| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| HeLa | Homo sapiens | | > 370000.0 nM | | | | NPASS |
| Trypanosoma brucei brucei | Trypanosoma brucei brucei | | | < 30000.0 nM | | | NPASS |
| SW480 | Homo sapiens | | | > 20000.0 nM | | | NPASS |
| P-glycoprotein 1 | Homo sapiens | P08183 | | | = 6309.57 nM | | NPASS |
| NON-PROTEIN TARGET | | | = 226000.0 nM|= 273000.0 nM | > 20000.0 nM | | | NPASS |
| MCF7 | Homo sapiens | | | = 51.05 ug.mL-1 | | | NPASS |
| HepG2 | Homo sapiens | | | > 20000.0 nM | | | NPASS |
| HT-29 | Homo sapiens | | | > 20000.0 nM | | | NPASS |
| RBL-2H3 | Rattus norvegicus | | | = 49000.0 nM | | | NPASS |
| COLO 205 | Homo sapiens | | | = 37.14 ug.mL-1 | | | NPASS |
| CHO | Cricetulus griseus | | | = 23.54 ug.mL-1 | | | NPASS |
| Broad substrate specificity ATP-binding cassette transporter ABCG2 | Homo sapiens | Q9UNQ0 | | 3000 nM | | | BindingDB |
| ATP-dependent translocase ABCB1 | Homo sapiens | P08183 | | | 6310 nM | | BindingDB |
| ATP-binding cassette sub-family G member 2 | Homo sapiens | Q9UNQ0 | | = 3000.0 nM | | | NPASS |
| A549 | Homo sapiens | | > 370000.0 nM | = 49.56 ug.mL-1 | | | NPASS |
| A-431 | Homo sapiens | | | = 39.02 ug.mL-1 | | | NPASS |
| HT-1080 | Homo sapiens | | = 358000.0 nM | | | | NPASS |