| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Alpha-2C adrenergic receptor | Homo sapiens | P18825 | | 27.1 nM | | 0.13 nM|0.3 nM|0.78 nM|3.02 nM|0.55 nM|0.25 nM|0.500000 nM|2.3 nM|1.9 nM|0.800000 nM | BindingDB |
| Alpha-2C adrenergic receptor | Didelphis virgia | P35405 | | | | 20 nM|0.08 nM|0.4 nM | BindingDB |
| Alpha-2B adrenergic receptor | Rattus norvegicus | P19328 | | | | 0.45 nM|1 nM|100 nM|16.8 nM|2 nM | BindingDB |
| Alpha-2B adrenergic receptor | Oryctolagus cuniculus | O77830 | | | | 21 nM|13.5 nM|11.3 nM|21.5 nM|13 nM | BindingDB |
| Alpha-2B adrenergic receptor | Homo sapiens | P18089 | | | | 0.37 nM|1.18 nM|77 nM|0.32 nM|1.2 nM|4.59 nM|13.6 nM|1.20 nM|1.99 nM|2 nM|4.6 nM|15 nM | BindingDB |
| Alpha-2B adrenergic receptor | Didelphis virgia | O77715 | | | | 28 nM|0.04 nM|0.18 nM|0.11 nM|0.19 nM | BindingDB |
| Alpha-2B adrenergic receptor | Canis lupus familiaris | | | | | 2 nM | BindingDB |
| Alpha-2C adrenergic receptor | Oithonidae environme sample | | | | | 0.12 nM|0.19 nM|28 nM|0.04 nM|0.18 nM | BindingDB |
| Alpha-2A/Alpha-2B/Alpha-2C adrenergic receptor | Homo sapiens | P08913|P18089|P18825 | | 170 nM|398000 nM|195000 nM|1800 nM|8.0 nM | 150000 nM|2300 nM|5400000 nM|47000 nM | | BindingDB |
| Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor | Rattus norvegicus | P19328|P22086|P22909 | | 165 nM|9.1 nM | | 13 nM|10 nM|150 nM|48 nM|45 nM|78 nM|190 nM|84 nM|56 nM | BindingDB |
| Alpha-2A adrenergic receptor [16-465] | Rattus norvegicus | P22909 | | 95 nM | | 19 nM|63.09 nM|63.6 nM|66 nM|59 nM | BindingDB |
| Alpha-2A adrenergic receptor | Sus scrofa | | | | | 0.26 nM|0.37 nM|4.4 nM | BindingDB |
| Alpha-2A adrenergic receptor | Mus musculus | | | | | 36.31 nM|61.66 nM | BindingDB |
| Alpha-2A adrenergic receptor | Homo sapiens | P08913 | 8.5 nM | 3.67 nM | | 0.32 nM|0.44 nM|0.5 nM|0.65 nM|132 nM|2.7 nM|1.6 nM|3.6 nM|0.43 nM|0.61 nM|3.76 nM|3.71 nM|0.71 nM|1.20 nM|7.94 nM|6.3 nM|3.16 nM|2.5 nM|3.5 nM|0.420000 nM|7.5 nM|3.1 nM|1.8 nM | BindingDB |
| Alpha-2A adrenergic receptor | Cavia porcellus | Q60474 | | | | 6 nM|15 nM | BindingDB |
| Alpha-2A adrenergic receptor | Bos taurus | Q28838 | | | | 3.38 nM|9.77 nM|9.5 nM|49 nM | BindingDB |
| Alpha-1D adrenergic receptor | Rattus norvegicus | P23944 | | | | 52 nM | BindingDB |
| Alpha-2C adrenergic receptor | Rattus norvegicus | P22086 | | | | 17 nM|6 nM|19 nM|10 nM|13 nM|0.83 nM|0.72 nM|2271 nM|14.3 nM|1.2 nM|7857 nM|43 nM|40 nM|320 nM|120 nM|18 nM|200 nM|0.44 nM|0.56 nM|31.62 nM|10.6 nM | BindingDB |
| Nischarin | Rattus norvegicus | Q4G017 | | | | >10000 nM | BindingDB |
| Cytochrome P450 2D6 | Homo sapiens | P10635 | | 8.4 nM | | 190 nM|180 nM|140 nM|230 nM|520 nM | BindingDB |
| Zinc finger protein mex-5 | Caenorhabditis elegans | Q9XUB2 | 103486 nM | | | | BindingDB |
| Voltage-dependent L-type calcium channel subunit alpha-1C | Rattus norvegicus | P22002 | | | | 1000 nM|>10000 nM|45 nM | BindingDB |
| Sodium-dependent serotonin transporter | Homo sapiens | P31645 | | | | 1000 nM | BindingDB |
