| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Histone-lysine N-methyltransferase, H3 lysine-9 specific 3 | Homo sapiens | Q96KQ7 | | > 100000.0 nM | | | NPASS |
| SK-MES-1 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| Plasmodium falciparum | Plasmodium falciparum | | | = 5000.0 nM | | | NPASS |
| Monoamine oxidase A | Homo sapiens | P21397 | | = 122000.0 nM | | | NPASS |
| MRC5 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| M-phase inducer phosphatase 2 | Homo sapiens | P30305 | | 9510 nM | | | BindingDB |
| J82 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| Histone-lysine N-methyltransferase, H3 lysine-9 specific 5 | Homo sapiens | Q9H9B1 | | > 100000.0 nM | | | NPASS |
| Histone-lysine N-methyltransferase EHMT1 | Homo sapiens | Q9H9B1 | | >100000 nM | | | BindingDB |
| HL-60 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| Glutamate NMDA receptor | Rattus norvegicus | Q9R1M7 | | > 1000000.0 nM | | | NPASS |
| Dual specificity protein phosphatase 6 | Rattus norvegicus | Q64346 | | >50000 nM|> 50000.0 nM | | | BindingDB, NPASS |
| Dual specificity protein phosphatase 1 | Mus musculus | P28563 | | >50000 nM|> 50000.0 nM | | | BindingDB, NPASS |
| Dual specificity phosphatase Cdc25B | Homo sapiens | P30305 | | = 9510.0 nM | | | NPASS |
| AGS | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| A2780 | Homo sapiens | | | = 580.0 nM | | | NPASS |
| Histone-lysine N-methyltransferase EHMT2 | Homo sapiens | Q96KQ7 | | >100000 nM | | | BindingDB |