| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| NCI-H2342 | Homo sapiens | | | = 134.45 nM | | | NPASS |
| NCI-H23 | Homo sapiens | | | = 34982.99 nM | | | NPASS |
| NCI-H226 | Homo sapiens | | | = 645.17 nM | | | NPASS |
| NCI-H2171 | Homo sapiens | | | = 908.96 nM | | | NPASS |
| NCI-H2227 | Homo sapiens | | | = 4886.99 nM | | | NPASS |
| NCI-H2196 | Homo sapiens | | | = 654.27 nM | | | NPASS |
| NCI-H2170 | Homo sapiens | | | = 1717.23 nM | | | NPASS |
| NCI-H2228 | Homo sapiens | | | = 900.95 nM | | | NPASS |
| NCI-H2347 | Homo sapiens | | | = 967.81 nM | | | NPASS |
| NCI-H292 | | | | = 853.29 nM | | | NPASS |
| NCI-H2452 | Homo sapiens | | | = 225928.37 nM | | | NPASS |
| NCI-H28 | Homo sapiens | | | = 1008.35 nM | | | NPASS |
| NCI-H322M | Homo sapiens | | | = 32481.64 nM | | | NPASS |
| NCI-H345 | Homo sapiens | | | = 989.57 nM | | | NPASS |
| NCI-H358 | Homo sapiens | | | = 657.76 nM | | | NPASS |
| NCI-H441 | Homo sapiens | | | = 15808.87 nM | | | NPASS |
| NCI-H2141 | Homo sapiens | | | = 1711.56 nM | | | NPASS |
| NCI-H446 | Homo sapiens | | | = 39554.32 nM | | | NPASS |
| NCI-H2405 | Homo sapiens | | | = 674.53 nM | | | NPASS |
| NCI-H2126 | Homo sapiens | | | = 15645.4 nM | | | NPASS |
| NCI-H1882 | Homo sapiens | | | = 576.09 nM | | | NPASS |
| NCI-H209 | Homo sapiens | | | = 12309.4 nM | | | NPASS |
| NCI-H1694 | Homo sapiens | | | = 840.09 nM | | | NPASS |
| NCI-H1703 | Homo sapiens | | | = 2297.23 nM | | | NPASS |
| NCI-H1734 | Homo sapiens | | | = 6895.11 nM | | | NPASS |
| NCI-H1755 | Homo sapiens | | | = 30252.11 nM | | | NPASS |
| NCI-H1770 | Homo sapiens | | | = 243.14 nM | | | NPASS |
| NCI-H1792 | Homo sapiens | | | = 104969.83 nM | | | NPASS |
| NCI-H1793 | Homo sapiens | | | = 916685.09 nM | | | NPASS |
| NCI-H1838 | Homo sapiens | | | = 22434.84 nM | | | NPASS |
| NCI-H2122 | Homo sapiens | | | = 27553.9 nM | | | NPASS |
| NCI-H187 | Homo sapiens | | | = 2359.32 nM | | | NPASS |
| NCI-H1963 | Homo sapiens | | | = 100.11 nM | | | NPASS |
| NCI-H1975 | Homo sapiens | | | = 4280.0 nM|= 4560.0 nM | | | NPASS |
| NCI-H1993 | Homo sapiens | | | = 2940.26 nM | | | NPASS |
| NCI-H2009 | Homo sapiens | | | = 20.54 nM | | | NPASS |
| NCI-H2030 | Homo sapiens | | | = 562.65 nM | | | NPASS |
| NCI-H2052 | Homo sapiens | | | = 61.13 nM | | | NPASS |
| NCI-H2081 | Homo sapiens | | | = 1524.77 nM | | | NPASS |
| NCI-H2087 | Homo sapiens | | | = 440.72 nM | | | NPASS |
| NCI-H460 | Homo sapiens | | | = 1277.69 nM|= 5040.0 nM|= 7570.0 nM | | | NPASS |
| NCI-H510A | Homo sapiens | | | = 165511.55 nM | | | NPASS |
| NCI-H716 | Homo sapiens | | | = 1136510.63 nM | | | NPASS |
| NCI-H522 | Homo sapiens | | | = 559.79 nM | | | NPASS |
| NOMO-1 | Homo sapiens | | | = 1155.91 nM | | | NPASS |
| NON-PROTEIN TARGET | | | | = 18100.0 nM|= 670.0 nM|= 1410.0 nM|= 40.0 nM | | | NPASS |
| NOS-1 | Homo sapiens | | | = 282233.85 nM | | | NPASS |
| NTERA-2-cl-D1 | Homo sapiens | | | = 143.57 nM | | | NPASS |
| NUGC-3 | Homo sapiens | | | = 765.43 nM | | | NPASS |
| NY | Homo sapiens | | | = 1045.57 nM | | | NPASS |
| Neuraminidase | InflueA virus (strain A/Brevig Mission/1/1918 H1N1) (InflueAvirus (strain A/South Carolina/1/1918 H1N1)) | Q9IGQ6 | | = 34100.0 nM | | | NPASS |
| OAW-28 | Homo sapiens | | | = 1198.21 nM | | | NPASS |
| NMC-G1 | Homo sapiens | | | = 1297.14 nM | | | NPASS |
| OAW-42 | Homo sapiens | | | = 577.68 nM | | | NPASS |
| OCUB-M | Homo sapiens | | | = 865.23 nM | | | NPASS |
| OE19 | Homo sapiens | | | = 807.34 nM | | | NPASS |
| OE33 | Homo sapiens | | | = 1813.21 nM | | | NPASS |
| OMC-1 | Homo sapiens | | | = 1748.88 nM | | | NPASS |
| ONS-76 | Homo sapiens | | | = 358.07 nM | | | NPASS |
| OPM-2 | Homo sapiens | | | = 343.26 nM | | | NPASS |
| OS-RC-2 | Homo sapiens | | | = 313.89 nM | | | NPASS |
| OVCAR-3 | Homo sapiens | | | = 382.81 nM | | | NPASS |
| OCI-AML2 | Homo sapiens | | | = 298.37 nM | | | NPASS |
| NKM-1 | Homo sapiens | | | = 101.2 nM | | | NPASS |
| NH-12 | Homo sapiens | | | = 850.19 nM | | | NPASS |
| NEC8 | Homo sapiens | | | = 839.9 nM | | | NPASS |
| NCI-H524 | Homo sapiens | | | = 998680.59 nM | | | NPASS |
| NCI-H526 | Homo sapiens | | | = 2636.52 nM | | | NPASS |
| NCI-H596 | | | | = 817.86 nM | | | NPASS |
| NCI-H630 | Homo sapiens | | | = 1303.9 nM | | | NPASS |
| NCI-H64 | Homo sapiens | | | = 547.1 nM | | | NPASS |
| NCI-H650 | Homo sapiens | | | = 665.19 nM | | | NPASS |
| NCI-H661 | Homo sapiens | | | = 5428.73 nM | | | NPASS |
| NCI-H69 | Homo sapiens | | | = 6713.8 nM | | | NPASS |
| NCI-H1693 | Homo sapiens | | | = 66678.0 nM | | | NPASS |
| NCI-H719 | Homo sapiens | | | = 2611.26 nM | | | NPASS |
| NCI-H720 | Homo sapiens | | | = 1136712.95 nM | | | NPASS |
| NCI-H727 | Homo sapiens | | | = 638.3 nM | | | NPASS |
| NCI-H747 | Homo sapiens | | | = 441.39 nM | | | NPASS |
| NCI-H748 | Homo sapiens | | | = 1782.46 nM | | | NPASS |
| NCI-H810 | Homo sapiens | | | = 502.62 nM | | | NPASS |
| NCI-H82 | Homo sapiens | | | = 407349.28 nM | | | NPASS |
| NCI-H838 | Homo sapiens | | | = 136106.82 nM | | | NPASS |
| NCI-H889 | Homo sapiens | | | = 1636835.36 nM | | | NPASS |
| NCI-N87 | Homo sapiens | | | = 2942.3 nM | | | NPASS |
| NCI-H520 | | | | = 1354.54 nM | | | NPASS |
| NCI-H1651 | Homo sapiens | | | = 22750.27 nM | | | NPASS |
| NCI-H1355 | Homo sapiens | | | = 2822.51 nM | | | NPASS |
