| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Alpha-2b adrenergic receptor | Homo sapiens | P18089 | | | | = 116.0 nM | NPASS |
| Alpha-2a adrenergic receptor | Rattus norvegicus | P22909 | | | | = 1210.0 nM | NPASS |
| Alpha-2c adrenergic receptor | Homo sapiens | P18825 | | | | = 28.0 nM | NPASS |
| Alpha-2a adrenergic receptor | Homo sapiens | P08913 | | | | = 106.0 nM | NPASS |
| Alpha-2C adrenergic receptor | Oithonidae environme sample | | | | | 20 nM|12 nM | BindingDB |
| Alpha-2A adrenergic receptor [16-465] | Rattus norvegicus | P22909 | | | | 1210 nM | BindingDB |
| Alpha-2B adrenergic receptor | Rattus norvegicus | P19328 | | | | 159 nM|208 nM | BindingDB |
| Alpha-2B adrenergic receptor | Homo sapiens | P18089 | | | | 116 nM | BindingDB |
| Alpha-2A adrenergic receptor | Homo sapiens | P08913 | | | | 71 nM|104 nM|130 nM|106 nM | BindingDB |
| Alpha-2A adrenergic receptor | Bos taurus | Q28838 | | | | 1826 nM | BindingDB |
| Alpha-2C adrenergic receptor | Homo sapiens | P18825 | | | | 28 nM | BindingDB |