| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| K562 | Homo sapiens | | | = 16100.0 nM|= 6000.0 nM|= 17000.0 nM|= 13600.0 nM|= 14000.0 nM | | | NPASS |
| KB | Homo sapiens | | | = 3800.0 nM|> 500000.0 nM | | | NPASS |
| MCF7 | Homo sapiens | | = 25900.0 nM|= 12000.0 nM | = 49000.0 nM|= 29000.0 nM|= 10370.0 nM|= 19.32 ug.mL-1|= 10420.0 nM|= 18200.0 nM|> 10000.0 nM|> 500000.0 nM | | | NPASS |
| MDA-MB-231 | Homo sapiens | | | = 9770.0 nM|> 20.0 ug.mL-1|> 500000.0 nM | | | NPASS |
| MGC-803 | Homo sapiens | | | = 17700.0 nM | | | NPASS |
| MIA PaCa-2 | Homo sapiens | | | > 10000.0 nM | | | NPASS |
| Influenza A virus | InflueA virus | | = 5700.0 nM | | | | NPASS |
| MRC5 | Homo sapiens | | | = 29500.0 nM|= 30000.0 nM | | | NPASS |
| NIH3T3 | Mus musculus | | = 19400.0 nM | | | | NPASS |
| NON-PROTEIN TARGET | | | = 29000.0 nM | = 10420.0 nM|= 10050.0 nM|= 13.81 ug.mL-1|= 16.77 ug.mL-1|= 44.71 ug.mL-1|> 50.0 ug.mL-1|= 127.64 ug.mL-1|= 12930.0 nM|= 13900.0 nM|= 14000.0 nM | | | NPASS |
| PC-3 | Homo sapiens | | | = 15000.0 nM|> 10000.0 nM | | | NPASS |
| Semliki forest virus | Semliki forest virus | | | = 13300.0 nM|= 13182.57 nM | | | NPASS |
| SARS coronavirus | SARS coronavirus | | = 630.0 nM | | | | NPASS |
| SK-MEL-2 | Homo sapiens | | | = 26000.0 nM | | | NPASS |
| SW-1736 | Homo sapiens | | | = 3050.0 nM | | | NPASS |
| SW948 | Homo sapiens | | | = 19170.0 nM | | | NPASS |
| SiHa | Homo sapiens | | | > 500000.0 nM | | | NPASS |
| Streptococcus | Streptococcus | | = 2880.0 nM | | | | NPASS |
| Streptococcus sp. 'group A' | Streptococcus sp. 'group A' | | = 1684.0 nM | | | | NPASS |
| Streptokinase A | Streptococcus pyogenes serotype M1 | P10520 | = 1848.0 nM | | | | NPASS |
| U2OS | Homo sapiens | | | = 38000.0 nM | | | NPASS |
| Vero | Chlorocebus aethiops | | | > 500000.0 nM | | | NPASS |
| Human immunodeficiency virus 1 | Human immunodeficiency virus 1 | | = 0.22 ug.mL-1 | = 21400.0 nM | | | NPASS |
| Plasmodium falciparum | Plasmodium falciparum | | | = 7870.0 nM | | | NPASS |
| Human herpesvirus 1 | Human herpesvirus 1 | | = 2500.0 nM | = 5700.0 nM | | | NPASS |
| FaDu | Homo sapiens | | = 17400.0 nM | | | | NPASS |
| HeLa | Homo sapiens | | | > 500000.0 nM | | | NPASS |
| 8505C | Homo sapiens | | | = 14000.0 nM | | | NPASS |
| A-375 | Homo sapiens | | = 14300.0 nM | = 28900.0 nM | | | NPASS |
| A-431 | Homo sapiens | | | = 3260.0 nM | | | NPASS |
| A2780 | Homo sapiens | | = 20400.0 nM|= 4700.0 nM | = 2980.0 nM|= 5970.0 nM | | | NPASS |
| A549 | Homo sapiens | | = 25900.0 nM | = 15000.0 nM|= 10090.0 nM|= 8.93 ug.mL-1|= 10420.0 nM|= 5700.0 nM|= 40000.0 nM | | | NPASS |
| BJ | Homo sapiens | | | = 39500.0 nM|= 39000.0 nM | | | NPASS |
| BV-2 | Mus musculus | | | > 100000.0 nM|= 60700.0 nM | | | NPASS |
| Bcap37 | Homo sapiens | | | = 25700.0 nM | | | NPASS |
| Bile acid receptor FXR | Homo sapiens | Q96RI1 | = 0.0 nM | | | | NPASS |
| Botulinum neurotoxin type A | Clostridium botulinum | P10845 | | < 100000.0 nM | | | NPASS |
| CCRF-CEM | Homo sapiens | | | = 20000.0 nM|= 17000.0 nM|= 8400.0 nM | | | NPASS |
| CEM-DNR | Homo sapiens | | | = 11000.0 nM | | | NPASS |
| COLO 205 | Homo sapiens | | | = 36800.0 nM | | | NPASS |
| Ca9-22 | Homo sapiens | | | = 14.47 ug.mL-1 | | | NPASS |
| DU-145 | Homo sapiens | | | = 36000.0 nM|> 500000.0 nM | | | NPASS |
| ECV-304 | Homo sapiens | | | < 4.0 ug.mL-1|= 0.28 ug.mL-1 | | | NPASS |
| G-protein coupled bile acid receptor 1 | Homo sapiens | Q8TDU6 | 4710 nM|= 4710.0 nM | | | | BindingDB, NPASS |
| H9 | Homo sapiens | | | = 1.8 ug.mL-1 | | | NPASS |
| HCT-116 | Homo sapiens | | | = 2610.0 nM|> 10000.0 nM|= 38100.0 nM|= 49400.0 nM|= 38000.0 nM | | | NPASS |
| HEK293 | Homo sapiens | | | > 500000.0 nM | | | NPASS |
| HEp-2 | Homo sapiens | | | > 500000.0 nM | | | NPASS |
| HT-29 | Homo sapiens | | = 18500.0 nM | = 17000.0 nM|= 10020.0 nM | | | NPASS |
| 5'-nucleotidase | Homo sapiens | P21589 | | = 43260.0 nM | | | NPASS |
| HepG2 | Homo sapiens | | | = 4.32 ug.mL-1 | | | NPASS |