
| Target name | Target organism | UniProt identifier | EC50 | IC50 | Kd | Ki | Source |
|---|---|---|---|---|---|---|---|
| Neurogenic locus notch homolog protein 1 | Homo sapiens | P46531 | 400 nM|= 400.0 nM | BindingDB, NPASS | |||
| Hs-578T | Homo sapiens | = 34.0 nM | NPASS | ||||
| MDA-MB-231 | Homo sapiens | = 0.1 ug.mL-1|= 102.0 nM | NPASS | ||||
| MCF7 | Homo sapiens | = 0.04 ug.mL-1 | NPASS | ||||
| HepG2 | Homo sapiens | = 1.1 ug.mL-1 | NPASS | ||||
| BT-549 | Homo sapiens | = 14.6 nM | NPASS | ||||
| A549 | Homo sapiens | = 0.01 ug.mL-1|= 104.0 nM | NPASS | ||||
| HeLa | Homo sapiens | = 275.0 nM | NPASS |