| NCI-H1648 | Homo sapiens | | | = 11147.41 nM | | | NPASS |
| MDA-MB-436 | Homo sapiens | | | = 3610.0 nM | | | NPASS |
| MDA-MB-453 | Homo sapiens | | | = 2518.94 nM | | | NPASS |
| MDA-MB-468 | Homo sapiens | | | = 966.84 nM|= 3280.0 nM | | | NPASS |
| ME-180 | Homo sapiens | | | = 278.91 nM | | | NPASS |
| MEG-01 | Homo sapiens | | | = 451.25 nM | | | NPASS |
| MEL-HO | Homo sapiens | | | = 148.82 nM | | | NPASS |
| MEL-JUSO | Homo sapiens | | | = 540.14 nM | | | NPASS |
| MES-SA | Homo sapiens | | | = 41.32 nM | | | NPASS |
| MDA-MB-415 | Homo sapiens | | | = 2276.74 nM | | | NPASS |
| MFE-280 | Homo sapiens | | | = 4946.54 nM | | | NPASS |
| MFH-ino | Homo sapiens | | | = 863.85 nM | | | NPASS |
| MFM-223 | Homo sapiens | | | = 898.77 nM | | | NPASS |
| MG-63 | Homo sapiens | | | = 256.77 nM|= 7360.0 nM|= 5670.0 nM | | | NPASS |
| MGC-803 | Homo sapiens | | | = 1510.0 nM|= 1280.0 nM | | | NPASS |
| MHH-CALL-2 | Homo sapiens | | | = 715.04 nM | | | NPASS |
| MHH-ES-1 | Homo sapiens | | | = 688.56 nM | | | NPASS |
| MHH-NB-11 | Homo sapiens | | | = 485.95 nM | | | NPASS |
| MHH-PREB-1 | Homo sapiens | | | = 251.57 nM | | | NPASS |
| MFE-296 | Homo sapiens | | | = 662.44 nM | | | NPASS |
| MDA-MB-361 | Homo sapiens | | | = 1732.36 nM | | | NPASS |
| MDA-MB-231 | Homo sapiens | | | = 6600.0 nM|= 1015.44 nM|= 3940.0 nM|= 8750.0 nM|= 6500.0 nM|= 2770.0 nM|= 1580.0 nM|= 108000.0 nM|= 7620.0 nM|= 8980.0 nM|= 2880.0 nM | | | NPASS |
| MDA-MB-175-VII | Homo sapiens | | | = 2053.07 nM | | | NPASS |
| OVCAR-4 | Homo sapiens | | | = 669.55 nM | | | NPASS |
| LS174T | Homo sapiens | | | = 8900.0 nM | | | NPASS |
| LU-134-A | Homo sapiens | | | = 809.71 nM | | | NPASS |
| LU-139 | Homo sapiens | | | = 6264.09 nM | | | NPASS |
| LU-165 | Homo sapiens | | | = 634.05 nM | | | NPASS |
| LU-99A | Homo sapiens | | | = 1295.65 nM | | | NPASS |
| LXF-289 cell line | | | | = 3271.56 nM | | | NPASS |
| LoVo | Homo sapiens | | | = 1335.09 nM | | | NPASS |
| Lu-65 | Homo sapiens | | | = 221073.67 nM | | | NPASS |
| M059J | Homo sapiens | | | = 134.19 nM | | | NPASS |
| M14 | Homo sapiens | | | = 1492.69 nM | | | NPASS |
| MC-CAR | Homo sapiens | | | = 813.62 nM | | | NPASS |
| MC-IXC | Homo sapiens | | | = 387.38 nM | | | NPASS |
| MC116 | Homo sapiens | | | = 1786.36 nM | | | NPASS |
| MCF-10A | Homo sapiens | | | = 93400.0 nM|= 23500.0 nM|= 20940.0 nM | | | NPASS |
| MCF10 | Homo sapiens | | | = 4560.0 nM | | | NPASS |
| MCF7 | Homo sapiens | | | = 1450.0 nM|= 1900.0 nM|= 434.85 nM|= 1800.0 nM|= 5490.0 nM|= 2400.0 nM|= 2700.0 nM|= 6500.0 nM|= 9550.0 nM|= 5400.0 nM|= 23410.0 nM|= 23600.0 nM|= 9320.0 nM|= 4570.0 nM|= 7750.0 nM|= 8320.0 nM|= 1030.0 nM|= 2110.0 nM|= 4990.0 nM | | | NPASS |
| MDA-MB-134-VI | Homo sapiens | | | = 709.4 nM | | | NPASS |
| MDA-MB-157 | Homo sapiens | | | = 636.63 nM | | | NPASS |
| MIA PaCa-2 | Homo sapiens | | | = 276.49 nM | | | NPASS |
| NCI-H1650 | Homo sapiens | | | = 1375.03 nM|= 8320.0 nM | | | NPASS |
| MKN-1 | Homo sapiens | | | = 235.76 nM | | | NPASS |
| MKN-45 | Homo sapiens | | | = 608.39 nM | | | NPASS |
| NB13 | Homo sapiens | | | = 316.93 nM | | | NPASS |
| NB5 | Homo sapiens | | | = 2432.63 nM | | | NPASS |
| NB6 | Homo sapiens | | | = 454.4 nM | | | NPASS |
| NB69 | Homo sapiens | | | = 212.73 nM | | | NPASS |
| NCCIT | Homo sapiens | | | = 517.16 nM | | | NPASS |
| NCI-H1092 | Homo sapiens | | | = 1393.11 nM | | | NPASS |
| NCI-H1155 | Homo sapiens | | | = 1998891.39 nM | | | NPASS |
| NCI-H1299 | Homo sapiens | | | = 1071.94 nM|= 1880.0 nM|= 3950.0 nM | | | NPASS |
| NB12 | Homo sapiens | | | = 666.31 nM | | | NPASS |
| NCI-H1304 | Homo sapiens | | | = 184889.62 nM | | | NPASS |
| NCI-H1417 | Homo sapiens | | | = 815.92 nM | | | NPASS |
| NCI-H1436 | Homo sapiens | | | = 603.96 nM | | | NPASS |
| NCI-H1437 | Homo sapiens | | | = 1557.48 nM | | | NPASS |
| NCI-H1522 | Homo sapiens | | | = 519.44 nM | | | NPASS |
| NCI-H1563 | Homo sapiens | | | = 626.38 nM | | | NPASS |
| NCI-H1581 | Homo sapiens | | | = 89965.84 nM | | | NPASS |
| NCI-H1618 | Homo sapiens | | | = 2019.66 nM | | | NPASS |
| NCI-H1623 | Homo sapiens | | | = 2727.21 nM | | | NPASS |
| NCI-H1395 | Homo sapiens | | | = 971830.1 nM | | | NPASS |
| NB10 | Homo sapiens | | | = 1343.65 nM | | | NPASS |
| NB1 | Homo sapiens | | | = 1034.34 nM | | | NPASS |
| NALM-6 | Homo sapiens | | | = 2.797 nM | | | NPASS |
| LS-513 | Homo sapiens | | | = 1477.97 nM | | | NPASS |
| MKN-7 | Homo sapiens | | | = 2205.51 nM | | | NPASS |
| ML-2 | Homo sapiens | | | = 617.74 nM | | | NPASS |
| MLMA | Homo sapiens | | | = 539.08 nM | | | NPASS |
| MMAC-SF | Homo sapiens | | | = 751.96 nM | | | NPASS |
| MN-60 | Homo sapiens | | | = 347.88 nM | | | NPASS |
| MOLT-16 | Homo sapiens | | | = 2762.98 nM | | | NPASS |
| MOLT-4 | Homo sapiens | | | = 410.12 nM | | | NPASS |
| MONO-MAC-6 | Homo sapiens | | | = 244.77 nM|= 2600.0 nM | | | NPASS |
| MPP-89 | Homo sapiens | | | = 857.25 nM | | | NPASS |
| MRK-nu-1 | Homo sapiens | | | = 101.93 nM | | | NPASS |
| MS-1 | Homo sapiens | | | = 1772.48 nM | | | NPASS |
| MSTO-211H | Homo sapiens | | | = 603751.69 nM | | | NPASS |
| MV4-11 | Homo sapiens | | | = 273.63 nM | | | NPASS |
| MZ1-PC | Homo sapiens | | | = 19.28 nM | | | NPASS |
| MZ2-MEL | Homo sapiens | | | = 385.22 nM | | | NPASS |
| MZ7-mel | Homo sapiens | | | = 113.72 nM | | | NPASS |
