| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| U-251 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| Solute carrier organic anion transporter family member 1B3 | Homo sapiens | Q9NPD5 | | 105 nM|= 104.71 nM | | 130 nM|= 80.0 nM | BindingDB, NPASS |
| Solute carrier organic anion transporter family member 1B1 | Homo sapiens | Q9Y6L6 | | 245 nM|= 245.47 nM | | 130 nM|= 130.0 nM | BindingDB, NPASS |
| MCF7 | Homo sapiens | | | = 49230.0 nM | | | NPASS |
| THP-1 | Homo sapiens | | | = 3300.0 nM | | | NPASS |
| Hep 3B2 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| Bcap37 | Homo sapiens | | | > 100000.0 nM | | | NPASS |
| Amyloid-beta precursor protein | Homo sapiens | P05067 | | >100000 nM | | | BindingDB |
| A549 | Homo sapiens | | | = 38150.0 nM | | | NPASS |
| HepG2 | Homo sapiens | | | = 40340.0 nM | | | NPASS |