800.0 nM|= 5490.0 nM|= 2400.0 nM|= 2700.0 nM|= 6500.0 nM|= 9550.0 nM|= 5400.0 nM|= 23410.0 nM|= 23600.0 nM|= 9320.0 nM|= 4570.0 nM|= 7750.0 nM|= 8320.0 nM|= 1030.0 nM|= 2110.0 nM|= 4990.0 nMNPASS
MDA-MB-134-VIHomo sapiens= 709.4 nMNPASS
MDA-MB-157Homo sapiens= 636.63 nMNPASS
MIA PaCa-2Homo sapiens= 276.49 nMNPASS
NCI-H1650Homo sapiens= 1375.03 nM|= 8320.0 nMNPASS
MKN-1Homo sapiens= 235.76 nMNPASS
MKN-45Homo sapiens= 608.39 nMNPASS
NB13Homo sapiens= 316.93 nMNPASS
NB5Homo sapiens= 2432.63 nMNPASS
NB6Homo sapiens= 454.4 nMNPASS
NB69Homo sapiens= 212.73 nMNPASS
NCCITHomo sapiens= 517.16 nMNPASS
NCI-H1092Homo sapiens= 1393.11 nMNPASS
NCI-H1155Homo sapiens= 1998891.39 nMNPASS
NCI-H1299Homo sapiens= 1071.94 nM|= 1880.0 nM|= 3950.0 nMNPASS
NB12Homo sapiens= 666.31 nMNPASS
NCI-H1304Homo sapiens= 184889.62 nMNPASS
NCI-H1417Homo sapiens= 815.92 nMNPASS
NCI-H1436Homo sapiens= 603.96 nMNPASS
NCI-H1437Homo sapiens= 1557.48 nMNPASS
NCI-H1522Homo sapiens= 519.44 nMNPASS
NCI-H1563Homo sapiens= 626.38 nMNPASS
NCI-H1581Homo sapiens= 89965.84 nMNPASS
NCI-H1618Homo sapiens= 2019.66 nMNPASS
NCI-H1623Homo sapiens= 2727.21 nMNPASS
NCI-H1395Homo sapiens= 971830.1 nMNPASS
NB10Homo sapiens= 1343.65 nMNPASS
NB1Homo sapiens= 1034.34 nMNPASS
NALM-6Homo sapiens= 2.797 nMNPASS
LS-513Homo sapiens= 1477.97 nMNPASS
MKN-7Homo sapiens= 2205.51 nMNPASS
ML-2Homo sapiens= 617.74 nMNPASS
MLMAHomo sapiens= 539.08 nMNPASS
MMAC-SFHomo sapiens= 751.96 nMNPASS
MN-60Homo sapiens= 347.88 nMNPASS
MOLT-16Homo sapiens= 2762.98 nMNPASS
MOLT-4Homo sapiens= 410.12 nMNPASS
MONO-MAC-6Homo sapiens= 244.77 nM|= 2600.0 nMNPASS
MPP-89Homo sapiens= 857.25 nMNPASS
MRK-nu-1Homo sapiens= 101.93 nMNPASS
MS-1Homo sapiens= 1772.48 nMNPASS
MSTO-211HHomo sapiens= 603751.69 nMNPASS
MV4-11Homo sapiens= 273.63 nMNPASS
MZ1-PCHomo sapiens= 19.28 nMNPASS
MZ2-MELHomo sapiens= 385.22 nMNPASS
MZ7-melHomo sapiens= 113.72 nMNPASS
MeWoHomo sapiens= 517.32 nMNPASS
MoHomo sapiens= 819.71 nMNPASS
MKN-28Homo sapiens= 616.87 nMNPASS
OVCAR-5Homo sapiens= 1123.89 nMNPASS
TALL-1Homo sapiens= 754677.12 nMNPASS
P12-IchikawaHomo sapiens= 1388.36 nMNPASS
SW1573Homo sapiens= 371.8 nMNPASS
SW1710Homo sapiens= 2.91 nMNPASS
SW1783Homo sapiens= 1068.84 nMNPASS
SW1990Homo sapiens= 1617.18 nMNPASS
SW48Homo sapiens= 1258.27 nMNPASS
SW626Homo sapiens= 635.13 nMNPASS
SW684Homo sapiens= 777.33 nMNPASS
SW756Homo sapiens= 761.77 nMNPASS
SW1463Homo sapiens= 8606.36 nMNPASS
SW780Homo sapiens= 405.52 nMNPASS
SW872Homo sapiens= 367.48 nM|= 760.0 nMNPASS
SW948Homo sapiens= 11909.0 nMNPASS
SW982Homo sapiens= 60.23 nM|= 2800.0 nMNPASS
SiHaHomo sapiens= 18601.72 nMNPASS
T-24Homo sapiens= 2462.32 nMNPASS
T47DHomo sapiens= 223.06 nMNPASS
T84Homo sapiens= 14520.28 nMNPASS
T98GHomo sapiens= 1082.08 nMNPASS
SW837Homo sapiens= 19784.09 nMNPASS
TCC-SUPHomo sapiens= 554.45 nMNPASS
SW1417Homo sapiens= 825.83 nMNPASS