| MeWo | Homo sapiens | | | = 517.32 nM | | | NPASS |
| Mo | Homo sapiens | | | = 819.71 nM | | | NPASS |
| MKN-28 | Homo sapiens | | | = 616.87 nM | | | NPASS |
| OVCAR-5 | Homo sapiens | | | = 1123.89 nM | | | NPASS |
| TALL-1 | Homo sapiens | | | = 754677.12 nM | | | NPASS |
| P12-Ichikawa | Homo sapiens | | | = 1388.36 nM | | | NPASS |
| SW1573 | Homo sapiens | | | = 371.8 nM | | | NPASS |
| SW1710 | Homo sapiens | | | = 2.91 nM | | | NPASS |
| SW1783 | Homo sapiens | | | = 1068.84 nM | | | NPASS |
| SW1990 | Homo sapiens | | | = 1617.18 nM | | | NPASS |
| SW48 | Homo sapiens | | | = 1258.27 nM | | | NPASS |
| SW626 | Homo sapiens | | | = 635.13 nM | | | NPASS |
| SW684 | Homo sapiens | | | = 777.33 nM | | | NPASS |
| SW756 | Homo sapiens | | | = 761.77 nM | | | NPASS |
| SW1463 | Homo sapiens | | | = 8606.36 nM | | | NPASS |
| SW780 | Homo sapiens | | | = 405.52 nM | | | NPASS |
| SW872 | Homo sapiens | | | = 367.48 nM|= 760.0 nM | | | NPASS |
| SW948 | Homo sapiens | | | = 11909.0 nM | | | NPASS |
| SW982 | Homo sapiens | | | = 60.23 nM|= 2800.0 nM | | | NPASS |
| SiHa | Homo sapiens | | | = 18601.72 nM | | | NPASS |
| T-24 | Homo sapiens | | | = 2462.32 nM | | | NPASS |
| T47D | Homo sapiens | | | = 223.06 nM | | | NPASS |
| T84 | Homo sapiens | | | = 14520.28 nM | | | NPASS |
| T98G | Homo sapiens | | | = 1082.08 nM | | | NPASS |
| SW837 | Homo sapiens | | | = 19784.09 nM | | | NPASS |
| TCC-SUP | Homo sapiens | | | = 554.45 nM | | | NPASS |
| SW1417 | Homo sapiens | | | = 825.83 nM | | | NPASS |
| SW1088 | Homo sapiens | | | = 699.55 nM | | | NPASS |
| SNB-75 | Homo sapiens | | | = 745.95 nM | | | NPASS |
| SNG-M | Homo sapiens | | | = 272.37 nM | | | NPASS |
| SNU-16 | Homo sapiens | | | = 5100648.67 nM | | | NPASS |
| SNU-387 | Homo sapiens | | | = 1068.57 nM | | | NPASS |
| SNU-423 | Homo sapiens | | | = 163.07 nM | | | NPASS |
| SNU-449 | Homo sapiens | | | = 813.25 nM | | | NPASS |
| SNU-475 | Homo sapiens | | | = 14058.92 nM | | | NPASS |
| SNU-5 | Homo sapiens | | | = 9536.71 nM | | | NPASS |
| SW13 | Homo sapiens | | | = 1409.19 nM | | | NPASS |
| SNU-C1 | Homo sapiens | | | = 722279.37 nM | | | NPASS |
| SNU1 | Homo sapiens | | | = 1602.2 nM | | | NPASS |
| SR | Homo sapiens | | | = 140.73 nM | | | NPASS |
| ST486 | Homo sapiens | | | = 6.179 nM | | | NPASS |
| SU-DHL-1 | Homo sapiens | | | = 499.22 nM | | | NPASS |
| SUP-T1 | Homo sapiens | | | = 1822.91 nM | | | NPASS |
| SW 954 | Homo sapiens | | | = 466.71 nM | | | NPASS |
| SW 962 | Homo sapiens | | | = 568.3 nM | | | NPASS |
| SW-620 | Homo sapiens | | | = 358.55 nM | | | NPASS |
| SNU-C2B | Homo sapiens | | | = 24926.79 nM | | | NPASS |
| TE-1 | Homo sapiens | | | = 15796.45 nM | | | NPASS |
| TE-10 | Homo sapiens | | | = 986.09 nM | | | NPASS |
| TE-11 | Homo sapiens | | | = 4014.26 nM | | | NPASS |
| UACC-62 | Homo sapiens | | | = 1229.98 nM | | | NPASS |
| UACC-812 | Homo sapiens | | | = 5077.15 nM | | | NPASS |
| UACC-893 | Homo sapiens | | | = 119208.02 nM | | | NPASS |
| UMC-11 | Homo sapiens | | | = 46792.08 nM | | | NPASS |
| UMUC3 | Homo sapiens | | | = 967.27 nM | | | NPASS |
| UO-31 | Homo sapiens | | | = 770.84 nM | | | NPASS |
| VA-ES-BJ | Homo sapiens | | | = 400.58 nM | | | NPASS |
| VM-CUB-1 | Homo sapiens | | | = 1028.56 nM | | | NPASS |
| UACC-257 | Homo sapiens | | | = 26356.58 nM | | | NPASS |
| VMRC-RCZ | Homo sapiens | | | = 546.67 nM | | | NPASS |
| WM-115 | Homo sapiens | | | = 10644.2 nM | | | NPASS |
| WSU-NHL | Homo sapiens | | | = 260.33 nM | | | NPASS |
| YAPC | Homo sapiens | | | = 243833.84 nM | | | NPASS |
| YKG-1 | Homo sapiens | | | = 228.91 nM | | | NPASS |
| YT | Homo sapiens | | | = 383.89 nM | | | NPASS |
| no-10 | Homo sapiens | | | = 290.23 nM | | | NPASS |
| no-11 | Homo sapiens | | | = 805.42 nM | | | NPASS |
| LS-411N | Homo sapiens | | | = 3189.61 nM | | | NPASS |
| Vero | Chlorocebus sabaeus | | | = 6760.0 nM | | | NPASS |
| U2OS | Homo sapiens | | | = 597438.89 nM | | | NPASS |
| U-937 | Homo sapiens | | | = 1200.0 nM | | | NPASS |
| U-87 MG | Homo sapiens | | | = 1275.78 nM | | | NPASS |
| TE-12 | Homo sapiens | | | = 2343.25 nM | | | NPASS |
| TE-15 | Homo sapiens | | | = 400.31 nM | | | NPASS |
| TE-441-T | Homo sapiens | | | = 2.238 nM | | | NPASS |
| TE-5 | Homo sapiens | | | = 1004.32 nM | | | NPASS |
| TE-6 | Homo sapiens | | | = 2967.91 nM | | | NPASS |
| TE-8 | Homo sapiens | | | = 1280.63 nM | | | NPASS |
| TE-9 | Homo sapiens | | | = 407.52 nM | | | NPASS |
| TGBC1TKB | Homo sapiens | | | = 1428.19 nM | | | NPASS |
| TGBC24TKB | Homo sapiens | | | = 27882.74 nM | | | NPASS |
| TGW | Homo sapiens | | | = 521.64 nM | | | NPASS |
| THP-1 | Homo sapiens | | | = 891.43 nM|= 820.0 nM | | | NPASS |
| TK-10 | Homo sapiens | | | = 1224.02 nM | | | NPASS |
| TT | Homo sapiens | | | = 1698.76 nM | | | NPASS |
| TUR | Homo sapiens | | | = 465.99 nM | | | NPASS |
| TYK-nu | Homo sapiens | | | = 1152.13 nM | | | NPASS |
| U-118-MG | Homo sapiens | | | = 841.85 nM | | | NPASS |
| U-251 | Homo sapiens | | | = 1432.46 nM | | | NPASS |
| U-266 | Homo sapiens | | | = 675.16 nM | | | NPASS |
| U-698-M | Homo sapiens | | | = 300.87 nM | | | NPASS |
| SN12C | Homo sapiens | | | = 1762.58 nM | | | NPASS |
| SKG-IIIa | Homo sapiens | | | = 4388.27 nM | | | NPASS |
| SK-UT-1 | Homo sapiens | | | = 7.438 nM | | | NPASS |
| SK-PN-DW | Homo sapiens | | | = 36.55 nM | | | NPASS |
