| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| SARS-CoV-2 | Severe acute respiratory syndrome coronavirus 2 | | | > 20000.0 nM|> 19952.62 nM | | | NPASS |
| Sodium channel protein type 1/2/3 subunit alpha | Homo sapiens | P35498|Q99250|Q9NY46 | | 21000 nM | | | BindingDB |
| Sodium channel alpha subunits; brain (Types I, II, III) | Homo sapiens | Q9NY46 | | = 21000.0 nM | | | NPASS |
| SW480 | Homo sapiens | | | > 40000.0 nM | | | NPASS |
| SMMC-7721 | Homo sapiens | | | > 40000.0 nM | | | NPASS |
| MCF7 | Homo sapiens | | | > 40000.0 nM | | | NPASS |
| Glycine receptor | Rattus norvegicus | P20781 | | = 8.295 nM | | = 4.689 nM | NPASS |
| Glycine receptor subunit alpha-1/beta | Homo sapiens | P23415|P48167 | | 180 nM|182 nM|58 nM|510 nM|513 nM|60 nM | | | BindingDB |
| Glycine receptor subunit alpha-1 | Rattus norvegicus | P07727 | | | | 12 nM|= 12.0 nM | BindingDB, NPASS |
| Glycine receptor subunit alpha-1 | Homo sapiens | P23415 | | 51 nM|93 nM|150 nM|151 nM|50 nM|134 nM|27 nM|= 93.33 nM|= 93.0 nM|= 51.0 nM|= 151.36 nM|= 150.0 nM|= 27.0 nM|= 134.0 nM|= 50.0 nM | | 23 nM|123 nM|5.0 nM|= 23.0 nM|= 123.0 nM|= 5.0 nM | BindingDB, NPASS |
| Glycine receptor (alpha-1/beta) | Homo sapiens | | | = 181.97 nM|= 180.0 nM|= 58.0 nM|= 512.86 nM|= 510.0 nM|= 60.0 nM | | | NPASS |
| A549 | Homo sapiens | | | > 40000.0 nM | | | NPASS |
| HL-60 | Homo sapiens | | | > 40000.0 nM | | | NPASS |