SW1088Homo sapiens= 699.55 nMNPASS
SNB-75Homo sapiens= 745.95 nMNPASS
SNG-MHomo sapiens= 272.37 nMNPASS
SNU-16Homo sapiens= 5100648.67 nMNPASS
SNU-387Homo sapiens= 1068.57 nMNPASS
SNU-423Homo sapiens= 163.07 nMNPASS
SNU-449Homo sapiens= 813.25 nMNPASS
SNU-475Homo sapiens= 14058.92 nMNPASS
SNU-5Homo sapiens= 9536.71 nMNPASS
SW13Homo sapiens= 1409.19 nMNPASS
SNU-C1Homo sapiens= 722279.37 nMNPASS
SNU1Homo sapiens= 1602.2 nMNPASS
SRHomo sapiens= 140.73 nMNPASS
ST486Homo sapiens= 6.179 nMNPASS
SU-DHL-1Homo sapiens= 499.22 nMNPASS
SUP-T1Homo sapiens= 1822.91 nMNPASS
SW 954Homo sapiens= 466.71 nMNPASS
SW 962Homo sapiens= 568.3 nMNPASS
SW-620Homo sapiens= 358.55 nMNPASS
SNU-C2BHomo sapiens= 24926.79 nMNPASS
TE-1Homo sapiens= 15796.45 nMNPASS
TE-10Homo sapiens= 986.09 nMNPASS
TE-11Homo sapiens= 4014.26 nMNPASS
UACC-62Homo sapiens= 1229.98 nMNPASS
UACC-812Homo sapiens= 5077.15 nMNPASS
UACC-893Homo sapiens= 119208.02 nMNPASS
UMC-11Homo sapiens= 46792.08 nMNPASS
UMUC3Homo sapiens= 967.27 nMNPASS
UO-31Homo sapiens= 770.84 nMNPASS
VA-ES-BJHomo sapiens= 400.58 nMNPASS
VM-CUB-1Homo sapiens= 1028.56 nMNPASS
UACC-257Homo sapiens= 26356.58 nMNPASS
VMRC-RCZHomo sapiens= 546.67 nMNPASS
WM-115Homo sapiens= 10644.2 nMNPASS
WSU-NHLHomo sapiens= 260.33 nMNPASS
YAPCHomo sapiens= 243833.84 nMNPASS
YKG-1Homo sapiens= 228.91 nMNPASS
YTHomo sapiens= 383.89 nMNPASS
no-10Homo sapiens= 290.23 nMNPASS
no-11Homo sapiens= 805.42 nMNPASS
LS-411NHomo sapiens= 3189.61 nMNPASS
VeroChlorocebus sabaeus= 6760.0 nMNPASS
U2OSHomo sapiens= 597438.89 nMNPASS
U-937Homo sapiens= 1200.0 nMNPASS
U-87 MGHomo sapiens= 1275.78 nMNPASS
TE-12Homo sapiens= 2343.25 nMNPASS
TE-15Homo sapiens= 400.31 nMNPASS
TE-441-THomo sapiens= 2.238 nMNPASS
TE-5Homo sapiens= 1004.32 nMNPASS
TE-6Homo sapiens= 2967.91 nMNPASS
TE-8Homo sapiens= 1280.63 nMNPASS
TE-9Homo sapiens= 407.52 nMNPASS
TGBC1TKBHomo sapiens= 1428.19 nMNPASS
TGBC24TKBHomo sapiens= 27882.74 nMNPASS
TGWHomo sapiens= 521.64 nMNPASS
THP-1Homo sapiens= 891.43 nM|= 820.0 nMNPASS
TK-10Homo sapiens= 1224.02 nMNPASS
TTHomo sapiens= 1698.76 nMNPASS
TURHomo sapiens= 465.99 nMNPASS
TYK-nuHomo sapiens= 1152.13 nMNPASS
U-118-MGHomo sapiens= 841.85 nMNPASS
U-251Homo sapiens= 1432.46 nMNPASS
U-266Homo sapiens= 675.16 nMNPASS
U-698-MHomo sapiens= 300.87 nMNPASS
SN12CHomo sapiens= 1762.58 nMNPASS
SKG-IIIaHomo sapiens= 4388.27 nMNPASS
SK-UT-1Homo sapiens= 7.438 nMNPASS
SK-PN-DWHomo sapiens= 36.55 nMNPASS
REHHomo sapiens= 146.96 nMNPASS
RERF-LC-MSHomo sapiens= 4189.97 nMNPASS
RH-1Homo sapiens= 719.88 nMNPASS
RKOHomo sapiens= 270.3 nMNPASS
RLHomo sapiens= 464793.4 nMNPASS
RL95-2Homo sapiens= 719.73 nMNPASS
RMG-IHomo sapiens= 864.23 nMNPASS
RO82-W-1Homo sapiens= 2842.95 nMNPASS
RDHomo sapiens= 449.06 nMNPASS
RPMI 8402Homo sapiens= 1498.31 nMNPASS
RPMI-6666Homo sapiens= 587.13 nMNPASS
RPMI-7951Homo sapiens= 156.09 nMNPASS