| REH | Homo sapiens | | | = 146.96 nM | | | NPASS |
| RERF-LC-MS | Homo sapiens | | | = 4189.97 nM | | | NPASS |
| RH-1 | Homo sapiens | | | = 719.88 nM | | | NPASS |
| RKO | Homo sapiens | | | = 270.3 nM | | | NPASS |
| RL | Homo sapiens | | | = 464793.4 nM | | | NPASS |
| RL95-2 | Homo sapiens | | | = 719.73 nM | | | NPASS |
| RMG-I | Homo sapiens | | | = 864.23 nM | | | NPASS |
| RO82-W-1 | Homo sapiens | | | = 2842.95 nM | | | NPASS |
| RD | Homo sapiens | | | = 449.06 nM | | | NPASS |
| RPMI 8402 | Homo sapiens | | | = 1498.31 nM | | | NPASS |
| RPMI-6666 | Homo sapiens | | | = 587.13 nM | | | NPASS |
| RPMI-7951 | Homo sapiens | | | = 156.09 nM | | | NPASS |
| RPMI-8226 | Homo sapiens | | | = 471.88 nM | | | NPASS |
| RPMI-8866 | Homo sapiens | | | = 536.04 nM | | | NPASS |
| RS4-11 | Homo sapiens | | | = 416.76 nM | | | NPASS |
| RT-112 | Homo sapiens | | | = 70.37 nM | | | NPASS |
| RT-4 | Homo sapiens | | | = 10121.92 nM | | | NPASS |
| RVH-421 | Homo sapiens | | | = 1467.47 nM | | | NPASS |
| RPMI-2650 | Homo sapiens | | | = 374.74 nM | | | NPASS |
| RCM-1 | Homo sapiens | | | = 2002.19 nM | | | NPASS |
| RCC10RGB | Homo sapiens | | | = 1563.9 nM | | | NPASS |
| QIMR-WIL | Homo sapiens | | | = 181.89 nM | | | NPASS |
| P30-OHK | Homo sapiens | | | = 220.48 nM | | | NPASS |
| P31-FUJ | Homo sapiens | | | = 2066.09 nM | | | NPASS |
| PA-1 | Homo sapiens | | | = 201.28 nM|= 920.0 nM | | | NPASS |
| PANC-03-27 | Homo sapiens | | | = 167.4 nM | | | NPASS |
| PANC-08-13 | Homo sapiens | | | = 10430.49 nM | | | NPASS |
| PBMC | Homo sapiens | | | = 5000.0 nM | | | NPASS |
| PC-14 | Homo sapiens | | | = 1507.16 nM | | | NPASS |
| PC-3 | Homo sapiens | | | = 858.79 nM | | | NPASS |
| PF-382 | Homo sapiens | | | = 789.51 nM | | | NPASS |
| PFSK-1 | Homo sapiens | | | = 76572.12 nM | | | NPASS |
| PLC-PRF-5 | Homo sapiens | | | = 1815.79 nM | | | NPASS |
| PSN1 | Homo sapiens | | | = 71023.8 nM | | | NPASS |
| Panc1005 | Homo sapiens | | | = 415.63 nM | | | NPASS |
| Plasmodium berghei | Plasmodium berghei | | | = 1370.0 nM | | | NPASS |
| Plasmodium falciparum | Plasmodium falciparum | | | > 5000.0 nM | | | NPASS |
| Protein-tyrosine phosphatase 1 | Saccharomyces cerevisiae S288c | P25044 | | = 70000.0 nM | | | NPASS |
| Protein-tyrosine phosphatase 1B | Homo sapiens | P18031 | | = 25000.0 nM | | | NPASS |
| Pyruvate kinase isozymes M1/M2 | Homo sapiens | P14618 | | = 12960.0 nM|= 8820.0 nM|= 10000.0 nM|= 500.0 nM|= 1520.0 nM|= 381.0 nM|= 326.0 nM|> 10000.0 nM|= 800.0 nM|= 301.0 nM|= 1420.0 nM|= 2576.0 nM | | | NPASS |
| Pyruvate kinase isozymes R/L | Homo sapiens | P30613 | | = 39250.0 nM | | | NPASS |
| RXF 393 | Homo sapiens | | | = 749.01 nM | | | NPASS |
| OVCAR-8 | Homo sapiens | | | = 460.05 nM | | | NPASS |
| Raji | Homo sapiens | | | = 631.17 nM | | | NPASS |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome coronavirus 2 | P0DTD1 | | = 15750.0 nM|= 15739.83 nM|= 1600.0 nM|= 670.0 nM | | | NPASS |
| SK-BR-3 | Homo sapiens | | | = 3750.0 nM | | | NPASS |
| SK-CO-1 | Homo sapiens | | | = 2054.9 nM | | | NPASS |
| SK-HEP1 | Homo sapiens | | | = 547.51 nM | | | NPASS |
| SK-LMS-1 | Homo sapiens | | | = 108.41 nM | | | NPASS |
| SK-LU-1 | Homo sapiens | | | = 750.1 nM | | | NPASS |
| SK-MEL-1 | Homo sapiens | | | = 138410.24 nM | | | NPASS |
| SK-MEL-2 | Homo sapiens | | | = 6328.9 nM | | | NPASS |
| SK-MEL-24 | Homo sapiens | | | = 1133.44 nM | | | NPASS |
| SJSA-1 | Homo sapiens | | | = 5525.33 nM | | | NPASS |
| SK-MEL-28 | Homo sapiens | | | = 277189.39 nM | | | NPASS |
| SK-MEL3 | Homo sapiens | | | = 2642.21 nM | | | NPASS |
| SK-MES-1 | Homo sapiens | | | = 6286.32 nM | | | NPASS |
| SK-MM-2 | Homo sapiens | | | = 498.97 nM | | | NPASS |
| SK-N-AS | Homo sapiens | | | = 1786.2 nM | | | NPASS |
| SK-N-DZ | Homo sapiens | | | = 1803.2 nM | | | NPASS |
| SK-N-FI | Homo sapiens | | | = 7693.54 nM | | | NPASS |
| SK-NEP-1 | Homo sapiens | | | = 1081.12 nM | | | NPASS |
| SK-OV-3 | Homo sapiens | | | = 1560.3 nM|= 3460.0 nM | | | NPASS |
| SK-MEL-30 | Homo sapiens | | | = 694.8 nM | | | NPASS |
| SJRH30 | Homo sapiens | | | = 369.2 nM | | | NPASS |
| SIMA | Homo sapiens | | | = 2318.43 nM | | | NPASS |
| SIG-M5 | Homo sapiens | | | = 169.86 nM | | | NPASS |
| S-117 | Homo sapiens | | | = 387.1 nM | | | NPASS |
| SAOS-2 | Homo sapiens | | | = 2367.35 nM | | | NPASS |
| SARS-CoV-2 | Severe acute respiratory syndrome coronavirus 2 | | | > 20000.0 nM|> 19952.62 nM|= 670.0 nM | | | NPASS |
| SAS | Homo sapiens | | | = 853.74 nM | | | NPASS |
| SBC-1 | Homo sapiens | | | = 12149.22 nM | | | NPASS |
| SBC-5 | Homo sapiens | | | = 215.46 nM | | | NPASS |
| SCC-15 | Homo sapiens | | | = 650.5 nM | | | NPASS |
| SCC-25 | Homo sapiens | | | = 382.64 nM | | | NPASS |
| SCC-3 | Homo sapiens | | | = 1003.43 nM | | | NPASS |
| SCC-4 | Homo sapiens | | | = 440.6 nM|= 10100.0 nM | | | NPASS |
| SCC-9 | Homo sapiens | | | = 196.75 nM | | | NPASS |
| SCH | Homo sapiens | | | = 195008.47 nM | | | NPASS |
| SCLC-21H | Homo sapiens | | | = 1364.86 nM | | | NPASS |
| SF-126 | Homo sapiens | | | = 772.97 nM | | | NPASS |
| SF-268 | Homo sapiens | | | = 5577.43 nM | | | NPASS |
| SF-295 | Homo sapiens | | | = 664.18 nM | | | NPASS |
| SF-539 | Homo sapiens | | | = 856.82 nM | | | NPASS |
| SH-4 | Homo sapiens | | | = 371.35 nM | | | NPASS |
