| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|
| Raji | Homo sapiens | | | = 20.0 nM | | | NPASS |
| PANC-1 | Homo sapiens | | | > 10000.0 nM | | | NPASS |
| Neurogenic locus notch homolog protein 1 | Homo sapiens | P46531 | | 800 nM|= 800.0 nM | | | BindingDB, NPASS |
| NON-PROTEIN TARGET | | | | = 41.3 nM | | | NPASS |
| MDA-MB-231 | Homo sapiens | | | = 0.16 ug.mL-1|= 440.0 nM | | | NPASS |
| MCF7 | Homo sapiens | | | = 0.08 ug.mL-1 | | | NPASS |
| NCI-H187 | Homo sapiens | | | = 471.0 nM | | | NPASS |
| Hs-578T | Homo sapiens | | | = 60.0 nM | | | NPASS |
| HepG2 | Homo sapiens | | | = 40.0 nM|= 0.11 ug.mL-1 | | | NPASS |
| HeLa | Homo sapiens | | | > 10000.0 nM | | | NPASS |
| DU-145 | Homo sapiens | | | = 30.0 nM | | | NPASS |
| BT-549 | Homo sapiens | | | = 30.0 nM | | | NPASS |
| A549 | Homo sapiens | | | = 0.02 ug.mL-1 | | | NPASS |
| KB | Homo sapiens | | | = 0.015 ug.mL-1|= 62.0 nM | | | NPASS |