| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Solute carrier family 22 member 1 | Homo sapiens | O15245 | | 235500 nM|= 235500.0 nM | | | BindingDB, NPASS |
| Rattus norvegicus | Rattus norvegicus | | | = 2600.0 nM|= 22000.0 nM | | | NPASS |
| Potassium voltage-gated channel subfamily H member 2 | Homo sapiens | Q12809 | | 301995.17 nM | | | BindingDB |
| Opioid receptor | Mus musculus | P33534 | | = 10000.0 nM | | | NPASS |
| Mu-type opioid receptor | Homo sapiens | P35372 | | 105 nM | | | BindingDB |
| Mu opioid receptor | Homo sapiens | P35372 | = 6100.0 nM | = 105.0 nM | | = 6300.0 nM|= 727.0 nM | NPASS |
| Mas-related G-protein coupled receptor member X2 | Human | Q96LB1 | 1.0e+4 nM|6.8e+3 nM | | | | BindingDB |
| Kappa-type opioid receptor | Homo sapiens | P41145 | | 15000 nM | | | BindingDB |
| HERG | Homo sapiens | Q12809 | | = 301995.17 nM | | | NPASS |
| Delta-type/Kappa-type/Mu-type opioid receptor | Rattus norvegicus | P33533|P33535|P34975 | 800000 nM | | | | BindingDB |
| Kappa opioid receptor | Homo sapiens | P41145 | | = 15000.0 nM | | = 25411.0 nM | NPASS |
| Delta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1 | Mus musculus | O55242|P32300|P33534|P42866 | | 10000 nM | | | BindingDB |
| Delta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1 | Rattus norvegicus | P33533|P33535|P34975|Q9R0C9 | | 10.0 nM | | | BindingDB |
| Cytochrome P450 2D18 | Rattus norvegicus | Q64680 | | = 2216000.0 nM | | | NPASS |
| Cytochrome P450 2D2 | Rattus norvegicus | P10634 | | = 238000.0 nM | | | NPASS |
| Cytochrome P450 2D26 | Rattus norvegicus | P10634 | | 238000 nM | | | BindingDB |
| Cytochrome P450 2D1 | Rattus norvegicus | P10633 | | 1320000 nM|= 1320000.0 nM | | | BindingDB, NPASS |
| Cytochrome P450 2D4 | Rattus norvegicus | Q64680 | | 2216000 nM | | | BindingDB |
| Cytochrome P450 2D6 | Homo sapiens | P10635 | | 104000 nM|= 104000.0 nM | | | BindingDB, NPASS |
| Delta opioid receptor | Homo sapiens | P41143 | | > 9300.0 nM | | = 52207.0 nM | NPASS |
| Delta-type opioid receptor | Homo sapiens | P41143 | | >9300 nM | | | BindingDB |
| Cytochrome P450 2D3 | Rattus norvegicus | P12938 | | 4089000 nM|= 4089000.0 nM | | | BindingDB, NPASS |