| SHP77 | Homo sapiens | | | = 445.54 nM | | | NPASS |
| Ramos-2G6-4C10 | Homo sapiens | | | = 315.03 nM | | | NPASS |
| LS-123 | Homo sapiens | | | = 537.66 nM | | | NPASS |
| COLO-320-HSR | Homo sapiens | | | = 384.48 nM | | | NPASS |
| LP-1 | Homo sapiens | | | = 686.37 nM | | | NPASS |
| CP66-MEL | Homo sapiens | | | = 2396.67 nM | | | NPASS |
| CPC-N | Homo sapiens | | | = 24262.4 nM | | | NPASS |
| CTB-1 | Homo sapiens | | | = 859.02 nM | | | NPASS |
| CTV-1 | Homo sapiens | | | = 32752.88 nM | | | NPASS |
| CW-2 | Homo sapiens | | | = 676152.07 nM | | | NPASS |
| CWR22R | Homo sapiens | | | = 4614.94 nM | | | NPASS |
| Ca-Ski | Homo sapiens | | | = 650.31 nM | | | NPASS |
| Ca9-22 | Homo sapiens | | | = 580.63 nM|= 12810.0 nM|= 13590.0 nM | | | NPASS |
| CP50-MEL-B | Homo sapiens | | | = 1433.36 nM | | | NPASS |
| CaR-1 | Homo sapiens | | | = 1308.43 nM | | | NPASS |
| Calu-3 | Homo sapiens | | | = 1108.34 nM|= 7220.0 nM | | | NPASS |
| Calu-6 | Homo sapiens | | | = 15732.0 nM | | | NPASS |
| Caov-3 cell line | | | | = 766.5 nM | | | NPASS |
| Caov-4 | Homo sapiens | | | = 1884.19 nM | | | NPASS |
| Capan-2 | Homo sapiens | | | = 1005.29 nM | | | NPASS |
| ChaGo-K-1 | Homo sapiens | | | = 656.72 nM | | | NPASS |
| D-247MG | Homo sapiens | | | = 1660.02 nM | | | NPASS |
| D-263MG | Homo sapiens | | | = 2230.07 nM | | | NPASS |
| Calu-1 | Homo sapiens | | | = 1232.12 nM | | | NPASS |
| D-336MG | Homo sapiens | | | = 1749.77 nM | | | NPASS |
| COR-L88 | Homo sapiens | | | = 109652.36 nM | | | NPASS |
| COR-L23 | Homo sapiens | | | = 301.5 nM | | | NPASS |
| CGTH-W-1 | Homo sapiens | | | = 499.93 nM | | | NPASS |
| CHL-1 | Homo sapiens | | | = 167.8 nM | | | NPASS |
| CHP-126 | Homo sapiens | | | = 695.35 nM | | | NPASS |
| CHP-212 | Homo sapiens | | | = 1096.47 nM | | | NPASS |
| CMK | Homo sapiens | | | = 352.13 nM | | | NPASS |
| CNE | Homo sapiens | | | = 700.0 nM | | | NPASS |
| COLO 205 | Homo sapiens | | | = 537.72 nM | | | NPASS |
| COLO-668 | Homo sapiens | | | = 6196.13 nM | | | NPASS |
| COR-L279 | Homo sapiens | | | = 188288.43 nM | | | NPASS |
| COLO-678 | Homo sapiens | | | = 1628.64 nM | | | NPASS |
| COLO-680N | Homo sapiens | | | = 590.03 nM | | | NPASS |
| COLO-684 | Homo sapiens | | | = 400.53 nM | | | NPASS |
| COLO-741 | Homo sapiens | | | = 2694.21 nM | | | NPASS |
| COLO-792 | Homo sapiens | | | = 81952.6 nM | | | NPASS |
| COLO-800 | Homo sapiens | | | = 3260066.91 nM | | | NPASS |
| COLO-824 | Homo sapiens | | | = 715.2 nM | | | NPASS |
| COLO-829 | Homo sapiens | | | = 657.99 nM | | | NPASS |
| COR-L105 | Homo sapiens | | | = 230.34 nM | | | NPASS |
| COLO-679 | Homo sapiens | | | = 184.01 nM | | | NPASS |
| D-392MG | Homo sapiens | | | = 915.29 nM | | | NPASS |
| D-502MG | Homo sapiens | | | = 4365.48 nM | | | NPASS |
| D-542MG | Homo sapiens | | | = 580.88 nM | | | NPASS |
| DoTc2-4510 | Homo sapiens | | | = 262.79 nM | | | NPASS |
| Dual specificity phosphatase Cdc25A | Homo sapiens | P30304 | | = 220.0 nM|= 2140.0 nM | | | NPASS |
| Dual specificity phosphatase Cdc25B | Homo sapiens | P30305 | | = 400.0 nM|= 5820.0 nM | | | NPASS |
| Dual specificity phosphatase Cdc25C | Homo sapiens | P30307 | | = 4780.0 nM | | | NPASS |
| EB-3 | Homo sapiens | | | = 1142.2 nM | | | NPASS |
| EB2 | Homo sapiens | | | = 310.95 nM | | | NPASS |
| EC-GI-10 | Homo sapiens | | | = 57446.9 nM | | | NPASS |
| ECC12 | Homo sapiens | | | = 9648.24 nM | | | NPASS |
| Detroit562 | Homo sapiens | | | = 29295.97 nM | | | NPASS |
| ECC4 | Homo sapiens | | | = 1203.45 nM | | | NPASS |
| EFO-21 | Homo sapiens | | | = 1338.59 nM | | | NPASS |
| EFO-27 | Homo sapiens | | | = 330.34 nM | | | NPASS |
| EGI-1 | Homo sapiens | | | = 2511.08 nM | | | NPASS |
| EHEB | Homo sapiens | | | = 2094.47 nM | | | NPASS |
| EKVX | Homo sapiens | | | = 3674.07 nM | | | NPASS |
| EM-2 | Homo sapiens | | | = 976.93 nM | | | NPASS |
| EOL1 | Homo sapiens | | | = 508.75 nM | | | NPASS |
| ES1 | Homo sapiens | | | = 502.89 nM | | | NPASS |
| EFM-19 | Homo sapiens | | | = 212.1 nM | | | NPASS |
| Daudi | Homo sapiens | | | = 3442.87 nM | | | NPASS |
| Daoy | Homo sapiens | | | = 158.77 nM | | | NPASS |
| DV-90 | Homo sapiens | | | = 206842.58 nM | | | NPASS |
| D283 Med | | | | = 835.31 nM | | | NPASS |
| DB | Homo sapiens | | | = 726.29 nM | | | NPASS |
| DBTRG-05MG | Homo sapiens | | | = 611.1 nM | | | NPASS |
| DEL | Homo sapiens | | | = 153.81 nM | | | NPASS |
| DG-75 | Homo sapiens | | | = 1167.49 nM | | | NPASS |
| DJM-1 | Homo sapiens | | | = 6387.23 nM | | | NPASS |
| DK-MG | Homo sapiens | | | = 9817.5 nM | | | NPASS |
| DMS-114 | Homo sapiens | | | = 35541.18 nM | | | NPASS |
| DMS-153 | Homo sapiens | | | = 27808.34 nM | | | NPASS |
| DMS-273 | Homo sapiens | | | = 395.79 nM | | | NPASS |
| DMS-53 | Homo sapiens | | | = 21456.74 nM | | | NPASS |
| DMS-79 | Homo sapiens | | | = 271650.96 nM | | | NPASS |
| DNA topoisomerase I | Homo sapiens | P11387 | | = 208000.0 nM | | | NPASS |
| DNA topoisomerase II | Homo sapiens | Q02880 | | = 6200.0 nM|= 6700.0 nM|= 16000.0 nM|= 12500.0 nM|= 5700.0 nM|= 7800.0 nM | | | NPASS |
| DOHH-2 | Homo sapiens | | | = 706.26 nM | | | NPASS |
| DOK | Homo sapiens | | | = 5185.18 nM | | | NPASS |
| DSH1 | Homo sapiens | | | = 10584.2 nM | | | NPASS |
| DU-145 | Homo sapiens | | | = 193.09 nM|= 16000.0 nM | | | NPASS |
| DU-4475 | Homo sapiens | | | = 179.84 nM | | | NPASS |