RPMI-8226Homo sapiens= 471.88 nMNPASS
RPMI-8866Homo sapiens= 536.04 nMNPASS
RS4-11Homo sapiens= 416.76 nMNPASS
RT-112Homo sapiens= 70.37 nMNPASS
RT-4Homo sapiens= 10121.92 nMNPASS
RVH-421Homo sapiens= 1467.47 nMNPASS
RPMI-2650Homo sapiens= 374.74 nMNPASS
RCM-1Homo sapiens= 2002.19 nMNPASS
RCC10RGBHomo sapiens= 1563.9 nMNPASS
QIMR-WILHomo sapiens= 181.89 nMNPASS
P30-OHKHomo sapiens= 220.48 nMNPASS
P31-FUJHomo sapiens= 2066.09 nMNPASS
PA-1Homo sapiens= 201.28 nM|= 920.0 nMNPASS
PANC-03-27Homo sapiens= 167.4 nMNPASS
PANC-08-13Homo sapiens= 10430.49 nMNPASS
PBMCHomo sapiens= 5000.0 nMNPASS
PC-14Homo sapiens= 1507.16 nMNPASS
PC-3Homo sapiens= 858.79 nMNPASS
PF-382Homo sapiens= 789.51 nMNPASS
PFSK-1Homo sapiens= 76572.12 nMNPASS
PLC-PRF-5Homo sapiens= 1815.79 nMNPASS
PSN1Homo sapiens= 71023.8 nMNPASS
Panc1005Homo sapiens= 415.63 nMNPASS
Plasmodium bergheiPlasmodium berghei= 1370.0 nMNPASS
Plasmodium falciparumPlasmodium falciparum> 5000.0 nMNPASS
Protein-tyrosine phosphatase 1Saccharomyces cerevisiae S288cP25044= 70000.0 nMNPASS
Protein-tyrosine phosphatase 1BHomo sapiensP18031= 25000.0 nMNPASS
Pyruvate kinase isozymes M1/M2Homo sapiensP14618= 12960.0 nM|= 8820.0 nM|= 10000.0 nM|= 500.0 nM|= 1520.0 nM|= 381.0 nM|= 326.0 nM|> 10000.0 nM|= 800.0 nM|= 301.0 nM|= 1420.0 nM|= 2576.0 nMNPASS
Pyruvate kinase isozymes R/LHomo sapiensP30613= 39250.0 nMNPASS
RXF 393Homo sapiens= 749.01 nMNPASS
OVCAR-8Homo sapiens= 460.05 nMNPASS
RajiHomo sapiens= 631.17 nMNPASS
Replicase polyprotein 1abSevere acute respiratory syndrome coronavirus 2P0DTD1= 15750.0 nM|= 15739.83 nM|= 1600.0 nM|= 670.0 nMNPASS
SK-BR-3Homo sapiens= 3750.0 nMNPASS
SK-CO-1Homo sapiens= 2054.9 nMNPASS
SK-HEP1Homo sapiens= 547.51 nMNPASS
SK-LMS-1Homo sapiens= 108.41 nMNPASS
SK-LU-1Homo sapiens= 750.1 nMNPASS
SK-MEL-1Homo sapiens= 138410.24 nMNPASS
SK-MEL-2Homo sapiens= 6328.9 nMNPASS
SK-MEL-24Homo sapiens= 1133.44 nMNPASS
SJSA-1Homo sapiens= 5525.33 nMNPASS
SK-MEL-28Homo sapiens= 277189.39 nMNPASS
SK-MEL3Homo sapiens= 2642.21 nMNPASS
SK-MES-1Homo sapiens= 6286.32 nMNPASS
SK-MM-2Homo sapiens= 498.97 nMNPASS
SK-N-ASHomo sapiens= 1786.2 nMNPASS
SK-N-DZHomo sapiens= 1803.2 nMNPASS
SK-N-FIHomo sapiens= 7693.54 nMNPASS
SK-NEP-1Homo sapiens= 1081.12 nMNPASS
SK-OV-3Homo sapiens= 1560.3 nM|= 3460.0 nMNPASS
SK-MEL-30Homo sapiens= 694.8 nMNPASS
SJRH30Homo sapiens= 369.2 nMNPASS
SIMAHomo sapiens= 2318.43 nMNPASS
SIG-M5Homo sapiens= 169.86 nMNPASS
S-117Homo sapiens= 387.1 nMNPASS
SAOS-2Homo sapiens= 2367.35 nMNPASS
SARS-CoV-2Severe acute respiratory syndrome coronavirus 2> 20000.0 nM|> 19952.62 nM|= 670.0 nMNPASS
SASHomo sapiens= 853.74 nMNPASS
SBC-1Homo sapiens= 12149.22 nMNPASS
SBC-5Homo sapiens= 215.46 nMNPASS
SCC-15Homo sapiens= 650.5 nMNPASS
SCC-25Homo sapiens= 382.64 nMNPASS
SCC-3Homo sapiens= 1003.43 nMNPASS
SCC-4Homo sapiens= 440.6 nM|= 10100.0 nMNPASS
