| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Sodium- and chloride-dependent GABA transporter 1 | Mus musculus | P31648 | | 12500 nM | | | BindingDB |
| Sodium- and chloride-dependent GABA transporter 1 | Rattus norvegicus | P23978 | | 20900 nM|2770 nM|2590 nM|2660 nM|2900 nM|1680 nM|2650 nM|2790 nM | | | BindingDB |
| Sodium- and chloride-dependent GABA transporter 2 | Homo sapiens | Q9NSD5 | | 66000 nM | | | BindingDB |
| Sodium- and chloride-dependent GABA transporter 2 | Mus musculus | P31649 | | 72400 nM | | | BindingDB |
| Sodium- and chloride-dependent betaine transporter | Homo sapiens | P48065 | | 1870000 nM | | | BindingDB |
| Sodium- and chloride-dependent GABA transporter 3 | Homo sapiens | P48066 | | 119000 nM|110000 nM | | | BindingDB |
| Sodium- and chloride-dependent GABA transporter 3 | Mus musculus | P31650 | | 114800 nM | | | BindingDB |
| Sodium- and chloride-dependent betaine transporter | Mus musculus | P31651 | | >1000000 nM | | | BindingDB |
| Sodium- and chloride-dependent GABA transporter 1 | Homo sapiens | P30531 | | 14000 nM | | | BindingDB |
| Sodium- and chloride-dependent GABA transporter 2 | Rattus norvegicus | P31646 | | 58000 nM | | | BindingDB |
| Rattus norvegicus | Rattus norvegicus | | | = 4920.0 nM|= 7300.0 nM|= 12000.0 nM | | | NPASS |
| GABA transporter 3 | Mus musculus | P31649 | | = 25703.96 nM|= 72400.0 nM | | | NPASS |
| GABA transporter 4 | Mus musculus | P31650 | | = 25703.96 nM|= 114800.0 nM | | | NPASS |
| GABA transporter 3 | Homo sapiens | P48066 | | = 119000.0 nM|= 110000.0 nM | | | NPASS |
| GABA transporter 2 | Rattus norvegicus | P31646 | | = 58000.0 nM | | | NPASS |
| GABA transporter 2 | Mus musculus | P31651 | | = 489778.82 nM|> 1000000.0 nM | | | NPASS |
| GABA transporter 2 | Homo sapiens | Q9NSD5 | | = 66000.0 nM | | | NPASS |
| GABA transporter 1 | Rattus norvegicus | P23978 | | = 2650.0 nM|= 1680.0 nM|= 2900.0 nM|= 2260.0 nM|= 2660.0 nM|= 1760.0 nM|= 1870.0 nM|= 2790.0 nM|= 1910.0 nM|= 2770.0 nM|= 1850.0 nM|= 2590.0 nM|= 2560.0 nM | | | NPASS |
| GABA transporter 1 | Mus musculus | P31648 | | = 13489.63 nM|= 12589.25 nM|= 14000.0 nM|= 20900.0 nM | | | NPASS |
| GABA transporter 1 | Homo sapiens | P30531 | | = 14000.0 nM | | | NPASS |
| Corticotropin-releasing factor-binding protein | Homo sapiens | P24387 | >53000 nM | | | | BindingDB |
| Betaine transporter | Homo sapiens | P48065 | | = 1870000.0 nM | | | NPASS |
| Mus musculus | Mus musculus | | | = 32000.0 nM|= 29000.0 nM | | | NPASS |
