| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Xanthine dehydrogenase | Homo sapiens | P47989 | | = 213000.0 nM | | | NPASS |
| XF498 | Homo sapiens | | | = 18750.0 nM | | | NPASS |
| Testis-specific androgen-binding protein | Homo sapiens | P04278 | | = 230000.0 nM | | | NPASS |
| SK-OV-3 | Homo sapiens | | | > 30000.0 nM|> 110400.0 nM | | | NPASS |
| SK-MEL-2 | Homo sapiens | | | > 40.0 ug.mL-1|= 21470.0 nM|> 110400.0 nM | | | NPASS |
| RAW264.7 | Mus musculus | | | = 172000.0 nM|> 200000.0 nM|> 100000.0 nM|= 132000.0 nM | | | NPASS |
| NON-PROTEIN TARGET | | | = 60.2 ug.mL-1 | > 5.0 ug.mL-1|> 40.0 ug.mL-1 | | | NPASS |
| Matrix metalloproteinase-1 | Homo sapiens | P03956 | | = 50120.0 nM | | | NPASS |
| NCI-H187 | Homo sapiens | | | > 5.0 ug.mL-1 | | | NPASS |
| HT-1080 | Homo sapiens | | = 5.9 ug.mL-1 | | | | NPASS |
| HCT-15 | Homo sapiens | | | > 110400.0 nM | | | NPASS |
| Cytochrome P450 3A4 | Homo sapiens | P08684 | | 47300 nM|= 47300.0 nM | | | BindingDB, NPASS |
| Cytochrome P450 2D6 | Homo sapiens | P10635 | | >100000 nM|> 100000.0 nM | | | BindingDB, NPASS |
| BV-2 | Mus musculus | | | = 87620.0 nM | | | NPASS |
| B16-F10 | Mus musculus | | | > 110400.0 nM | | | NPASS |
| A549 | Homo sapiens | | | > 40.0 ug.mL-1|> 30000.0 nM|> 110400.0 nM | | | NPASS |
| KB | Homo sapiens | | | > 5.0 ug.mL-1 | | | NPASS |