SCC-9Homo sapiens= 196.75 nMNPASS
SCHHomo sapiens= 195008.47 nMNPASS
SCLC-21HHomo sapiens= 1364.86 nMNPASS
SF-126Homo sapiens= 772.97 nMNPASS
SF-268Homo sapiens= 5577.43 nMNPASS
SF-295Homo sapiens= 664.18 nMNPASS
SF-539Homo sapiens= 856.82 nMNPASS
SH-4Homo sapiens= 371.35 nMNPASS
SHP77Homo sapiens= 445.54 nMNPASS
Ramos-2G6-4C10Homo sapiens= 315.03 nMNPASS
LS-123Homo sapiens= 537.66 nMNPASS
COLO-320-HSRHomo sapiens= 384.48 nMNPASS
LP-1Homo sapiens= 686.37 nMNPASS
CP66-MELHomo sapiens= 2396.67 nMNPASS
CPC-NHomo sapiens= 24262.4 nMNPASS
CTB-1Homo sapiens= 859.02 nMNPASS
CTV-1Homo sapiens= 32752.88 nMNPASS
CW-2Homo sapiens= 676152.07 nMNPASS
CWR22RHomo sapiens= 4614.94 nMNPASS
Ca-SkiHomo sapiens= 650.31 nMNPASS
Ca9-22Homo sapiens= 580.63 nM|= 12810.0 nM|= 13590.0 nMNPASS
CP50-MEL-BHomo sapiens= 1433.36 nMNPASS
CaR-1Homo sapiens= 1308.43 nMNPASS
Calu-3Homo sapiens= 1108.34 nM|= 7220.0 nMNPASS
Calu-6Homo sapiens= 15732.0 nMNPASS
Caov-3 cell line= 766.5 nMNPASS
Caov-4Homo sapiens= 1884.19 nMNPASS
Capan-2Homo sapiens= 1005.29 nMNPASS
ChaGo-K-1Homo sapiens= 656.72 nMNPASS
D-247MGHomo sapiens= 1660.02 nMNPASS
D-263MGHomo sapiens= 2230.07 nMNPASS
Calu-1Homo sapiens= 1232.12 nMNPASS
D-336MGHomo sapiens= 1749.77 nMNPASS
COR-L88Homo sapiens= 109652.36 nMNPASS
COR-L23Homo sapiens= 301.5 nMNPASS
CGTH-W-1Homo sapiens= 499.93 nMNPASS
CHL-1Homo sapiens= 167.8 nMNPASS
CHP-126Homo sapiens= 695.35 nMNPASS
CHP-212Homo sapiens= 1096.47 nMNPASS
CMKHomo sapiens= 352.13 nMNPASS
CNEHomo sapiens= 700.0 nMNPASS
COLO 205Homo sapiens= 537.72 nMNPASS
COLO-668Homo sapiens= 6196.13 nMNPASS
COR-L279Homo sapiens= 188288.43 nMNPASS
COLO-678Homo sapiens= 1628.64 nMNPASS
COLO-680NHomo sapiens= 590.03 nMNPASS
COLO-684Homo sapiens= 400.53 nMNPASS
COLO-741Homo sapiens= 2694.21 nMNPASS
COLO-792Homo sapiens= 81952.6 nMNPASS
COLO-800Homo sapiens= 3260066.91 nMNPASS
COLO-824Homo sapiens= 715.2 nMNPASS
COLO-829Homo sapiens= 657.99 nMNPASS
COR-L105Homo sapiens= 230.34 nMNPASS
COLO-679Homo sapiens= 184.01 nMNPASS
D-392MGHomo sapiens= 915.29 nMNPASS
D-502MGHomo sapiens= 4365.48 nMNPASS
D-542MGHomo sapiens= 580.88 nMNPASS
DoTc2-4510Homo sapiens= 262.79 nMNPASS
Dual specificity phosphatase Cdc25AHomo sapiensP30304= 220.0 nM|= 2140.0 nMNPASS
Dual specificity phosphatase Cdc25BHomo sapiensP30305= 400.0 nM|= 5820.0 nMNPASS
Dual specificity phosphatase Cdc25CHomo sapiensP30307= 4780.0 nMNPASS
EB-3Homo sapiens= 1142.2 nMNPASS
EB2Homo sapiens= 310.95 nMNPASS
EC-GI-10Homo sapiens= 57446.9 nMNPASS
ECC12Homo sapiens= 9648.24 nMNPASS
Detroit562Homo sapiens= 29295.97 nMNPASS
ECC4Homo sapiens= 1203.45 nMNPASS
EFO-21Homo sapiens= 1338.59 nMNPASS
EFO-27Homo sapiens= 330.34 nMNPASS
EGI-1Homo sapiens= 2511.08 nMNPASS
EHEBHomo sapiens= 2094.47 nMNPASS
EKVXHomo sapiens= 3674.07 nMNPASS
EM-2Homo sapiens= 976.93 nMNPASS
EOL1Homo sapiens= 508.75 nMNPASS
