| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Xanthine dehydrogenase/oxidase | Bos taurus | P80457 | | 176100 nM | | | BindingDB |
| Nitric oxide synthase, inducible | Mus musculus | P29477 | | 7800 nM|= 7800.0 nM | | | BindingDB, NPASS |
| Prostaglandin G/H synthase 2 | Homo sapiens | P35354 | | 46000 nM | | | BindingDB |
| MV4-11 | Homo sapiens | | | = 30700.0 nM | | | NPASS |
| MCF7 | Homo sapiens | | | = 28000.0 nM|= 30000.0 nM|= 30.0 nM | | | NPASS |
| NON-PROTEIN TARGET | | | | = 36870.0 nM | | | NPASS |
| Prostaglandin G/H synthase 2 | Mus musculus | Q05769 | | 1070 nM | | | BindingDB |
| Lysine-specific histone demethylase 1A | Homo sapiens | O60341 | | 8870 nM | | | BindingDB |
| RAW264.7 | Mus musculus | | | = 1080.0 nM | | | NPASS |
| SW1353 | Homo sapiens | | | = 39000.0 nM | | | NPASS |
| SW480 | Homo sapiens | | | = 35060.0 nM | | | NPASS |
| Serotonin 7 (5-HT7) receptor | Homo sapiens | P34969 | | > 350000.0 nM | | | NPASS |
| Trypsin | Homo sapiens | P07477|P07478|P35030 | | 105000 nM | | | BindingDB |
| Trypsin | Homo sapiens | P35030 | | = 105000.0 nM | | | NPASS |
| Xanthine dehydrogenase | Bos taurus | P80457 | | = 176100.0 nM | | | NPASS |
| Pyruvate kinase isozymes M1/M2 | Homo sapiens | P14618 | | = 2010.0 nM | | = 3530.0 nM | NPASS |
| Lysine-specific histone demethylase 1 | Homo sapiens | O60341 | | = 8870.0 nM | | | NPASS |
| Cyclin-dependent kinase 9 | Homo sapiens | P50750 | | 190 nM|= 190.0 nM | | | BindingDB, NPASS |
| HepG2 | Homo sapiens | | | = 37890.0 nM|= 19000.0 nM|= 19054.61 nM|= 19500.0 nM|= 17600.0 nM | | | NPASS |
| Hepatitis B virus | Hepatitis B virus | | | = 4.0 ug.mL-1 | | | NPASS |
| 5-hydroxytryptamine receptor 7 | Homo sapiens | P34969 | | >350000 nM | | | BindingDB |
| A549 | Homo sapiens | | | = 15800.0 nM|= 20100.0 nM|= 42300.0 nM | | | NPASS |
| B16 | Mus musculus | | | = 26400.0 nM | | | NPASS |
| CDK7/Cyclin H/MNAT1 | Homo sapiens | | | = 12300.0 nM | | | NPASS |
| CDK8/Cyclin C | Homo sapiens | | | = 5900.0 nM | | | NPASS |
| CDK9/cyclin T1 | Homo sapiens | P50750 | | = 190.0 nM|= 198.0 nM | | | NPASS |
| CDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7 | Homo sapiens | P50613|P51946|P51948 | | 12300 nM | | | BindingDB |
| Cyclin-T1/Cyclin-dependent kinase 9 | Homo sapiens | O60563|P50750 | | 198 nM|190 nM | | | BindingDB |
| Cyclin-dependent kinase 2 | Homo sapiens | P24941 | | 1460 nM|= 1460.0 nM | | | BindingDB, NPASS |
| Cyclooxygenase-2 | Homo sapiens | P35354 | | = 46000.0 nM | | | NPASS |
| Cyclooxygenase-2 | Mus musculus | Q05769 | | = 1070.0 nM | | | NPASS |
| GABA-A receptor; anion channel | Homo sapiens | Q16445 | | | | = 2041.74 nM | NPASS |
| HCT-116 | Homo sapiens | | | = 27300.0 nM | | | NPASS |
| HT-29 | Homo sapiens | | | = 39550.0 nM | | | NPASS |
| Cyclin-A2/Cyclin-dependent kinase 2 | Homo sapiens | P20248|P24941 | | 1460 nM | | | BindingDB |