IMPPAT Phytochemical information: 
Andrographolide

Andrographolide
Bioactivity information
Target nameTarget organismUniProt identifierEC50IC50KdKiSource
KBHomo sapiens= 27370.0 nM|= 31730.0 nM|= 41530.0 nMNPASS
KBM5Homo sapiens= 8500.0 nMNPASS
enterovirus D68enterovirus D68= 3450.0 nMNPASS
MCF7Homo sapiens> 66000.0 nM|= 30820.0 nM|= 15400.0 nM|= 8480.0 nM|= 29060.0 nM|= 15000.0 nM|= 35100.0 nMNPASS
MDA-MB-231Homo sapiens= 16550.0 nM|> 30000.0 nM|= 20300.0 nMNPASS
MDA-MB-361Homo sapiens= 31500.0 nMNPASS
NIH3T3Mus musculus= 95280.0 nMNPASS
NON-PROTEIN TARGET= 23300.0 nM|= 32520.0 nM|= 21240.0 nMNPASS
Nuclear factor NF-kappa-B p105 subunitHomo sapiensP1983849600 nM|= 49600.0 nMBindingDB, NPASS
RAW264.7Mus musculus= 6960.0 nM|= 14420.0 nMNPASS
PC-3Homo sapiens= 30000.0 nMNPASS
K562Homo sapiens= 41850.0 nM|= 23660.0 nMNPASS
Replicase polyprotein 1abSevere acute respiratory syndrome coronavirus 2P0DTD115000 nM|= 15000.0 nMBindingDB, NPASS
SARS-CoV-2Severe acute respiratory syndrome coronavirus 2> 100000.0 nM|= 19030.0 nM|= 1680.0 nM|= 34.0 nM|= 280.0 nM|= 6580.0 nMNPASS
Signal transducer and activator of transcription 3Homo sapiensP40763>10000 nM|> 10000.0 nMBindingDB, NPASS
T47DHomo sapiens= 32400.0 nMNPASS
THP-1Homo sapiens= 6690.0 nMNPASS
U-937Homo sapiens= 12870.0 nMNPASS
Zika virusZika virus= 39300.0 nMNPASS
P388Mus musculus= 2250.0 nM|= 6520.0 nM|= 2900.0 nMNPASS
Indoleamine 2,3-dioxygenaseHomo sapiensP14902= 56.0 ug.mL-1NPASS
L5178YMus musculus= 14520.0 nM|= 14950.0 nMNPASS
Human immunodeficiency virusHuman immunodeficiency virus= 7900.0 nM|= 2320.0 nMNPASS
A2058Homo sapiens= 26000.0 nMNPASS
A549Homo sapiens= 9.71 ug.mL-1|= 27900.0 nM|= 32020.0 nM|= 12150.0 nMNPASS
ACHNHomo sapiens= 3.03 ug.mL-1NPASS
B16Mus musculus= 7.54 ug.mL-1NPASS
BT-549Homo sapiens= 23200.0 nMNPASS
Bile acid receptorHomo sapiensQ96RI19700 nMBindingDB
Bile acid receptor FXRHomo sapiensQ96RI1= 9700.0 nMNPASS
Chikungunya virusChikunguvirus= 77000.0 nM= 600.0 nMNPASS
Dengue virus 2Dengue virus 2= 21304.0 nM|= 22739.0 nMNPASS
BMMC= 1010.0 nMNPASS
HK-2Homo sapiens= 30600.0 nMNPASS
HCT-116Homo sapiens= 23930.0 nM|> 40000.0 nM|= 31800.0 nMNPASS
HuCC-A1Homo sapiens= 23610.0 nMNPASS
Hexokinase-2Homo sapiensP52789>50000 nMBindingDB
Hexokinase type IIHomo sapiensP52789> 50000.0 nMNPASS
Human immunodeficiency virus 1Human immunodeficiency virus 1= 590.0 nM|= 588.84 nMNPASS
HeLaHomo sapiens= 10.42 ug.mL-1NPASS
HT-29Homo sapiens= 9340.0 nM|= 8910.0 nM|= 10800.0 nM|> 30000.0 nMNPASS
HL-60Homo sapiens= 27000.0 nM|= 2400.0 nM|= 7000.0 nMNPASS
Hepatitis B virusHepatitis B virus= 54100.0 nMNPASS