ES1Homo sapiens= 502.89 nMNPASS
EFM-19Homo sapiens= 212.1 nMNPASS
DaudiHomo sapiens= 3442.87 nMNPASS
DaoyHomo sapiens= 158.77 nMNPASS
DV-90Homo sapiens= 206842.58 nMNPASS
D283 Med= 835.31 nMNPASS
DBHomo sapiens= 726.29 nMNPASS
DBTRG-05MGHomo sapiens= 611.1 nMNPASS
DELHomo sapiens= 153.81 nMNPASS
DG-75Homo sapiens= 1167.49 nMNPASS
DJM-1Homo sapiens= 6387.23 nMNPASS
DK-MGHomo sapiens= 9817.5 nMNPASS
DMS-114Homo sapiens= 35541.18 nMNPASS
DMS-153Homo sapiens= 27808.34 nMNPASS
DMS-273Homo sapiens= 395.79 nMNPASS
DMS-53Homo sapiens= 21456.74 nMNPASS
DMS-79Homo sapiens= 271650.96 nMNPASS
DNA topoisomerase IHomo sapiensP11387= 208000.0 nMNPASS
DNA topoisomerase IIHomo sapiensQ02880= 6200.0 nM|= 6700.0 nM|= 16000.0 nM|= 12500.0 nM|= 5700.0 nM|= 7800.0 nMNPASS
DOHH-2Homo sapiens= 706.26 nMNPASS
DOKHomo sapiens= 5185.18 nMNPASS
DSH1Homo sapiens= 10584.2 nMNPASS
DU-145Homo sapiens= 193.09 nM|= 16000.0 nMNPASS
DU-4475Homo sapiens= 179.84 nMNPASS
CESSHomo sapiens= 776.45 nMNPASS
ES3Homo sapiens= 656.49 nMNPASS
CCRF-CEMHomo sapiens= 567.02 nMNPASS
CAS-1Homo sapiens= 462.11 nMNPASS
A4-FukHomo sapiens= 249.73 nMNPASS
A498Homo sapiens= 81.9 nMNPASS
A549Homo sapiens= 3530.0 nM|= 7300.0 nM|= 6500.0 nM|= 6130.0 nM|= 10250.0 nM|= 5060.0 nM|= 10370.0 nM|= 1708.0 nM|= 3130.0 nM|= 11680.0 nM|= 7730.0 nM|= 1800.0 nM|= 4470.0 nM|= 3370.0 nM|= 2510.0 nMNPASS
A673Homo sapiens= 1220.48 nMNPASS
A704Homo sapiens= 2704.66 nMNPASS
ABC-1Homo sapiens= 707.48 nMNPASS
ACHNHomo sapiens= 146.38 nMNPASS
ACNHomo sapiens= 916.95 nMNPASS
A388Homo sapiens= 866.56 nMNPASS
AGSHomo sapiens= 612.57 nMNPASS
AM-38Homo sapiens= 96.31 nMNPASS
AN3-CAHomo sapiens= 79.65 nMNPASS
ARH-77Homo sapiens= 873.49 nMNPASS
ASPC1Homo sapiens= 618.87 nMNPASS
ATN-1Homo sapiens= 849.13 nMNPASS
AU565Homo sapiens= 1239.81 nMNPASS
Acyl coenzyme A:cholesterol acyltransferase 1Homo sapiensP35610= 70400.0 nMNPASS
Acyl coenzyme A:cholesterol acyltransferase 2Homo sapiensO75908= 138200.0 nMNPASS
ALL-POHomo sapiens= 315.12 nMNPASS
B16-F10Mus musculus= 17900.0 nM|= 3720.0 nMNPASS
A3-KAWHomo sapiens= 2140.29 nMNPASS
A253 cell line= 7.493 nMNPASS
LS-1034Homo sapiens= 2747.15 nMNPASS
23132-87Homo sapiens= 2108.3 nMNPASS
5637Homo sapiens= 206270.21 nMNPASS
639-VHomo sapiens= 265.01 nMNPASS
647-VHomo sapiens= 358.52 nMNPASS
697Homo sapiens= 875.65 nMNPASS
769-PHomo sapiens= 688.6 nMNPASS
786-0Homo sapiens= 343.75 nMNPASS
A2780Homo sapiens= 2562.45 nM|= 390.0 nMNPASS
8-MG-BAHomo sapiens= 85.56 nMNPASS
8505CHomo sapiens= 3099.47 nMNPASS
A-375Homo sapiens= 311.11 nMNPASS
A-427Homo sapiens= 17.99 nMNPASS
A-431Homo sapiens= 106.97 nMNPASS
A101DHomo sapiens= 0.7121 nMNPASS
A172Homo sapiens= 469.75 nMNPASS
A204Homo sapiens= 126.54 nMNPASS
A2058Homo sapiens= 919.12 nMNPASS
8305CHomo sapiens= 304.84 nMNPASS
BB30-HNCHomo sapiens= 243.49 nMNPASS
BB49-HNCHomo sapiens= 38584.67 nMNPASS
