IMPPAT Phytochemical information: 
Codeine

Codeine
Bioactivity information
Target nameTarget organismUniProt identifierEC50IC50KdKiSource
Solute carrier family 22 member 1Homo sapiensO15245235500 nM|= 235500.0 nMBindingDB, NPASS
Rattus norvegicusRattus norvegicus= 2600.0 nM|= 22000.0 nMNPASS
Potassium voltage-gated channel subfamily H member 2Homo sapiensQ12809301995.17 nMBindingDB
Opioid receptorMus musculusP33534= 10000.0 nMNPASS
Mu-type opioid receptorHomo sapiensP35372105 nMBindingDB
Mu opioid receptorHomo sapiensP35372= 6100.0 nM= 105.0 nM= 6300.0 nM|= 727.0 nMNPASS
Mas-related G-protein coupled receptor member X2HumanQ96LB11.0e+4 nM|6.8e+3 nMBindingDB
Kappa-type opioid receptorHomo sapiensP4114515000 nMBindingDB
HERGHomo sapiensQ12809= 301995.17 nMNPASS
Delta-type/Kappa-type/Mu-type opioid receptorRattus norvegicusP33533|P33535|P34975800000 nMBindingDB
Kappa opioid receptorHomo sapiensP41145= 15000.0 nM= 25411.0 nMNPASS
Delta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1Mus musculusO55242|P32300|P33534|P4286610000 nMBindingDB
Delta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1Rattus norvegicusP33533|P33535|P34975|Q9R0C910.0 nMBindingDB
Cytochrome P450 2D18Rattus norvegicusQ64680= 2216000.0 nMNPASS
Cytochrome P450 2D2Rattus norvegicusP10634= 238000.0 nMNPASS
Cytochrome P450 2D26Rattus norvegicusP10634238000 nMBindingDB
Cytochrome P450 2D1Rattus norvegicusP106331320000 nM|= 1320000.0 nMBindingDB, NPASS
Cytochrome P450 2D4Rattus norvegicusQ646802216000 nMBindingDB
Cytochrome P450 2D6Homo sapiensP10635104000 nM|= 104000.0 nMBindingDB, NPASS
Delta opioid receptorHomo sapiensP41143> 9300.0 nM= 52207.0 nMNPASS
Delta-type opioid receptorHomo sapiensP41143>9300 nMBindingDB
Cytochrome P450 2D3Rattus norvegicusP129384089000 nM|= 4089000.0 nMBindingDB, NPASS