| CESS | Homo sapiens | | | = 776.45 nM | | | NPASS |
| ES3 | Homo sapiens | | | = 656.49 nM | | | NPASS |
| CCRF-CEM | Homo sapiens | | | = 567.02 nM | | | NPASS |
| CAS-1 | Homo sapiens | | | = 462.11 nM | | | NPASS |
| A4-Fuk | Homo sapiens | | | = 249.73 nM | | | NPASS |
| A498 | Homo sapiens | | | = 81.9 nM | | | NPASS |
| A549 | Homo sapiens | | | = 3530.0 nM|= 7300.0 nM|= 6500.0 nM|= 6130.0 nM|= 10250.0 nM|= 5060.0 nM|= 10370.0 nM|= 1708.0 nM|= 3130.0 nM|= 11680.0 nM|= 7730.0 nM|= 1800.0 nM|= 4470.0 nM|= 3370.0 nM|= 2510.0 nM | | | NPASS |
| A673 | Homo sapiens | | | = 1220.48 nM | | | NPASS |
| A704 | Homo sapiens | | | = 2704.66 nM | | | NPASS |
| ABC-1 | Homo sapiens | | | = 707.48 nM | | | NPASS |
| ACHN | Homo sapiens | | | = 146.38 nM | | | NPASS |
| ACN | Homo sapiens | | | = 916.95 nM | | | NPASS |
| A388 | Homo sapiens | | | = 866.56 nM | | | NPASS |
| AGS | Homo sapiens | | | = 612.57 nM | | | NPASS |
| AM-38 | Homo sapiens | | | = 96.31 nM | | | NPASS |
| AN3-CA | Homo sapiens | | | = 79.65 nM | | | NPASS |
| ARH-77 | Homo sapiens | | | = 873.49 nM | | | NPASS |
| ASPC1 | Homo sapiens | | | = 618.87 nM | | | NPASS |
| ATN-1 | Homo sapiens | | | = 849.13 nM | | | NPASS |
| AU565 | Homo sapiens | | | = 1239.81 nM | | | NPASS |
| Acyl coenzyme A:cholesterol acyltransferase 1 | Homo sapiens | P35610 | | = 70400.0 nM | | | NPASS |
| Acyl coenzyme A:cholesterol acyltransferase 2 | Homo sapiens | O75908 | | = 138200.0 nM | | | NPASS |
| ALL-PO | Homo sapiens | | | = 315.12 nM | | | NPASS |
| B16-F10 | Mus musculus | | | = 17900.0 nM|= 3720.0 nM | | | NPASS |
| A3-KAW | Homo sapiens | | | = 2140.29 nM | | | NPASS |
| A253 cell line | | | | = 7.493 nM | | | NPASS |
| LS-1034 | Homo sapiens | | | = 2747.15 nM | | | NPASS |
| 23132-87 | Homo sapiens | | | = 2108.3 nM | | | NPASS |
| 5637 | Homo sapiens | | | = 206270.21 nM | | | NPASS |
| 639-V | Homo sapiens | | | = 265.01 nM | | | NPASS |
| 647-V | Homo sapiens | | | = 358.52 nM | | | NPASS |
| 697 | Homo sapiens | | | = 875.65 nM | | | NPASS |
| 769-P | Homo sapiens | | | = 688.6 nM | | | NPASS |
| 786-0 | Homo sapiens | | | = 343.75 nM | | | NPASS |
| A2780 | Homo sapiens | | | = 2562.45 nM|= 390.0 nM | | | NPASS |
| 8-MG-BA | Homo sapiens | | | = 85.56 nM | | | NPASS |
| 8505C | Homo sapiens | | | = 3099.47 nM | | | NPASS |
| A-375 | Homo sapiens | | | = 311.11 nM | | | NPASS |
| A-427 | Homo sapiens | | | = 17.99 nM | | | NPASS |
| A-431 | Homo sapiens | | | = 106.97 nM | | | NPASS |
| A101D | Homo sapiens | | | = 0.7121 nM | | | NPASS |
| A172 | Homo sapiens | | | = 469.75 nM | | | NPASS |
| A204 | Homo sapiens | | | = 126.54 nM | | | NPASS |
| A2058 | Homo sapiens | | | = 919.12 nM | | | NPASS |
| 8305C | Homo sapiens | | | = 304.84 nM | | | NPASS |
| BB30-HNC | Homo sapiens | | | = 243.49 nM | | | NPASS |
| BB49-HNC | Homo sapiens | | | = 38584.67 nM | | | NPASS |
| BB65-RCC | Homo sapiens | | | = 695.45 nM | | | NPASS |
| C32 | Homo sapiens | | | = 2677.89 nM | | | NPASS |
| C3A | Homo sapiens | | | = 657.06 nM | | | NPASS |
| C8166 | Homo sapiens | | | = 407.51 nM | | | NPASS |
| CA46 | Homo sapiens | | | = 191.85 nM | | | NPASS |
| CAKI-1 | Homo sapiens | | | = 894.13 nM | | | NPASS |
| CAL-120 | Homo sapiens | | | = 1360.85 nM | | | NPASS |
| CAL-12T | Homo sapiens | | | = 1902.22 nM | | | NPASS |
| CAL-148 | Homo sapiens | | | = 676.6 nM | | | NPASS |
| C2BBe1 | Homo sapiens | | | = 755.64 nM | | | NPASS |
| CAL-27 | Homo sapiens | | | = 83274.14 nM | | | NPASS |
| CAL-39 | Homo sapiens | | | = 483.23 nM | | | NPASS |
| CAL-51 | Homo sapiens | | | = 20.85 nM | | | NPASS |
| CAL-54 | Homo sapiens | | | = 1419.9 nM | | | NPASS |
| CAL-62 | Homo sapiens | | | = 1279.99 nM | | | NPASS |
| CAL-72 | Homo sapiens | | | = 1012.93 nM | | | NPASS |
| CAL-85-1 | Homo sapiens | | | = 160.73 nM | | | NPASS |
| CAMA-1 | Homo sapiens | | | = 1516.69 nM | | | NPASS |
| CAPAN-1 | Homo sapiens | | | = 758.89 nM | | | NPASS |
| CAL-33 | Homo sapiens | | | = 2000.04 nM | | | NPASS |
| C-4-II | Homo sapiens | | | = 587.72 nM | | | NPASS |
| C-33-A | Homo sapiens | | | = 912.75 nM | | | NPASS |
| Bel-7402 | Homo sapiens | | | = 54500.0 nM|= 1240.0 nM | | | NPASS |
| BC-3 | Homo sapiens | | | = 926.19 nM | | | NPASS |
| BC1 cell line | | | | = 2681.4 nM | | | NPASS |
| BCPAP | Homo sapiens | | | = 922.59 nM | | | NPASS |
| BE-13 | Homo sapiens | | | = 1195.23 nM | | | NPASS |
| BEAS-2B | Homo sapiens | | | = 5360.0 nM | | | NPASS |
| BEN | Homo sapiens | | | = 813.72 nM | | | NPASS |
| BFTC-905 | Homo sapiens | | | = 283.61 nM | | | NPASS |
| BFTC-909 | Homo sapiens | | | = 3627.83 nM | | | NPASS |
| BHT-101 | Homo sapiens | | | = 1250.23 nM | | | NPASS |
| BHY | Homo sapiens | | | = 563.96 nM | | | NPASS |
| BL-41 | Homo sapiens | | | = 483.4 nM | | | NPASS |
| BL-70 | Homo sapiens | | | = 278.02 nM | | | NPASS |
| BOKU | Homo sapiens | | | = 1874.88 nM | | | NPASS |
| BPH-1 | Homo sapiens | | | = 1259.99 nM | | | NPASS |
| BT-20 | Homo sapiens | | | = 2561.3 nM | | | NPASS |
| BT-474 | Homo sapiens | | | = 208.36 nM|= 5740.0 nM | | | NPASS |
| BV-173 | Homo sapiens | | | = 435.95 nM | | | NPASS |
| BXPC-3 | Homo sapiens | | | = 333.58 nM | | | NPASS |
| Becker | Homo sapiens | | | = 1582.22 nM | | | NPASS |
| CCF-STTG1 | Homo sapiens | | | = 768.01 nM | | | NPASS |