BB65-RCCHomo sapiens= 695.45 nMNPASS
C32Homo sapiens= 2677.89 nMNPASS
C3AHomo sapiens= 657.06 nMNPASS
C8166Homo sapiens= 407.51 nMNPASS
CA46Homo sapiens= 191.85 nMNPASS
CAKI-1Homo sapiens= 894.13 nMNPASS
CAL-120Homo sapiens= 1360.85 nMNPASS
CAL-12THomo sapiens= 1902.22 nMNPASS
CAL-148Homo sapiens= 676.6 nMNPASS
C2BBe1Homo sapiens= 755.64 nMNPASS
CAL-27Homo sapiens= 83274.14 nMNPASS
CAL-39Homo sapiens= 483.23 nMNPASS
CAL-51Homo sapiens= 20.85 nMNPASS
CAL-54Homo sapiens= 1419.9 nMNPASS
CAL-62Homo sapiens= 1279.99 nMNPASS
CAL-72Homo sapiens= 1012.93 nMNPASS
CAL-85-1Homo sapiens= 160.73 nMNPASS
CAMA-1Homo sapiens= 1516.69 nMNPASS
CAPAN-1Homo sapiens= 758.89 nMNPASS
CAL-33Homo sapiens= 2000.04 nMNPASS
C-4-IIHomo sapiens= 587.72 nMNPASS
C-33-AHomo sapiens= 912.75 nMNPASS
Bel-7402Homo sapiens= 54500.0 nM|= 1240.0 nMNPASS
BC-3Homo sapiens= 926.19 nMNPASS
BC1 cell line= 2681.4 nMNPASS
BCPAPHomo sapiens= 922.59 nMNPASS
BE-13Homo sapiens= 1195.23 nMNPASS
BEAS-2BHomo sapiens= 5360.0 nMNPASS
BENHomo sapiens= 813.72 nMNPASS
BFTC-905Homo sapiens= 283.61 nMNPASS
BFTC-909Homo sapiens= 3627.83 nMNPASS
BHT-101Homo sapiens= 1250.23 nMNPASS
BHYHomo sapiens= 563.96 nMNPASS
BL-41Homo sapiens= 483.4 nMNPASS
BL-70Homo sapiens= 278.02 nMNPASS
BOKUHomo sapiens= 1874.88 nMNPASS
BPH-1Homo sapiens= 1259.99 nMNPASS
BT-20Homo sapiens= 2561.3 nMNPASS
BT-474Homo sapiens= 208.36 nM|= 5740.0 nMNPASS
BV-173Homo sapiens= 435.95 nMNPASS
BXPC-3Homo sapiens= 333.58 nMNPASS
BeckerHomo sapiens= 1582.22 nMNPASS
CCF-STTG1Homo sapiens= 768.01 nMNPASS
ES4Homo sapiens= 4634.59 nMNPASS
EFE-184Homo sapiens= 543.94 nMNPASS
ES6Homo sapiens= 7878.52 nMNPASS
JVM-3Homo sapiens= 913180.9 nMNPASS
JurkatHomo sapiens= 970.0 nMNPASS
K052Homo sapiens= 1098.89 nMNPASS
K5Homo sapiens= 734.38 nMNPASS
K562Homo sapiens= 630.0 nM|= 600.0 nM|= 106057.88 nM|= 700.0 nM|= 1020.0 nM|= 20290.0 nM|= 120540.0 nMNPASS
KALS-1Homo sapiens= 1317.29 nMNPASS
KARPAS-299Homo sapiens= 799.41 nMNPASS
KARPAS-422Homo sapiens= 26611.7 nMNPASS
JVM-2Homo sapiens= 3868.13 nMNPASS
KARPAS-45Homo sapiens= 9989.05 nMNPASS
KG-1= 1597.73 nMNPASS
KGNHomo sapiens= 1307.27 nMNPASS
KINGS-1Homo sapiens= 14077.46 nMNPASS
KLEHomo sapiens= 684.66 nMNPASS
KM-H2Homo sapiens= 1036.17 nMNPASS
KM12Homo sapiens= 739.71 nMNPASS
KMOE-2Homo sapiens= 1240.66 nMNPASS
KMS-12-PEHomo sapiens= 559.38 nMNPASS
KE-37Homo sapiens= 244.45 nMNPASS
JIYOYEHomo sapiens= 1387.92 nMNPASS
JEG-3Homo sapiens= 3171.65 nMNPASS
JARHomo sapiens= 3262.95 nMNPASS
HuCCT-1Homo sapiens= 483.02 nMNPASS
HuO-3N1Homo sapiens= 4433.41 nMNPASS
HuO9Homo sapiens= 1658.0 nMNPASS
HuP-T3Homo sapiens= 833.73 nMNPASS
HuP-T4Homo sapiens= 1361.78 nMNPASS
HuTu80Homo sapiens= 370.2 nMNPASS
Huh-7Homo sapiens= 1955.26 nMNPASS
IA-LMHomo sapiens= 2080.5 nMNPASS
ES5Homo sapiens= 2634.45 nMNPASS
IGROV-1Homo sapiens= 55.61 nMNPASS
