IMPPAT Phytochemical information: 
Calotropin

Calotropin
Bioactivity information
Target nameTarget organismUniProt identifierEC50IC50KdKiSource
RajiHomo sapiens= 20.0 nMNPASS
PANC-1Homo sapiens> 10000.0 nMNPASS
Neurogenic locus notch homolog protein 1Homo sapiensP46531800 nM|= 800.0 nMBindingDB, NPASS
NON-PROTEIN TARGET= 41.3 nMNPASS
MDA-MB-231Homo sapiens= 0.16 ug.mL-1|= 440.0 nMNPASS
MCF7Homo sapiens= 0.08 ug.mL-1NPASS
NCI-H187Homo sapiens= 471.0 nMNPASS
Hs-578THomo sapiens= 60.0 nMNPASS
HepG2Homo sapiens= 40.0 nM|= 0.11 ug.mL-1NPASS
HeLaHomo sapiens> 10000.0 nMNPASS
DU-145Homo sapiens= 30.0 nMNPASS
BT-549Homo sapiens= 30.0 nMNPASS
A549Homo sapiens= 0.02 ug.mL-1NPASS
KBHomo sapiens= 0.015 ug.mL-1|= 62.0 nMNPASS