| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| OVCAR-3 | Homo sapiens | | | = 1400.0 nM|= 1600.0 nM|= 1700.0 nM | | | NPASS |
| Plasmodium falciparum | Plasmodium falciparum | | | = 230.0 nM | | | NPASS |
| SK-LU-1 | Homo sapiens | | | = 210.0 nM | | | NPASS |
| SW872 | Homo sapiens | | | = 1400.0 nM|= 1200.0 nM | | | NPASS |
| Telomerase reverse transcriptase | Homo sapiens | O14746 | | = 4000.0 nM | | | NPASS |
| X-box-binding protein 1 | Homo sapiens | P17861 | | 2140 nM|= 2430.0 nM | | | BindingDB, NPASS |
| Type-1 angiotensin II receptor | Homo sapiens | P30556 | | 18639 nM|= 18639.0 nM | | | BindingDB, NPASS |
| ZR-75-1 | Homo sapiens | | | = 700.0 nM|= 800.0 nM|= 1100.0 nM | | | NPASS |
| p53-binding protein Mdm-2 | Homo sapiens | Q00987 | = 420.0 nM | | | | NPASS |
| NON-PROTEIN TARGET | | | | = 2400.0 nM|= 390.0 nM|= 1300.0 nM|= 900.0 nM|= 500.0 nM|= 1200.0 nM|= 700.0 nM|= 270.0 nM | | | NPASS |
| Transcriptional activator Myb | Gallus gallus | P01103 | | 2371 nM|2370 nM|= 2371.37 nM|= 2370.0 nM | | | BindingDB, NPASS |
| MCF7 | Homo sapiens | | | = 800.0 nM|= 500.0 nM|= 700.0 nM | | | NPASS |
| Platelet | | | | = 4280.0 nM | | | NPASS |
| Jurkat | Homo sapiens | | | = 0.03 ug.mL-1|= 460.0 nM|= 1020.0 nM | | | NPASS |
| HeLa | Homo sapiens | | = 700.0 nM | | | | NPASS |
| HL-60 | Homo sapiens | | | = 320.0 nM|= 700.0 nM | | | NPASS |
| HEp-2 | Homo sapiens | | | = 900.0 nM|= 800.0 nM | | | NPASS |
| HCT-15 | Homo sapiens | | | = 290.0 nM | | | NPASS |
| G-protein coupled receptor 55 | Homo sapiens | Q9Y2T6 | | 2642.275 nM|= 2642.28 nM | | | BindingDB, NPASS |
| E3 ubiquitin-protein ligase Mdm2 | Homo sapiens | Q00987 | 420 nM|1110 nM|180 nM | | | | BindingDB |
| DNA damage-inducible transcript 3 protein | Mus musculus | P35639 | | 2450 nM|= 2610.0 nM | | | BindingDB, NPASS |
| Beta-galactosidase | Escherichia coli | Q8VNN2 | > 40000.0 nM | | | | NPASS |
| Apelin receptor | Homo sapiens | P35414 | | 21300 nM | | | BindingDB |
| A-431 | Homo sapiens | | | = 900.0 nM|= 800.0 nM | | | NPASS |
| K562 | Homo sapiens | | | = 280.0 nM | | | NPASS |