IM-9Homo sapiens= 3412.07 nMNPASS
IMR-5Homo sapiens= 589.4 nMNPASS
IPC-298Homo sapiens= 557135.23 nMNPASS
IST-MEL1Homo sapiens= 14955.39 nMNPASS
IST-MES1Homo sapiens= 1696.61 nMNPASS
IST-SL1Homo sapiens= 65198.14 nMNPASS
IST-SL2Homo sapiens= 200.14 nMNPASS
J-RT3-T3-5Homo sapiens= 2086.36 nMNPASS
J82Homo sapiens= 142.55 nMNPASS
KNS-42Homo sapiens= 18658.43 nMNPASS
Hs-578THomo sapiens= 6223.4 nMNPASS
KNS-81-FDHomo sapiens= 1081.94 nMNPASS
KP-4Homo sapiens= 500.8 nMNPASS
LB1047-RCCHomo sapiens= 302.44 nMNPASS
LB2241-RCCHomo sapiens= 1288.29 nMNPASS
LB2518-MELHomo sapiens= 3283.31 nMNPASS
LB373-MEL-DHomo sapiens= 390.74 nMNPASS
LB647-SCLCHomo sapiens= 232.78 nMNPASS
LB771-HNCHomo sapiens= 20788.0 nMNPASS
LB831-BLCHomo sapiens= 1916.8 nMNPASS
LB996-RCCHomo sapiens= 191158.51 nMNPASS
LAN-6Homo sapiens= 3219.16 nMNPASS
LC-1FHomo sapiens= 409800.31 nMNPASS
LC4-1Homo sapiens= 360.29 nMNPASS
LCLC-103H cell line= 345.6 nMNPASS
LCLC-97TM1Homo sapiens= 613.12 nMNPASS
LK-2Homo sapiens= 8570.71 nMNPASS
LN-405Homo sapiens= 6914.68 nMNPASS
LNCaP-Clone-FGCHomo sapiens= 41593.88 nMNPASS
LOUCYHomo sapiens= 586.06 nMNPASS
LOX IMVIHomo sapiens= 411.85 nMNPASS
LC-2-adHomo sapiens= 952.55 nMNPASS
LAMA-84Homo sapiens= 1209.53 nMNPASS
L929Mus musculus= 3200.0 nMNPASS
L02Homo sapiens= 3410.0 nM|= 13000.0 nM|= 6220.0 nM|= 65340.0 nM|= 3257.0 nM|= 5120.0 nM|= 10520.0 nM|= 10450.0 nM|= 83800.0 nMNPASS
KP-N-YSHomo sapiens= 351.7 nMNPASS
KS-1Homo sapiens= 41.5 nMNPASS
KU-19-19Homo sapiens= 3183.07 nMNPASS
KU812 cell line= 8.306 nMNPASS
KURAMOCHIHomo sapiens= 3159.36 nMNPASS
KY821Homo sapiens= 746.85 nMNPASS
KYSE-140Homo sapiens= 373.93 nMNPASS
KYSE-150 cell line= 901.94 nMNPASS
KYSE-180Homo sapiens= 1010.32 nMNPASS
KYSE-270Homo sapiens= 216.92 nMNPASS
KYSE-410Homo sapiens= 752.42 nMNPASS
KYSE-450Homo sapiens= 138.15 nMNPASS
KYSE-510Homo sapiens= 252.7 nMNPASS
KYSE-520 cell line= 598.42 nMNPASS
KYSE-70 cell line= 2415.66 nMNPASS
Kasumi 1= 123.71 nMNPASS
L-363Homo sapiens= 75850.1 nMNPASS
L-428Homo sapiens= 1205.02 nMNPASS
L-540Homo sapiens= 4900.04 nMNPASS
KOSC-2Homo sapiens= 1490.84 nMNPASS
Histone-lysine N-methyltransferase SETD7Homo sapiensQ8WTS6= 21620.0 nMNPASS
IGR-1Homo sapiens= 153.98 nMNPASS
HeLaHomo sapiens= 13390.0 nM|= 6420.0 nM|= 2450.0 nM|= 6860.0 nM|= 6500.0 nM|= 7840.0 nM|= 2818.0 nM|= 11070.0 nM|= 5750.0 nM|= 6440.0 nM|= 4800.0 nM|= 9230.0 nM|= 3110.0 nMNPASS
GCIYHomo sapiens= 35.98 nMNPASS
GCTHomo sapiens= 1151.53 nMNPASS
GDM-1Homo sapiens= 2676.06 nMNPASS
GI-1Homo sapiens= 568.29 nMNPASS
GI-ME-NHomo sapiens= 551.75 nMNPASS
GMS-10Homo sapiens= 11494.56 nMNPASS
GOTOHomo sapiens= 4588.35 nMNPASS
GP5dHomo sapiens= 1337.76 nMNPASS
GB-1Homo sapiens= 1329.99 nMNPASS
HepG2Homo sapiens= 240.0 nM|= 28100.0 nM|= 6920.0 nM|= 2920.0 nM|= 920.0 nM|= 2730.0 nM|= 1288.0 nM|= 9360.0 nM|= 420.0 nMNPASS
H4Homo sapiens= 283.93 nMNPASS
