| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Procathepsin L | Homo sapiens | P07711 | | | | 9300 nM | BindingDB |
| Rhodesain | Trypanosoma brucei rhodesiense | Q95PM0 | | | | = 5310.0 nM | NPASS |
| Telomerase reverse transcriptase | Homo sapiens | O14746 | | = 500.0 nM | | | NPASS |
| Transient receptor potential cation channel subfamily A member 1 | Homo sapiens | O75762 | 1910 nM|= 1910.0 nM | | | | BindingDB, NPASS |
| Plasmodium berghei | Plasmodium berghei | | | = 6800.0 nM|= 39400.0 nM | | | NPASS |
| Transient receptor potential cation channel subfamily V member 1 | Rattus norvegicus | O35433 | 51220 nM | | | | BindingDB |
| Trypanosoma brucei brucei | Trypanosoma brucei brucei | | | = 13800.0 nM | | | NPASS |
| U-937 | Homo sapiens | | | = 19700.0 nM | | | NPASS |
| Vanilloid receptor | Rattus norvegicus | O35433 | = 51220.0 nM | | | | NPASS |
| Transient receptor potential cation channel subfamily A member 1 | Mus musculus | Q8BLA8 | 1320 nM|= 1320.0 nM | | | | BindingDB, NPASS |
| Plasmodium yoelii | Plasmodium yoelii | | | = 40000.0 nM | | | NPASS |
| NCI-N87 | Homo sapiens | | | = 16800.0 nM | | | NPASS |
| Mitochondrial 2-oxodicarboxylate carrier | Homo sapiens | Q9BQT8 | | 11 nM|= 11.0 nM | | | BindingDB, NPASS |
| HeLa | Homo sapiens | | | = 103500.0 nM | | | NPASS |
| HT-29 | Homo sapiens | | | = 83800.0 nM | | | NPASS |
| HL-60 | Homo sapiens | | | = 5500.0 nM | | | NPASS |
| Daudi | Homo sapiens | | | = 35300.0 nM | | | NPASS |
| Cysteine protease | Trypanosoma brucei rhodesiense | | | | | 5310 nM | BindingDB |
| Cathepsin L | Homo sapiens | P07711 | | | | = 9300.0 nM | NPASS |
| Cathepsin B | Homo sapiens | P07858 | | | | 8600 nM|= 8600.0 nM | BindingDB, NPASS |
| Plasmodium falciparum | Plasmodium falciparum | | | = 5210.0 nM | | | NPASS |