| ES4 | Homo sapiens | | | = 4634.59 nM | | | NPASS |
| EFE-184 | Homo sapiens | | | = 543.94 nM | | | NPASS |
| ES6 | Homo sapiens | | | = 7878.52 nM | | | NPASS |
| JVM-3 | Homo sapiens | | | = 913180.9 nM | | | NPASS |
| Jurkat | Homo sapiens | | | = 970.0 nM | | | NPASS |
| K052 | Homo sapiens | | | = 1098.89 nM | | | NPASS |
| K5 | Homo sapiens | | | = 734.38 nM | | | NPASS |
| K562 | Homo sapiens | | | = 630.0 nM|= 600.0 nM|= 106057.88 nM|= 700.0 nM|= 1020.0 nM|= 20290.0 nM|= 120540.0 nM | | | NPASS |
| KALS-1 | Homo sapiens | | | = 1317.29 nM | | | NPASS |
| KARPAS-299 | Homo sapiens | | | = 799.41 nM | | | NPASS |
| KARPAS-422 | Homo sapiens | | | = 26611.7 nM | | | NPASS |
| JVM-2 | Homo sapiens | | | = 3868.13 nM | | | NPASS |
| KARPAS-45 | Homo sapiens | | | = 9989.05 nM | | | NPASS |
| KG-1 | | | | = 1597.73 nM | | | NPASS |
| KGN | Homo sapiens | | | = 1307.27 nM | | | NPASS |
| KINGS-1 | Homo sapiens | | | = 14077.46 nM | | | NPASS |
| KLE | Homo sapiens | | | = 684.66 nM | | | NPASS |
| KM-H2 | Homo sapiens | | | = 1036.17 nM | | | NPASS |
| KM12 | Homo sapiens | | | = 739.71 nM | | | NPASS |
| KMOE-2 | Homo sapiens | | | = 1240.66 nM | | | NPASS |
| KMS-12-PE | Homo sapiens | | | = 559.38 nM | | | NPASS |
| KE-37 | Homo sapiens | | | = 244.45 nM | | | NPASS |
| JIYOYE | Homo sapiens | | | = 1387.92 nM | | | NPASS |
| JEG-3 | Homo sapiens | | | = 3171.65 nM | | | NPASS |
| JAR | Homo sapiens | | | = 3262.95 nM | | | NPASS |
| HuCCT-1 | Homo sapiens | | | = 483.02 nM | | | NPASS |
| HuO-3N1 | Homo sapiens | | | = 4433.41 nM | | | NPASS |
| HuO9 | Homo sapiens | | | = 1658.0 nM | | | NPASS |
| HuP-T3 | Homo sapiens | | | = 833.73 nM | | | NPASS |
| HuP-T4 | Homo sapiens | | | = 1361.78 nM | | | NPASS |
| HuTu80 | Homo sapiens | | | = 370.2 nM | | | NPASS |
| Huh-7 | Homo sapiens | | | = 1955.26 nM | | | NPASS |
| IA-LM | Homo sapiens | | | = 2080.5 nM | | | NPASS |
| ES5 | Homo sapiens | | | = 2634.45 nM | | | NPASS |
| IGROV-1 | Homo sapiens | | | = 55.61 nM | | | NPASS |
| IM-9 | Homo sapiens | | | = 3412.07 nM | | | NPASS |
| IMR-5 | Homo sapiens | | | = 589.4 nM | | | NPASS |
| IPC-298 | Homo sapiens | | | = 557135.23 nM | | | NPASS |
| IST-MEL1 | Homo sapiens | | | = 14955.39 nM | | | NPASS |
| IST-MES1 | Homo sapiens | | | = 1696.61 nM | | | NPASS |
| IST-SL1 | Homo sapiens | | | = 65198.14 nM | | | NPASS |
| IST-SL2 | Homo sapiens | | | = 200.14 nM | | | NPASS |
| J-RT3-T3-5 | Homo sapiens | | | = 2086.36 nM | | | NPASS |
| J82 | Homo sapiens | | | = 142.55 nM | | | NPASS |
| KNS-42 | Homo sapiens | | | = 18658.43 nM | | | NPASS |
| Hs-578T | Homo sapiens | | | = 6223.4 nM | | | NPASS |
| KNS-81-FD | Homo sapiens | | | = 1081.94 nM | | | NPASS |
| KP-4 | Homo sapiens | | | = 500.8 nM | | | NPASS |
| LB1047-RCC | Homo sapiens | | | = 302.44 nM | | | NPASS |
| LB2241-RCC | Homo sapiens | | | = 1288.29 nM | | | NPASS |
| LB2518-MEL | Homo sapiens | | | = 3283.31 nM | | | NPASS |
| LB373-MEL-D | Homo sapiens | | | = 390.74 nM | | | NPASS |
| LB647-SCLC | Homo sapiens | | | = 232.78 nM | | | NPASS |
| LB771-HNC | Homo sapiens | | | = 20788.0 nM | | | NPASS |
| LB831-BLC | Homo sapiens | | | = 1916.8 nM | | | NPASS |
| LB996-RCC | Homo sapiens | | | = 191158.51 nM | | | NPASS |
| LAN-6 | Homo sapiens | | | = 3219.16 nM | | | NPASS |
| LC-1F | Homo sapiens | | | = 409800.31 nM | | | NPASS |
| LC4-1 | Homo sapiens | | | = 360.29 nM | | | NPASS |
| LCLC-103H cell line | | | | = 345.6 nM | | | NPASS |
| LCLC-97TM1 | Homo sapiens | | | = 613.12 nM | | | NPASS |
| LK-2 | Homo sapiens | | | = 8570.71 nM | | | NPASS |
| LN-405 | Homo sapiens | | | = 6914.68 nM | | | NPASS |
| LNCaP-Clone-FGC | Homo sapiens | | | = 41593.88 nM | | | NPASS |
| LOUCY | Homo sapiens | | | = 586.06 nM | | | NPASS |
| LOX IMVI | Homo sapiens | | | = 411.85 nM | | | NPASS |
| LC-2-ad | Homo sapiens | | | = 952.55 nM | | | NPASS |
| LAMA-84 | Homo sapiens | | | = 1209.53 nM | | | NPASS |
| L929 | Mus musculus | | | = 3200.0 nM | | | NPASS |
| L02 | Homo sapiens | | | = 3410.0 nM|= 13000.0 nM|= 6220.0 nM|= 65340.0 nM|= 3257.0 nM|= 5120.0 nM|= 10520.0 nM|= 10450.0 nM|= 83800.0 nM | | | NPASS |
| KP-N-YS | Homo sapiens | | | = 351.7 nM | | | NPASS |
| KS-1 | Homo sapiens | | | = 41.5 nM | | | NPASS |
| KU-19-19 | Homo sapiens | | | = 3183.07 nM | | | NPASS |
| KU812 cell line | | | | = 8.306 nM | | | NPASS |
| KURAMOCHI | Homo sapiens | | | = 3159.36 nM | | | NPASS |
| KY821 | Homo sapiens | | | = 746.85 nM | | | NPASS |
| KYSE-140 | Homo sapiens | | | = 373.93 nM | | | NPASS |
| KYSE-150 cell line | | | | = 901.94 nM | | | NPASS |
| KYSE-180 | Homo sapiens | | | = 1010.32 nM | | | NPASS |
| KYSE-270 | Homo sapiens | | | = 216.92 nM | | | NPASS |
| KYSE-410 | Homo sapiens | | | = 752.42 nM | | | NPASS |
| KYSE-450 | Homo sapiens | | | = 138.15 nM | | | NPASS |
| KYSE-510 | Homo sapiens | | | = 252.7 nM | | | NPASS |
| KYSE-520 cell line | | | | = 598.42 nM | | | NPASS |
| KYSE-70 cell line | | | | = 2415.66 nM | | | NPASS |
| Kasumi 1 | | | | = 123.71 nM | | | NPASS |
| L-363 | Homo sapiens | | | = 75850.1 nM | | | NPASS |
| L-428 | Homo sapiens | | | = 1205.02 nM | | | NPASS |
| L-540 | Homo sapiens | | | = 4900.04 nM | | | NPASS |
| KOSC-2 | Homo sapiens | | | = 1490.84 nM | | | NPASS |
| Histone-lysine N-methyltransferase SETD7 | Homo sapiens | Q8WTS6 | | = 21620.0 nM | | | NPASS |