HAL-01Homo sapiens= 195.73 nMNPASS
HC-1Homo sapiens= 17215.51 nMNPASS
HCC 2998Homo sapiens= 46035.14 nMNPASS
HCC1143Homo sapiens= 529.69 nMNPASS
HCC1187Homo sapiens= 1019.79 nMNPASS
HCC1395Homo sapiens= 15686.74 nMNPASS
HCC1419Homo sapiens= 1689.76 nMNPASS
GT3TKBHomo sapiens= 345.5 nMNPASS
GAMGHomo sapiens= 1709.71 nMNPASS
GAKHomo sapiens= 1037.69 nMNPASS
G-402Homo sapiens= 881.67 nMNPASS
ES7Homo sapiens= 548.49 nMNPASS
ES8Homo sapiens= 777.79 nMNPASS
ESS-1Homo sapiens= 34139.91 nMNPASS
ETK-1Homo sapiens= 2445.68 nMNPASS
EVSA-THomo sapiens= 409.8 nMNPASS
EW-1Homo sapiens= 843.9 nMNPASS
EW-11Homo sapiens= 447.16 nMNPASS
EW-13Homo sapiens= 266.74 nMNPASS
EW-16Homo sapiens= 299.15 nMNPASS
EW-18Homo sapiens= 528.62 nMNPASS
EW-24Homo sapiens= 14592.71 nMNPASS
EW-3Homo sapiens= 721.5 nMNPASS
EW-7Homo sapiens= 1290.91 nMNPASS
Epidermal growth factor receptor erbB1Homo sapiensP00533= 139.2 nMNPASS
FTC-133Homo sapiens= 5743.15 nMNPASS
FaDuHomo sapiens= 1766.39 nMNPASS
FibroblastHomo sapiens= 1200.0 nM|= 1240.0 nMNPASS
G-361Homo sapiens= 473.21 nMNPASS
G-401Homo sapiens= 234.92 nMNPASS
HCC1569Homo sapiens= 809.94 nMNPASS
HCC1599Homo sapiens= 388.27 nMNPASS
GR-STHomo sapiens= 102.18 nMNPASS
HCC1937Homo sapiens= 1662.86 nMNPASS
HNHomo sapiens= 1367.64 nMNPASS
HO-1-N-1Homo sapiens= 462.12 nMNPASS
HOP-62Homo sapiens= 1160.87 nMNPASS
HOP-92Homo sapiens= 2010.24 nMNPASS
HOSHomo sapiens= 186.08 nMNPASS
HPAF-IIHomo sapiens= 1266.25 nMNPASS
HSC-2Homo sapiens= 223.18 nMNPASS
HSC-3Homo sapiens= 336.66 nMNPASS
HMV-2 cell line= 56.4 nMNPASS
HSC-4Homo sapiens= 2118.83 nMNPASS
HT-1080Homo sapiens= 259.95 nMNPASS
HT-1376Homo sapiens= 915.31 nMNPASS
HT-144Homo sapiens= 561.17 nMNPASS
HT-29Homo sapiens= 16700.0 nM|= 15800.0 nM|= 644.57 nM|= 2800.0 nMNPASS
HT-3Homo sapiens= 948.27 nMNPASS
HT1197Homo sapiens= 275.82 nMNPASS
HT55Homo sapiens= 1689.62 nMNPASS
HTC-C3Homo sapiens= 542.37 nMNPASS
HCC1806Homo sapiens= 1270.34 nMNPASS
HLEHomo sapiens= 88.31 nMNPASS
HTHomo sapiens= 1087.45 nMNPASS
HHHomo sapiens= 1117.63 nMNPASS
HCC2157Homo sapiens= 337.83 nMNPASS
HCC2218Homo sapiens= 496.03 nMNPASS
HCC38Homo sapiens= 786.51 nMNPASS
HCC70Homo sapiens= 2008.36 nMNPASS
HCC827Homo sapiens= 9210.0 nMNPASS
HCE-4Homo sapiens= 388.84 nMNPASS
HCE-THomo sapiens= 720.09 nMNPASS
HL-60Homo sapiens= 440.0 nM|= 1030.0 nM|= 1923.05 nM|= 1200.0 nMNPASS
HCC1954Homo sapiens= 901.82 nMNPASS
HCT-116Homo sapiens= 230.0 nM|= 386.26 nM|= 1840.0 nM|= 2470.0 nMNPASS
HCT-8Homo sapiens= 9200.0 nMNPASS
HD-MY-ZHomo sapiens= 470.14 nMNPASS
HDLM-2Homo sapiens= 89557.42 nMNPASS
HEC-1Homo sapiens= 1134.41 nMNPASS
HEK-293THomo sapiens= 62760.0 nM|= 1520.0 nM|= 2630.0 nM|= 9270.0 nMNPASS
HELHomo sapiens= 2043.04 nMNPASS
HFF-1Homo sapiens< 5000.0 nMNPASS
HGC-27Homo sapiens= 228.34 nMNPASS
HCT-15Homo sapiens= 7300.0 nM|= 267.58 nM|= 860.0 nM|= 940.0 nMNPASS