| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Muscarinic acetylcholine receptor M3 | Rattus norvegicus | P08483 | | | | 5700 nM|= 5700.0 nM | BindingDB, NPASS |
| Muscarinic acetylcholine receptor M4 | Homo sapiens | P08173 | 130 nM|= 130.0 nM | 13500 nM|47500 nM|= 13500.0 nM|= 47500.0 nM | | 2400 nM|26 nM|60000 nM|= 2400.0 nM|= 26.0 nM|= 60000.0 nM | BindingDB, NPASS |
| Muscarinic acetylcholine receptor M4 | Rattus norvegicus | P08485 | | | | 2400 nM|= 2400.0 nM | BindingDB, NPASS |
| Muscarinic acetylcholine receptor M5 | Homo sapiens | P08912 | 600 nM|= 600.0 nM | 62500 nM|= 62500.0 nM | | 56000 nM|56234 nM|= 56000.0 nM|= 56234.13 nM | BindingDB, NPASS |
| Muscarinic acetylcholine receptors; M2 & M3 | Homo sapiens | P08172 | = 140.0 nM | | | | NPASS |
| Neuronal acetylcholine receptor | Rattus norvegicus | Q05941 | | | | = 224.0 nM | NPASS |
| Reverse transcriptase | Human immunodeficiency virus 1 | | | >1280000 nM | | | BindingDB |
| Neuronal acetylcholine receptor; alpha4/beta2 | Rattus norvegicus | P12390 | | | | = 270.0 nM | NPASS |
| Nicotinic acetylcholine receptor alpha 5 subunit | Musca domestica | A9XFY4 | | | | = 516000.0 nM | NPASS |
| Oryctolagus cuniculus | Oryctolagus cuniculus | | | = 545.0 nM | | | NPASS |
| SARS-CoV-2 | Severe acute respiratory syndrome coronavirus 2 | | | > 20000.0 nM|> 19952.62 nM | | | NPASS |
| Muscarinic acetylcholine receptor M3 | Mus musculus | Q9ERZ3 | 12000 nM|= 12000.0 nM | | | | BindingDB, NPASS |
| Neuronal acetylcholine receptor subunit alpha-4/beta-2 | Rattus norvegicus | P09483|P12390 | | | | 270 nM | BindingDB |
| Muscarinic acetylcholine receptor M3 | Homo sapiens | P20309 | 100 nM|340 nM|= 340.0 nM|= 100.0 nM | 11000 nM|58000 nM|= 11000.0 nM|= 58000.0 nM | | 43000 nM|5700 nM|= 43000.0 nM|= 5700.0 nM | BindingDB, NPASS |
| Voltage-dependent L-type calcium channel subunit alpha-1C | Cavia porcellus | O35505 | | = 33730.0 nM | | | NPASS |
| Muscarinic acetylcholine receptor M2 | Homo sapiens | P08172 | 25 nM|83 nM|10000 nM|= 83.0 nM|= 25.0 nM|= 10000.0 nM | 1800 nM|4500 nM|= 1800.0 nM|= 4500.0 nM | | 40 nM|2400 nM|2455 nM|= 40.0 nM|= 2400.0 nM|= 2454.71 nM | BindingDB, NPASS |
| A9 | Mus musculus | | = 3080000.0 nM | = 1200.0 nM | | | NPASS |
| Bile salt export pump | Homo sapiens | O95342 | | >1000000 nM|> 1000000.0 nM | | | BindingDB, NPASS |
| Cavia porcellus | Cavia porcellus | | = 150.0 nM | = 600.0 nM|> 1000.0 nM | | | NPASS |
| Ion channel NompC | Danio rerio | | 29900 nM | | | | BindingDB |
| Mucolipin-3 | Homo sapiens | Q8TDD5 | 2260 nM | | | | BindingDB |
| Muscarinic acetylcholine receptor | Homo sapiens | P08912 | = 73.0 nM | | | | NPASS |
| Muscarinic acetylcholine receptor M2 | Rattus norvegicus | P10980 | | 11000 nM|9150 nM|590 nM|= 11000.0 nM|= 590.0 nM|= 9150.0 nM | | 5270 nM|1000 nM|40 nM|= 40.0 nM | BindingDB, NPASS |
| Muscarinic acetylcholine receptor M1 | Homo sapiens | P11229 | 3200 nM|5603 nM|= 3200.0 nM|= 5603.0 nM | 545 nM|115 nM|115500 nM|65000 nM|145000 nM|= 115500.0 nM|= 115.0 nM|= 65000.0 nM|= 545.0 nM|= 145000.0 nM | | 4.1 nM|14 nM|29000 nM|29512 nM|= 14.0 nM|= 29000.0 nM|= 29512.09 nM | BindingDB, NPASS |
| Muscarinic acetylcholine receptor M1 | Mus musculus | P12657 | 27000 nM|= 27000.0 nM | | | 5.5 nM|3.3 nM|= 3.33 nM|= 5.45 nM | BindingDB, NPASS |
| Muscarinic acetylcholine receptor M1 | Rattus norvegicus | P08482 | >= 220.0 nM | 77 nM|1300 nM|1740 nM|469000 nM|11920 nM|460000 nM|1100 nM|1738 nM|= 1740.0 nM|= 77.0 nM|= 1300.0 nM|= 1100.0 nM|= 1737.8 nM|= 11920.0 nM|= 469000.0 nM|= 460000.0 nM | | 5950 nM|86000 nM|88000 nM|= 86000.0 nM|= 88000.0 nM | BindingDB, NPASS |
| Muscarinic acetylcholine receptor M1/M2/M3/M4/M5 | Homo sapiens | P08172|P08173|P08912|P11229|P20309 | 73 nM | | | | BindingDB |
| Muscarinic acetylcholine receptor M1/M2/M3/M4/M5 | Rattus norvegicus | P08482|P08483|P08485|P08911|P10980 | | 20 nM|5600 nM|1000 nM|77 nM|24 nM|1.9 nM|106000 nM|115 nM|25400 nM|120 nM|25000 nM | | 40 nM|7120 nM | BindingDB |
| Muscarinic acetylcholine receptor | Rattus norvegicus | P10980 | | = 20.0 nM|= 1000.0 nM|= 28000.0 nM|= 1700.0 nM|= 2100.0 nM|= 16.0 nM|= 24.0 nM|= 115.0 nM|= 25400.0 nM|= 1.9 nM|= 5600.0 nM|= 77.0 nM|= 19000.0 nM|= 106000.0 nM|= 62.7 nM|= 120.0 nM|= 25000.0 nM | | = 40.0 nM|= 31.0 nM|= 1900.0 nM|= 5.3 nM|= 7120.0 nM | NPASS |