| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| KB | Homo sapiens | | | = 27370.0 nM|= 31730.0 nM|= 41530.0 nM | | | NPASS |
| KBM5 | Homo sapiens | | | = 8500.0 nM | | | NPASS |
| enterovirus D68 | enterovirus D68 | | | = 3450.0 nM | | | NPASS |
| MCF7 | Homo sapiens | | | > 66000.0 nM|= 30820.0 nM|= 15400.0 nM|= 8480.0 nM|= 29060.0 nM|= 15000.0 nM|= 35100.0 nM | | | NPASS |
| MDA-MB-231 | Homo sapiens | | | = 16550.0 nM|> 30000.0 nM|= 20300.0 nM | | | NPASS |
| MDA-MB-361 | Homo sapiens | | | = 31500.0 nM | | | NPASS |
| NIH3T3 | Mus musculus | | | = 95280.0 nM | | | NPASS |
| NON-PROTEIN TARGET | | | | = 23300.0 nM|= 32520.0 nM|= 21240.0 nM | | | NPASS |
| Nuclear factor NF-kappa-B p105 subunit | Homo sapiens | P19838 | | 49600 nM|= 49600.0 nM | | | BindingDB, NPASS |
| RAW264.7 | Mus musculus | | | = 6960.0 nM|= 14420.0 nM | | | NPASS |
| PC-3 | Homo sapiens | | | = 30000.0 nM | | | NPASS |
| K562 | Homo sapiens | | | = 41850.0 nM|= 23660.0 nM | | | NPASS |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome coronavirus 2 | P0DTD1 | | 15000 nM|= 15000.0 nM | | | BindingDB, NPASS |
| SARS-CoV-2 | Severe acute respiratory syndrome coronavirus 2 | | | > 100000.0 nM|= 19030.0 nM|= 1680.0 nM|= 34.0 nM|= 280.0 nM|= 6580.0 nM | | | NPASS |
| Signal transducer and activator of transcription 3 | Homo sapiens | P40763 | >10000 nM|> 10000.0 nM | | | | BindingDB, NPASS |
| T47D | Homo sapiens | | | = 32400.0 nM | | | NPASS |
| THP-1 | Homo sapiens | | | = 6690.0 nM | | | NPASS |
| U-937 | Homo sapiens | | | = 12870.0 nM | | | NPASS |
| Zika virus | Zika virus | | = 39300.0 nM | | | | NPASS |
| P388 | Mus musculus | | | = 2250.0 nM|= 6520.0 nM|= 2900.0 nM | | | NPASS |
| Indoleamine 2,3-dioxygenase | Homo sapiens | P14902 | | = 56.0 ug.mL-1 | | | NPASS |
| L5178Y | Mus musculus | | | = 14520.0 nM|= 14950.0 nM | | | NPASS |
| Human immunodeficiency virus | Human immunodeficiency virus | | | = 7900.0 nM|= 2320.0 nM | | | NPASS |
| A2058 | Homo sapiens | | | = 26000.0 nM | | | NPASS |
| A549 | Homo sapiens | | | = 9.71 ug.mL-1|= 27900.0 nM|= 32020.0 nM|= 12150.0 nM | | | NPASS |
| ACHN | Homo sapiens | | | = 3.03 ug.mL-1 | | | NPASS |
| B16 | Mus musculus | | | = 7.54 ug.mL-1 | | | NPASS |
| BT-549 | Homo sapiens | | | = 23200.0 nM | | | NPASS |
| Bile acid receptor | Homo sapiens | Q96RI1 | | 9700 nM | | | BindingDB |
| Bile acid receptor FXR | Homo sapiens | Q96RI1 | | = 9700.0 nM | | | NPASS |
| Chikungunya virus | Chikunguvirus | | = 77000.0 nM | = 600.0 nM | | | NPASS |
| Dengue virus 2 | Dengue virus 2 | | = 21304.0 nM|= 22739.0 nM | | | | NPASS |
| BMMC | | | | = 1010.0 nM | | | NPASS |
| HK-2 | Homo sapiens | | | = 30600.0 nM | | | NPASS |
| HCT-116 | Homo sapiens | | | = 23930.0 nM|> 40000.0 nM|= 31800.0 nM | | | NPASS |
| HuCC-A1 | Homo sapiens | | | = 23610.0 nM | | | NPASS |
| Hexokinase-2 | Homo sapiens | P52789 | | >50000 nM | | | BindingDB |
| Hexokinase type II | Homo sapiens | P52789 | | > 50000.0 nM | | | NPASS |
| Human immunodeficiency virus 1 | Human immunodeficiency virus 1 | | | = 590.0 nM|= 588.84 nM | | | NPASS |
| HeLa | Homo sapiens | | | = 10.42 ug.mL-1 | | | NPASS |
| HT-29 | Homo sapiens | | | = 9340.0 nM|= 8910.0 nM|= 10800.0 nM|> 30000.0 nM | | | NPASS |
| HL-60 | Homo sapiens | | | = 27000.0 nM|= 2400.0 nM|= 7000.0 nM | | | NPASS |
| Hepatitis B virus | Hepatitis B virus | | | = 54100.0 nM | | | NPASS |