
| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|---|---|---|---|---|---|---|
| NCI-H226 | Homo sapiens | > 10000.0 nM | NPASS | ||||
| HL-60 | Homo sapiens | = 7500.0 nM | NPASS | ||||
| HCT-116 | Homo sapiens | = 8800.0 nM | NPASS | ||||
| Cyclin-T1/Cyclin-dependent kinase 9 | Homo sapiens | O60563|P50750 | 300 nM | BindingDB | |||
| MCF7 | Homo sapiens | > 10000.0 nM | NPASS | ||||
| CDK9/cyclin T1 | Homo sapiens | P50750 | = 300.0 nM | NPASS | |||
| CDK2/Cyclin A | Homo sapiens | P20248 | = 7300.0 nM | NPASS | |||
| A549 | Homo sapiens | > 10000.0 nM | NPASS | ||||
| Cyclin-A2/Cyclin-dependent kinase 2 | Homo sapiens | P20248|P24941 | 7300 nM | BindingDB |