| IGR-1 | Homo sapiens | | | = 153.98 nM | | | NPASS |
| HeLa | Homo sapiens | | | = 13390.0 nM|= 6420.0 nM|= 2450.0 nM|= 6860.0 nM|= 6500.0 nM|= 7840.0 nM|= 2818.0 nM|= 11070.0 nM|= 5750.0 nM|= 6440.0 nM|= 4800.0 nM|= 9230.0 nM|= 3110.0 nM | | | NPASS |
| GCIY | Homo sapiens | | | = 35.98 nM | | | NPASS |
| GCT | Homo sapiens | | | = 1151.53 nM | | | NPASS |
| GDM-1 | Homo sapiens | | | = 2676.06 nM | | | NPASS |
| GI-1 | Homo sapiens | | | = 568.29 nM | | | NPASS |
| GI-ME-N | Homo sapiens | | | = 551.75 nM | | | NPASS |
| GMS-10 | Homo sapiens | | | = 11494.56 nM | | | NPASS |
| GOTO | Homo sapiens | | | = 4588.35 nM | | | NPASS |
| GP5d | Homo sapiens | | | = 1337.76 nM | | | NPASS |
| GB-1 | Homo sapiens | | | = 1329.99 nM | | | NPASS |
| HepG2 | Homo sapiens | | | = 240.0 nM|= 28100.0 nM|= 6920.0 nM|= 2920.0 nM|= 920.0 nM|= 2730.0 nM|= 1288.0 nM|= 9360.0 nM|= 420.0 nM | | | NPASS |
| H4 | Homo sapiens | | | = 283.93 nM | | | NPASS |
| HAL-01 | Homo sapiens | | | = 195.73 nM | | | NPASS |
| HC-1 | Homo sapiens | | | = 17215.51 nM | | | NPASS |
| HCC 2998 | Homo sapiens | | | = 46035.14 nM | | | NPASS |
| HCC1143 | Homo sapiens | | | = 529.69 nM | | | NPASS |
| HCC1187 | Homo sapiens | | | = 1019.79 nM | | | NPASS |
| HCC1395 | Homo sapiens | | | = 15686.74 nM | | | NPASS |
| HCC1419 | Homo sapiens | | | = 1689.76 nM | | | NPASS |
| GT3TKB | Homo sapiens | | | = 345.5 nM | | | NPASS |
| GAMG | Homo sapiens | | | = 1709.71 nM | | | NPASS |
| GAK | Homo sapiens | | | = 1037.69 nM | | | NPASS |
| G-402 | Homo sapiens | | | = 881.67 nM | | | NPASS |
| ES7 | Homo sapiens | | | = 548.49 nM | | | NPASS |
| ES8 | Homo sapiens | | | = 777.79 nM | | | NPASS |
| ESS-1 | Homo sapiens | | | = 34139.91 nM | | | NPASS |
| ETK-1 | Homo sapiens | | | = 2445.68 nM | | | NPASS |
| EVSA-T | Homo sapiens | | | = 409.8 nM | | | NPASS |
| EW-1 | Homo sapiens | | | = 843.9 nM | | | NPASS |
| EW-11 | Homo sapiens | | | = 447.16 nM | | | NPASS |
| EW-13 | Homo sapiens | | | = 266.74 nM | | | NPASS |
| EW-16 | Homo sapiens | | | = 299.15 nM | | | NPASS |
| EW-18 | Homo sapiens | | | = 528.62 nM | | | NPASS |
| EW-24 | Homo sapiens | | | = 14592.71 nM | | | NPASS |
| EW-3 | Homo sapiens | | | = 721.5 nM | | | NPASS |
| EW-7 | Homo sapiens | | | = 1290.91 nM | | | NPASS |
| Epidermal growth factor receptor erbB1 | Homo sapiens | P00533 | | = 139.2 nM | | | NPASS |
| FTC-133 | Homo sapiens | | | = 5743.15 nM | | | NPASS |
| FaDu | Homo sapiens | | | = 1766.39 nM | | | NPASS |
| Fibroblast | Homo sapiens | | | = 1200.0 nM|= 1240.0 nM | | | NPASS |
| G-361 | Homo sapiens | | | = 473.21 nM | | | NPASS |
| G-401 | Homo sapiens | | | = 234.92 nM | | | NPASS |
| HCC1569 | Homo sapiens | | | = 809.94 nM | | | NPASS |
| HCC1599 | Homo sapiens | | | = 388.27 nM | | | NPASS |
| GR-ST | Homo sapiens | | | = 102.18 nM | | | NPASS |
| HCC1937 | Homo sapiens | | | = 1662.86 nM | | | NPASS |
| HN | Homo sapiens | | | = 1367.64 nM | | | NPASS |
| HO-1-N-1 | Homo sapiens | | | = 462.12 nM | | | NPASS |
| HOP-62 | Homo sapiens | | | = 1160.87 nM | | | NPASS |
| HOP-92 | Homo sapiens | | | = 2010.24 nM | | | NPASS |
| HOS | Homo sapiens | | | = 186.08 nM | | | NPASS |
| HPAF-II | Homo sapiens | | | = 1266.25 nM | | | NPASS |
| HSC-2 | Homo sapiens | | | = 223.18 nM | | | NPASS |
| HSC-3 | Homo sapiens | | | = 336.66 nM | | | NPASS |
| HMV-2 cell line | | | | = 56.4 nM | | | NPASS |
| HSC-4 | Homo sapiens | | | = 2118.83 nM | | | NPASS |
| HT-1080 | Homo sapiens | | | = 259.95 nM | | | NPASS |
| HT-1376 | Homo sapiens | | | = 915.31 nM | | | NPASS |
| HT-144 | Homo sapiens | | | = 561.17 nM | | | NPASS |
| HT-29 | Homo sapiens | | | = 16700.0 nM|= 15800.0 nM|= 644.57 nM|= 2800.0 nM | | | NPASS |
| HT-3 | Homo sapiens | | | = 948.27 nM | | | NPASS |
| HT1197 | Homo sapiens | | | = 275.82 nM | | | NPASS |
| HT55 | Homo sapiens | | | = 1689.62 nM | | | NPASS |
| HTC-C3 | Homo sapiens | | | = 542.37 nM | | | NPASS |
| HCC1806 | Homo sapiens | | | = 1270.34 nM | | | NPASS |
| HLE | Homo sapiens | | | = 88.31 nM | | | NPASS |
| HT | Homo sapiens | | | = 1087.45 nM | | | NPASS |
| HH | Homo sapiens | | | = 1117.63 nM | | | NPASS |
| HCC2157 | Homo sapiens | | | = 337.83 nM | | | NPASS |
| HCC2218 | Homo sapiens | | | = 496.03 nM | | | NPASS |
| HCC38 | Homo sapiens | | | = 786.51 nM | | | NPASS |
| HCC70 | Homo sapiens | | | = 2008.36 nM | | | NPASS |
| HCC827 | Homo sapiens | | | = 9210.0 nM | | | NPASS |
| HCE-4 | Homo sapiens | | | = 388.84 nM | | | NPASS |
| HCE-T | Homo sapiens | | | = 720.09 nM | | | NPASS |
| HL-60 | Homo sapiens | | | = 440.0 nM|= 1030.0 nM|= 1923.05 nM|= 1200.0 nM | | | NPASS |
| HCC1954 | Homo sapiens | | | = 901.82 nM | | | NPASS |
| HCT-116 | Homo sapiens | | | = 230.0 nM|= 386.26 nM|= 1840.0 nM|= 2470.0 nM | | | NPASS |
| HCT-8 | Homo sapiens | | | = 9200.0 nM | | | NPASS |
| HD-MY-Z | Homo sapiens | | | = 470.14 nM | | | NPASS |
| HDLM-2 | Homo sapiens | | | = 89557.42 nM | | | NPASS |
| HEC-1 | Homo sapiens | | | = 1134.41 nM | | | NPASS |
| HEK-293T | Homo sapiens | | | = 62760.0 nM|= 1520.0 nM|= 2630.0 nM|= 9270.0 nM | | | NPASS |
| HEL | Homo sapiens | | | = 2043.04 nM | | | NPASS |
| HFF-1 | Homo sapiens | | | < 5000.0 nM | | | NPASS |
| HGC-27 | Homo sapiens | | | = 228.34 nM | | | NPASS |
| HCT-15 | Homo sapiens | | | = 7300.0 nM|= 267.58 nM|= 860.0 nM|= 940.0 nM | | | NPASS |