| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Xanthine dehydrogenase | Homo sapiens | P47989 | | = 840.0 nM | | | NPASS |
| Dipeptidyl peptidase IV | Homo sapiens | P27487 | | = 280.0 nM | | | NPASS |
| Glycogen synthase kinase-3 beta | Homo sapiens | P49841 | | 26900 nM|= 26900.0 nM | | | BindingDB, NPASS |
| HeLa | Homo sapiens | | > 10000.0 nM | | | | NPASS |
| Histone deacetylase 6 | Homo sapiens | Q9UBN7 | | = 998.0 nM | | | NPASS |
| Lysine-specific histone demethylase 1 | Homo sapiens | O60341 | | = 78760.0 nM | | | NPASS |
| Lysine-specific histone demethylase 1A | Homo sapiens | O60341 | | 78760 nM | | | BindingDB |
| MCF7 | Homo sapiens | | > 10000.0 nM | | | | NPASS |
| Mitogen-activated protein kinase 14 | Homo sapiens | Q16539 | | 5.46e+4 nM | | | BindingDB |
| PC-3 | Homo sapiens | | | = 90000.0 nM|= 40000.0 nM | | | NPASS |
| RPMI-8226 | Homo sapiens | | > 10000.0 nM | | | | NPASS |
| Dipeptidyl peptidase 4 | Homo sapiens | P27487 | | 280 nM | | | BindingDB |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome coronavirus | P0C6X7 | | 60000 nM|8300 nM | 24500 nM | | BindingDB |
| SARS-CoV-2 | Severe acute respiratory syndrome coronavirus 2 | | | > 20000.0 nM|> 19952.62 nM | | | NPASS |
| THP-1 | Homo sapiens | | > 10000.0 nM | | | | NPASS |
| Trypanosoma brucei brucei | Trypanosoma brucei brucei | | | < 30000.0 nM | | | NPASS |
| U-266 | Homo sapiens | | > 10000.0 nM | | | | NPASS |
| RAW264.7 | Mus musculus | | | = 48590.0 nM|= 31200.0 nM | | | NPASS |
| Cytochrome P450 1B1 | Homo sapiens | Q16678 | | 511 nM|= 511.0 nM | | | BindingDB, NPASS |
| CCRF-CEM | Homo sapiens | | > 10000.0 nM | | | | NPASS |
| Cytochrome P450 1A1 | Homo sapiens | P04798 | | 2786 nM|= 2786.0 nM | | | BindingDB, NPASS |
| Cytochrome P450 1A2 | Homo sapiens | P05177 | | 34647 nM|= 34647.0 nM | | | BindingDB, NPASS |
| Acetylcholinesterase | Homo sapiens | P22303 | | 2476100 nM|= 2476100.0 nM | | | BindingDB, NPASS |
| Alpha-amylase 1A | Homo sapiens | P0DUB6 | | | | | BindingDB |
| BJ | Homo sapiens | | > 10000.0 nM | | | | NPASS |
| Butyrylcholinesterase | Equus caballus | Q9N1N9 | | = 1774100.0 nM | | | NPASS |
| Caco-2 | Homo sapiens | | | = 66670.0 nM | | | NPASS |
| Carbonic anhydrase 1 | Homo sapiens | P00915 | | | | >10000 nM | BindingDB |
| Carbonic anhydrase 12 | Homo sapiens | O43570 | | | | 454 nM | BindingDB |
| Alpha-glucosidase MAL62 | Saccharomyces cerevisiae | P07265 | | 149968 nM | | | BindingDB |
| Carbonic anhydrase 4 | Homo sapiens | P22748 | | | | 102 nM | BindingDB |
| Carbonic anhydrase 7 | Homo sapiens | P43166 | | | | 3.3 nM | BindingDB |
| Carbonic anhydrase I | Homo sapiens | P00915 | | | | > 10000.0 nM | NPASS |
| Carbonic anhydrase II | Homo sapiens | P00918 | | | | > 10000.0 nM | NPASS |
| Carbonic anhydrase IV | Homo sapiens | P22748 | | | | = 102.1 nM | NPASS |
| Carbonic anhydrase 2 | Homo sapiens | P00918 | | | | >10000 nM | BindingDB |
| Carbonic anhydrase VII | Homo sapiens | P43166 | | | | = 3.3 nM | NPASS |
| Carbonic anhydrase XII | Homo sapiens | O43570 | | | | = 454.1 nM | NPASS |
| Carboxylic ester hydrolase | Equus caballus | | | 1774100 nM | | | BindingDB |