
| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|---|---|---|---|---|---|---|
| Zinc finger protein GLI2 | Homo sapiens | P10070 | 910 nM|= 910.0 nM | BindingDB, NPASS | |||
| Zinc finger protein GLI1 | Homo sapiens | P08151 | 7100 nM|= 7100.0 nM | BindingDB, NPASS | |||
| Sensor histidine kinase yycG | Bacillus subtilis (strain 168) | Q45614 | > 500.0 ug.mL-1 | NPASS | |||
| SW480 | Homo sapiens | = 3.15 ug.mL-1 | NPASS | ||||
| PC-3 | Homo sapiens | = 9100.0 nM | NPASS | ||||
| P338 | Mus musculus | = 2.63 ug.mL-1 | NPASS | ||||
| RAW264.7 | Mus musculus | = 13600.0 nM | NPASS | ||||
| MCF7 | Homo sapiens | = 9.67 ug.mL-1 | NPASS | ||||
| HepG2 | Homo sapiens | = 13.34 ug.mL-1 | NPASS | ||||
| NON-PROTEIN TARGET | = 6.05 ug.mL-1 | NPASS | |||||
| HeLa | Homo sapiens | = 3.15 ug.mL-1 | NPASS | ||||
| DU-145 | Homo sapiens | = 5.5 nM|= 6900.0 nM | NPASS | ||||
| Cytochrome P450 3A4 | Homo sapiens | P08684 | 21800 nM|= 21800.0 nM | BindingDB, NPASS | |||
| Cytochrome P450 2D6 | Homo sapiens | P10635 | >100000 nM|> 100000.0 nM | BindingDB, NPASS |