| Sodium-dependent noradrenaline transporter | Homo sapiens | P23975 | | >20000 nM | | | BindingDB |
| Sodium-dependent dopamine transporter | Rattus norvegicus | P23977 | | | | 1000 nM | BindingDB |
| Sodium channel protein type 1/2/3 subunit alpha | Homo sapiens | P35498|Q99250|Q9NY46 | | 33000 nM | | | BindingDB |
| Sigma non-opioid intracellular receptor 1 | Rattus norvegicus | Q9R0C9 | | | | >10000 nM | BindingDB |
| POsterior Segregation | Caenorhabditis elegans | | 300000 nM | | | | BindingDB |
| M-phase inducer phosphatase 1 | Homo sapiens | P30304 | | 22300 nM | | | BindingDB |
| Importin subunit alpha-1 | Homo sapiens | P52292 | >500000 nM | | | | BindingDB |
| DNA topoisomerase 1 | Homo sapiens | P11387 | | 30000 nM | | | BindingDB |
| D(3) dopamine receptor | Rattus norvegicus | P19020 | | | | 2430 nM | BindingDB |
| D(3) dopamine receptor | Homo sapiens | P35462 | | | | 2489 nM|3981.07 nM | BindingDB |
| D(2) dopamine receptor | Rattus norvegicus | P61169 | | 1125 nM | | 158 nM|926 nM|501.18 nM | BindingDB |
| D(2) dopamine receptor | Homo sapiens | P14416 | | | | 280 nM|398.1 nM | BindingDB |
| D(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor | Rattus norvegicus | P18901|P19020|P25115|P30729|P61169 | | | | 2000 nM | BindingDB |
| D(1A) dopamine receptor | Homo sapiens | P21728 | | | | >10000 nM | BindingDB |
| Bile salt export pump | Homo sapiens | O95342 | | 254000 nM | | | BindingDB |
| Alpha-1B adrenergic receptor | Rattus norvegicus | P15823 | | | | 517 nM | BindingDB |
| Alpha-1D adrenergic receptor | Homo sapiens | P25100 | | | | 158.48 nM|954.99 nM|1.6 nM|289 nM | BindingDB |
| Alpha-1B adrenergic receptor | Homo sapiens | P35368 | | | | 158.48 nM|2398.83 nM|1.1 nM|7.2 nM|966 nM | BindingDB |
| 5-hydroxytryptamine receptor 2A | Homo sapiens | P28223 | | | | >10000 nM|1000 nM|252 nM|288.4 nM|3467.36 nM | BindingDB |
| 5-hydroxytryptamine receptor 1F | Rattus norvegicus | P30940 | | | | 562.34 nM | BindingDB |
| 5-hydroxytryptamine receptor 1F | Mus musculus | Q02284 | | | | 63.09 nM | BindingDB |
| 5-hydroxytryptamine receptor 1F | Homo sapiens | P30939 | | | | 91.2 nM|92 nM | BindingDB |
| 5-hydroxytryptamine receptor 1E | Homo sapiens | P28566 | | | | 3434 nM|1270 nM|1258.92 nM | BindingDB |
| 5-hydroxytryptamine receptor 1D | Rattus norvegicus | P28565 | | | | 30.9 nM | BindingDB |
| 5-hydroxytryptamine receptor 1D | Homo sapiens | P28221 | | | | 40 nM|27 nM|59 nM|51 nM|15.84 nM|58.88 nM|47.86 nM|21.87 nM|19.95 nM|25.11 nM | BindingDB |
| 5-hydroxytryptamine receptor 1D | Canis lupus familiaris | P11614 | | | | 5.24 nM|32.35 nM | BindingDB |
| 5-hydroxytryptamine receptor 1B | Rattus norvegicus | P28564 | | | | 8700 nM|7540 nM|6309.57 nM|4466.83 nM|151.35 nM | BindingDB |
| 5-hydroxytryptamine receptor 1B | Mus musculus | P28334 | | | | >10000 nM | BindingDB |
| 5-hydroxytryptamine receptor 1B | Homo sapiens | P28222 | | | | 5 nM|16 nM|22 nM|39.81 nM|46.77 nM|251.18 nM|26.91 nM|40.73 nM|5.01 nM|158.48 nM | BindingDB |
