IMPPAT Phytochemical information: 
Hispidulin

Hispidulin
Bioactivity information
Target nameTarget organismUniProt identifierEC50IC50KdKiSource
Mitogen-activated protein kinase 14Homo sapiensQ165391.86e+4 nMBindingDB
NeuraminidaseInflueA virusB4URF0= 46300.0 nM|= 26000.0 nM|= 33200.0 nMNPASS
NeuraminidaseInflueA virus (A/Puerto Rico/8/1934(H1N1))P03468= 13.9 ug.mL-1NPASS
NeuraminidaseInflueA virus (A/WSN/1933(H1N1))P0347026000 nM|33200 nM|46300 nMBindingDB
NeuraminidaseInflueA virus (strain A/Puerto Rico/8/1934 H1N1)P0346846600 nM|46200 nMBindingDB
No relevant target= 19270.0 nMNPASS
Nuclear receptor subfamily 0 group B member 1Homo sapiensP51843>833.72 nM|> 833.72 nMBindingDB, NPASS
Receptor-type tyrosine-protein kinase FLT3Homo sapiensP36888440 nM|390 nM|230 nMBindingDB
n.a.> 67536.0 nMNPASS
Serine/threonine-protein kinase PIM1Homo sapiensP11309= 2710.0 nMNPASS
Serine/threonine-protein kinase pim-1Homo sapiensP113092710 nMBindingDB
Steroidogenic factor 1Homo sapiensQ13285>67536 nMBindingDB
Tyrosine-protein kinase receptor FLT3Homo sapiensP36888= 230.0 nM|= 440.0 nM|= 390.0 nMNPASS
Mitogen-activated protein kinase 10Homo sapiensP537793.48e+4 nMBindingDB
Peroxisome proliferator-activated receptor gammaMus musculusP372387300 nM|= 7300.0 nMBindingDB, NPASS
MV4-11Homo sapiens= 8200.0 nM|= 6800.0 nMNPASS
Cell division protein kinase 5Rattus norvegicusQ03114= 19100.0 nMNPASS
MAP kinase-interacting serine/threonine-protein kinase MNK1Homo sapiensQ9BUB5= 1205.0 nMNPASS
Adenosine A1 receptorRattus norvegicusP25099= 1610.0 nMNPASS
Adenosine A2a receptorRattus norvegicusP30543= 6480.0 nMNPASS
Adenosine receptor A1Rattus norvegicusP250991622 nM|1610 nMBindingDB
Adenosine receptor A2aRattus norvegicusP305437586 nM|6480 nMBindingDB
Cyclin-dependent kinase 5Rattus norvegicusQ0311419100 nMBindingDB
Dipeptidyl peptidase 4Sus scrofaP22411490 nMBindingDB
MOLM-13Homo sapiens= 6400.0 nM|= 7000.0 nMNPASS
GABA-A receptor; anion channelHomo sapiensQ16445= 1000.0 nMNPASS
Hepatitis C virusHepatitis C virus= 36300.0 nMNPASS
Influenza A virusInflueA virus= 24700.0 nMNPASS
MAP kinase signal-integrating kinase 2Homo sapiensQ9HBH9= 252.0 nMNPASS
MAP kinase-interacting serine/threonine-protein kinase 1Homo sapiensQ9BUB51205 nMBindingDB
MAP kinase-interacting serine/threonine-protein kinase 2Homo sapiensQ9HBH9252 nMBindingDB
Dipeptidyl peptidase IVSus scrofaP22411= 490.0 nMNPASS