| 5-hydroxytryptamine receptor 1B | Cavia porcellus | O08892 | | | | 50.11 nM | BindingDB |
| 5-hydroxytryptamine receptor 1A/1B/1D/2C | Homo sapiens | P08908|P28221|P28222|P28335 | | | | 4500 nM | BindingDB |
| 5-hydroxytryptamine receptor 1A | Rattus norvegicus | P19327 | | | | 1318.26 nM|1548.82 nM|125.89 nM | BindingDB |
| 5-hydroxytryptamine receptor 1A | Homo sapiens | P08908 | | | | 1500 nM|642 nM|1258.92 nM|50.11 nM | BindingDB |
| 5-hydroxytryptamine 1D receptor | Bos taurus | | | | | 20 nM|79 nM | BindingDB |
| Alpha-1B adrenergic receptor | Mesocricetus auratus | P18841 | | | | 670 nM | BindingDB |
| 5-hydroxytryptamine receptor 2A | Rattus norvegicus | P14842 | | | | >10000 nM|2258 nM|1000 nM|1621.81 nM | BindingDB |
| 5-hydroxytryptamine receptor 2B | Homo sapiens | P41595 | | | | 398.1 nM|40.6 nM|15.1 nM|44.4 nM|28.84 nM|50.11 nM|14.3 nM|4.12 nM|43.2 nM|13.2 nM|31.62 nM|398.11 nM | BindingDB |
| Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor | Rattus norvegicus | P15823|P23944|P43140 | | 1300 nM|1000 nM | | 398 nM|360 nM | BindingDB |
| 5-hydroxytryptamine receptor 2C | Homo sapiens | P28335 | | | | >10000 nM|1690 nM|645.65 nM|1000 nM | BindingDB |
| 5-hydroxytryptamine receptor 2B | Rattus norvegicus | P30994 | | | | 50.11 nM|58.88 nM|35.48 nM|107.15 nM|53.7 nM|53.1 nM|35.8 nM|39.81 nM|50.12 nM | BindingDB |
| Alpha-1A adrenergic receptor | Oryctolagus cuniculus | O02824 | | | | 1100 nM|275 nM | BindingDB |
| Alpha-1A adrenergic receptor | Homo sapiens | P35348 | | | | 770 nM|199.52 nM|3162.28 nM|1057 nM | BindingDB |
| Alpha-1A adrenergic receptor | Canis lupus familiaris | O77621 | | | | 32 nM|13.4 nM | BindingDB |
| Alpha-1A adrenergic receptor | Bos taurus | P18130 | | | | 142 nM|220 nM|200 nM|3.6 nM | BindingDB |
| Acetylcholinesterase | Electrophorus electricus | O42275 | | 431000 nM | | | BindingDB |
| 5-hydroxytryptamine receptor 7 | Rattus norvegicus | P32305 | | | | 1000 nM | BindingDB |
| 5-hydroxytryptamine receptor 7 | Homo sapiens | P34969 | | | | 2850 nM | BindingDB |
| Alpha-1A adrenergic receptor | Rattus norvegicus | P43140 | | | | 150 nM|480 nM|562 nM|263 nM|64 nM|36 nM|236 nM|230 nM|1100 nM|251.18 nM | BindingDB |
| 5-hydroxytryptamine receptor 5B | Mus musculus | P31387 | | | | 1000 nM | BindingDB |
| 5-hydroxytryptamine receptor 5A | Rattus norvegicus | P35364 | | | | 1000 nM | BindingDB |
| 5-hydroxytryptamine receptor 5A | Mus musculus | P30966 | | | | 1000 nM|630.95 nM|>10000 nM | BindingDB |
| 5-hydroxytryptamine receptor 3A | Mus musculus | P23979 | | | | >10000 nM|1000 nM | BindingDB |
| 5-hydroxytryptamine receptor 2C | Sus scrofa | | | | | 1000 nM|1584.89 nM|>10000 nM | BindingDB |
| 5-hydroxytryptamine receptor 2C | Rattus norvegicus | P08909 | | | | >10000 nM|5011.87 nM | BindingDB |
| 5-hydroxytryptamine receptor 2C | Mus musculus | P34968 | | | | >10000 nM | BindingDB |
| 5-hydroxytryptamine receptor 5B | Rattus norvegicus | P35365 | | | | 1000 nM | BindingDB |